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DE1922702A1 - A process for the preparation of 1-glycosyl-5-azacytosinen - Google Patents

A process for the preparation of 1-glycosyl-5-azacytosinen

Info

Publication number
DE1922702A1
DE1922702A1 DE19691922702 DE1922702A DE1922702A1 DE 1922702 A1 DE1922702 A1 DE 1922702A1 DE 19691922702 DE19691922702 DE 19691922702 DE 1922702 A DE1922702 A DE 1922702A DE 1922702 A1 DE1922702 A1 DE 1922702A1
Authority
DE
Grant status
Application
Patent type
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19691922702
Other languages
German (de)
Inventor
Frantisek Sorm
Alois Piskala
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Akademie Ved Ceske Republiky (The Cezch Academy of Science)
Original Assignee
Akademie Ved Ceske Republiky (The Cezch Academy of Science)
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/02Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing nitrogen
    • C07H19/04Heterocyclic radicals containing only nitrogen atoms as ring hetero atom
    • C07H19/12Triazine radicals
DE19691922702 1968-05-08 1969-05-03 A process for the preparation of 1-glycosyl-5-azacytosinen Pending DE1922702A1 (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
CS339968 1968-05-08

Publications (1)

Publication Number Publication Date
DE1922702A1 true true DE1922702A1 (en) 1969-11-20

Family

ID=5373920

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19691922702 Pending DE1922702A1 (en) 1968-05-08 1969-05-03 A process for the preparation of 1-glycosyl-5-azacytosinen

Country Status (8)

Country Link
JP (1) JPS4916435B1 (en)
BE (1) BE732268A (en)
CA (1) CA921904A (en)
DE (1) DE1922702A1 (en)
ES (1) ES366910A1 (en)
FR (1) FR2008048A1 (en)
GB (1) GB1227691A (en)
NL (1) NL6906909A (en)

Cited By (14)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6887855B2 (en) 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US6943249B2 (en) 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US7038038B2 (en) 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
US7135464B2 (en) 2002-06-05 2006-11-14 Supergen, Inc. Method of administering decitabine
US7250416B2 (en) 2005-03-11 2007-07-31 Supergen, Inc. Azacytosine analogs and derivatives
US7276228B2 (en) 2001-04-24 2007-10-02 Supergen, Inc. Methods for treating hematological disorders through inhibition of DNA methylation and histone deacetylase
WO2008044041A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
WO2008044045A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
US7700567B2 (en) 2005-09-29 2010-04-20 Supergen, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
US8212021B2 (en) 2008-08-08 2012-07-03 Scinopharm Taiwan, Ltd. Process for making 5-azacytosine nucleosides and their derivatives
US9381207B2 (en) 2011-08-30 2016-07-05 Astex Pharmaceuticals, Inc. Drug formulations
WO2017090275A1 (en) 2015-11-27 2017-06-01 大原薬品工業株式会社 5'-position dibenzyl phosphoric acid ester of 5-azacytidine or 2'-deoxy body thereof
WO2017183217A1 (en) 2016-04-21 2017-10-26 大原薬品工業株式会社 Sugar moiety silyl ether derivative of 5-azacytidine
US9901641B2 (en) 2016-04-21 2018-02-27 Ohara Pharmaceutical Co., Ltd. Silyl etherified derivatives of 5-azacytidines in carbohydrate moiety

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2012888C3 (en) * 1970-03-14 1981-04-02 Schering Ag, 1000 Berlin Und 4619 Bergkamen, De
US20060014949A1 (en) * 2004-07-13 2006-01-19 Supergen Inc. Compositions and formulations of decitabine polymorphs and methods of use thereof
JP2011520880A (en) 2008-05-15 2011-07-21 セルジーン コーポレイション Oral formulations and methods of use thereof for cytidine analog

Cited By (32)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7276228B2 (en) 2001-04-24 2007-10-02 Supergen, Inc. Methods for treating hematological disorders through inhibition of DNA methylation and histone deacetylase
US7135464B2 (en) 2002-06-05 2006-11-14 Supergen, Inc. Method of administering decitabine
US7144873B2 (en) 2002-06-05 2006-12-05 Supergen, Inc. Kit for delivering decitabine in vivo
US8513406B2 (en) 2003-03-17 2013-08-20 Pharmion Llc Pharmaceutical compositions comprising forms of 5-azacytidine
US7078518B2 (en) 2003-03-17 2006-07-18 Pharmion Corporation Forms of 5-Azacytidine
US7038038B2 (en) 2003-03-17 2006-05-02 Pharmion Corporation Synthesis of 5-azacytidine
US8614313B2 (en) 2003-03-17 2013-12-24 Pharmion Llc Pharmaceutical compositions comprising forms of 5-azacytidine
US6943249B2 (en) 2003-03-17 2005-09-13 Ash Stevens, Inc. Methods for isolating crystalline Form I of 5-azacytidine
US9192620B2 (en) 2003-03-17 2015-11-24 Pharmion Llc Pharmaceutical compositions comprising forms of 5-azacytidine
US8975392B2 (en) 2003-03-17 2015-03-10 Pharmion Llc Methods for isolating crystalline form I of 5-azacytidine
US8779117B2 (en) 2003-03-17 2014-07-15 Pharmion Llc Pharmaceutical compositions comprising 5-azacytidine monohydrate
US7700770B2 (en) 2003-03-17 2010-04-20 Celgene Corporation Methods for isolating crystalline form I of 5-azacytidine
US7772199B2 (en) 2003-03-17 2010-08-10 Celgene Corporation Forms of 5-azacytidine
US7858774B2 (en) 2003-03-17 2010-12-28 Pharmion Llc Synthesis of 5-azacytidine
US8058424B2 (en) 2003-03-17 2011-11-15 Pharmion Llc Synthesis of 5-azacytidine
US8211862B2 (en) 2003-03-17 2012-07-03 Pharmion Llc Pharmaceutical compositions comprising crystal forms of 5-azacytidine
US6887855B2 (en) 2003-03-17 2005-05-03 Pharmion Corporation Forms of 5-azacytidine
US8481715B2 (en) 2003-03-17 2013-07-09 Pharmion Llc Methods for isolating crystalline form I of 5-azacytidine
US7250416B2 (en) 2005-03-11 2007-07-31 Supergen, Inc. Azacytosine analogs and derivatives
US9480698B2 (en) 2005-09-29 2016-11-01 Astex Pharmaceuticals, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
US8461123B2 (en) 2005-09-29 2013-06-11 Astex Pharmaceuticals, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
US7700567B2 (en) 2005-09-29 2010-04-20 Supergen, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
US9358248B2 (en) 2005-09-29 2016-06-07 Astex Pharmaceuticals, Inc. Oligonucleotide analogues incorporating 5-aza-cytosine therein
WO2008044045A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
WO2008044041A1 (en) 2006-10-12 2008-04-17 Astex Therapeutics Limited Pharmaceutical combinations
US8212021B2 (en) 2008-08-08 2012-07-03 Scinopharm Taiwan, Ltd. Process for making 5-azacytosine nucleosides and their derivatives
US9381207B2 (en) 2011-08-30 2016-07-05 Astex Pharmaceuticals, Inc. Drug formulations
US9913856B2 (en) 2011-08-30 2018-03-13 Astex Pharmaceuticals, Inc. Drug formulations
WO2017090275A1 (en) 2015-11-27 2017-06-01 大原薬品工業株式会社 5'-position dibenzyl phosphoric acid ester of 5-azacytidine or 2'-deoxy body thereof
US9670238B1 (en) 2015-11-27 2017-06-06 Ohara Pharmaceutical Co., Ltd. 5′-dibenzyl phosphates of 5-azacytidine or 2′-deoxy-5-azacytidine
WO2017183217A1 (en) 2016-04-21 2017-10-26 大原薬品工業株式会社 Sugar moiety silyl ether derivative of 5-azacytidine
US9901641B2 (en) 2016-04-21 2018-02-27 Ohara Pharmaceutical Co., Ltd. Silyl etherified derivatives of 5-azacytidines in carbohydrate moiety

Also Published As

Publication number Publication date Type
GB1227691A (en) 1971-04-07 application
ES366910A1 (en) 1971-03-16 application
CA921904A1 (en) grant
FR2008048A1 (en) 1970-01-16 application
CA921904A (en) 1973-02-27 grant
BE732268A (en) 1969-10-01 grant
JPS4916435B1 (en) 1974-04-22 grant
NL6906909A (en) 1969-11-11 application

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