DE2965513D1 - Process for producing alpha-aminophosphonic acids and their peptides and compounds thus obtained - Google Patents

Process for producing alpha-aminophosphonic acids and their peptides and compounds thus obtained

Info

Publication number
DE2965513D1
DE2965513D1 DE7979302080T DE2965513T DE2965513D1 DE 2965513 D1 DE2965513 D1 DE 2965513D1 DE 7979302080 T DE7979302080 T DE 7979302080T DE 2965513 T DE2965513 T DE 2965513T DE 2965513 D1 DE2965513 D1 DE 2965513D1
Authority
DE
Germany
Prior art keywords
peptides
compounds
producing alpha
aminophosphonic acids
aminophosphonic
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE7979302080T
Other languages
English (en)
Inventor
Eric Keith Baylis
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Novartis AG
Original Assignee
Ciba Geigy AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Ciba Geigy AG filed Critical Ciba Geigy AG
Application granted granted Critical
Publication of DE2965513D1 publication Critical patent/DE2965513D1/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
    • C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
    • C07F9/3808—Acyclic saturated acids which can have further substituents on alkyl
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/08—Tripeptides
    • C07K5/0827—Tripeptides containing heteroatoms different from O, S, or N
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Communicable Diseases (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Peptides Or Proteins (AREA)
DE7979302080T 1978-10-05 1979-10-02 Process for producing alpha-aminophosphonic acids and their peptides and compounds thus obtained Expired DE2965513D1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB7839399 1978-10-05

Publications (1)

Publication Number Publication Date
DE2965513D1 true DE2965513D1 (en) 1983-07-07

Family

ID=10500133

Family Applications (1)

Application Number Title Priority Date Filing Date
DE7979302080T Expired DE2965513D1 (en) 1978-10-05 1979-10-02 Process for producing alpha-aminophosphonic acids and their peptides and compounds thus obtained

Country Status (4)

Country Link
US (1) US4331591A (de)
EP (1) EP0010872B1 (de)
JP (1) JPS5589291A (de)
DE (1) DE2965513D1 (de)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0026867A1 (de) * 1979-09-28 1981-04-15 F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft Peptidylphosphonsäuren, deren Herstellung und Verwendung und sie enthaltende pharmazeutische Präparate
JPS57156498A (en) * 1981-03-20 1982-09-27 Kyowa Hakko Kogyo Co Ltd Novel physiologically active substance k-26
JPS5831992A (ja) * 1981-08-19 1983-02-24 Kyowa Hakko Kogyo Co Ltd 新規生理活性物質ｋ−４およびその製造法
EP0103867B1 (de) * 1982-09-17 1986-12-17 Kyowa Hakko Kogyo Co., Ltd. Phosphor enthaltendes Peptidderivat
PT77368A (en) * 1982-09-27 1983-10-01 Lilly Co Eli Improved process for preparing immunomodulating agents or rela-ting there to
US4463092A (en) * 1982-09-27 1984-07-31 Eli Lilly And Company Process for production antibiotic A53868
US4482488A (en) * 1982-09-27 1984-11-13 Eli Lilly And Company Antibiotic A53868 and process for production thereof
US4605522A (en) * 1983-05-27 1986-08-12 Stauffer Chemical Company Method for preparation of N-phosphonomethylglycine or salts
US4510169A (en) * 1983-08-23 1985-04-09 The Board Of Regents, The University Of Texas Method and apparatus for cryopreparing biological tissue for ultrastructural analysis
US5024830A (en) * 1983-08-23 1991-06-18 The Board Of Regents, The University Of Texas Method for cryopreparing biological tissue for ultrastructural analysis
US4745771A (en) * 1983-08-23 1988-05-24 Board Of Regents, The University Of Texas System Apparatus and method for cryopreparing biological tissue for ultrastructural analysis
US4799361A (en) * 1983-08-23 1989-01-24 Board Of Regents, The University Of Texas System Method for cryopreparing biological tissue for ultrastructural analysis
US4676070A (en) * 1984-11-30 1987-06-30 The Board Of Regents, The University Of Texas Apparatus and method for cryopreparing biological tissue
US4742690A (en) * 1983-08-23 1988-05-10 Board Of Regents, The University Of Texas System Apparatus and method for cryopreparing biological tissue for ultrastructural analysis
US4567847A (en) * 1983-08-23 1986-02-04 Board Of Regents, The University Of Texas System Apparatus and method for cryopreparing biological tissue for ultrastructural analysis
US5189030A (en) * 1985-06-11 1993-02-23 Ciba-Geigy Corporation 1-amino-2-phenylethanephosphonic acids as microbiocides
DE3544376A1 (de) * 1985-12-14 1987-06-19 Hoechst Ag Dipeptide mit c-terminalem phosphinothricin, verfahren zu ihrer herstellung und ihre verwendung zur bekaempfung unerwuenschten pflanzenwuchses
US4670193A (en) * 1986-05-12 1987-06-02 E. R. Squibb & Sons, Inc. Process for preparing phosphonic acids
US5044165A (en) * 1986-12-03 1991-09-03 Board Of Regents, The University Of Texas Cryo-slammer
GB8726714D0 (en) * 1987-11-14 1987-12-16 Beecham Group Plc Compounds
US5179173A (en) * 1991-04-10 1993-01-12 Nalco Chemical Company Aminoalkylphosphinates and phosphinic acid-containing polymers therefrom

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2899454A (en) * 1959-08-11 Ochzgfj
US2899455A (en) * 1959-08-11 O oxch
US2952699A (en) * 1955-12-23 1960-09-13 Lubrizol Corp Preparation of substituted phosphoric acids
NL135596C (de) * 1961-02-20
US3277217A (en) * 1963-04-24 1966-10-04 Gen Aniline & Film Corp Process for producing phosphate esters by oxidation of phosphites using hydrogen peroxide and organic peroxides as catalyst
NL124637C (de) * 1963-08-16
DE2331187A1 (de) * 1973-06-19 1975-01-09 Bayer Ag Mittel zur regulierung des pflanzenwachstums
IL48835A (en) * 1975-01-27 1979-05-31 Sparamedica Ag Amino acyl and peptidyl derivatives of phophonic acids, their preparation and pharmaceutical compositions containingthem
FR2351125A1 (fr) * 1976-05-14 1977-12-09 Hoffmann La Roche Derives peptidiques et procede pour leur preparation
US4028403A (en) * 1976-06-07 1977-06-07 Burlington Industries, Inc. Process for preparing m-aminobenzenephosphonic acid

Also Published As

Publication number Publication date
EP0010872B1 (de) 1983-05-25
US4331591A (en) 1982-05-25
EP0010872A1 (de) 1980-05-14
JPS5589291A (en) 1980-07-05

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Legal Events

Date Code Title Description
8339 Ceased/non-payment of the annual fee