DE102004004974A1 - Thieno-Iminosäure-Derivate als Inhibitoren von Matrix-Metalloproteinasen - Google Patents
Thieno-Iminosäure-Derivate als Inhibitoren von Matrix-Metalloproteinasen Download PDFInfo
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- DE102004004974A1 DE102004004974A1 DE102004004974A DE102004004974A DE102004004974A1 DE 102004004974 A1 DE102004004974 A1 DE 102004004974A1 DE 102004004974 A DE102004004974 A DE 102004004974A DE 102004004974 A DE102004004974 A DE 102004004974A DE 102004004974 A1 DE102004004974 A1 DE 102004004974A1
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- A—HUMAN NECESSITIES
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- A61P9/04—Inotropic agents, i.e. stimulants of cardiac contraction; Drugs for heart failure
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- A—HUMAN NECESSITIES
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Engineering & Computer Science (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Cardiology (AREA)
- Physical Education & Sports Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Rheumatology (AREA)
- Vascular Medicine (AREA)
- Urology & Nephrology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Oncology (AREA)
- Nutrition Science (AREA)
- Hematology (AREA)
- Immunology (AREA)
- Diabetes (AREA)
- Neurology (AREA)
- Dermatology (AREA)
- Biomedical Technology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
Priority Applications (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004004974A DE102004004974A1 (de) | 2004-01-31 | 2004-01-31 | Thieno-Iminosäure-Derivate als Inhibitoren von Matrix-Metalloproteinasen |
| JP2006550004A JP4733648B2 (ja) | 2004-01-31 | 2005-01-18 | マトリックスメタロプロテイナーゼ阻害剤としての使用のためのチエノ−イミノ酸誘導体 |
| EP05700992A EP1723148A2 (de) | 2004-01-31 | 2005-01-18 | Thieno-iminosaure-derivate als inhibitoren von matrix-metalloproteinasen |
| PCT/EP2005/000417 WO2005073236A2 (de) | 2004-01-31 | 2005-01-18 | Thieno-iminosäure-derivate als inhibitoren von matrix-metalloproteinasen |
| US11/461,189 US7399770B2 (en) | 2004-01-31 | 2006-07-31 | Thieno-imino acid derivatives for use as matrix metalloproteinase inhibitors |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE102004004974A DE102004004974A1 (de) | 2004-01-31 | 2004-01-31 | Thieno-Iminosäure-Derivate als Inhibitoren von Matrix-Metalloproteinasen |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE102004004974A1 true DE102004004974A1 (de) | 2005-08-18 |
Family
ID=34801393
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE102004004974A Withdrawn DE102004004974A1 (de) | 2004-01-31 | 2004-01-31 | Thieno-Iminosäure-Derivate als Inhibitoren von Matrix-Metalloproteinasen |
Country Status (5)
| Country | Link |
|---|---|
| US (1) | US7399770B2 (https=) |
| EP (1) | EP1723148A2 (https=) |
| JP (1) | JP4733648B2 (https=) |
| DE (1) | DE102004004974A1 (https=) |
| WO (1) | WO2005073236A2 (https=) |
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102005015040A1 (de) * | 2005-03-31 | 2006-10-05 | Sanofi-Aventis Deutschland Gmbh | Substituierte Tetrahydroisochinoline als MMP-Inhibitoren, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament |
| DE102004053982B4 (de) * | 2004-11-09 | 2011-07-21 | Koop, Daniel, 25337 | Verwendung von Reibhölzern und Verfahren zum Räuchern von Nahrungsmittelprodukten |
Families Citing this family (9)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE10361075A1 (de) * | 2003-12-22 | 2005-07-28 | Pac Tech - Packaging Technologies Gmbh | Verfahren und Vorichtung zur Trocknung von Schaltungssubstraten |
| SG10201510665WA (en) | 2009-12-04 | 2016-01-28 | Sunovion Pharmaceuticals Inc | Multicycle Compounds And Pharmaceutical Compositions Useful For The Treatment Of Neurological Disorders |
| MA45795A (fr) | 2016-07-29 | 2019-06-05 | Sunovion Pharmaceuticals Inc | Composés et compositions, et utilisations associées |
| PT3494119T (pt) | 2016-07-29 | 2024-12-10 | Pgi Drug Discovery Llc | Compostos e composições e seus usos |
| MX390141B (es) | 2017-02-16 | 2025-03-20 | Sunovion Pharmaceuticals Inc | Metodos para tratar esquizofrenia |
| CA3070993C (en) | 2017-08-02 | 2025-05-20 | Sunovion Pharmaceuticals Inc. | ISOCHROMANE COMPOUNDS AND THEIR USES |
| UA130249C2 (uk) | 2018-02-16 | 2025-12-31 | Сумітомо Фарма Америка, Інк. | Солі, кристалічні форми і способи їх отримання |
| EP3938045A1 (en) | 2019-03-14 | 2022-01-19 | Sunovion Pharmaceuticals Inc. | Salts of a isochromanyl compound and crystalline forms, processes for preparing, therapeutic uses, and pharmaceutical compositions thereof |
| CA3180115A1 (en) | 2020-04-14 | 2021-10-21 | Sunovion Pharmaceuticals Inc. | (s)-(4,5-dihydro-7h-thieno[2,3-c]pyran-7-yl)-n-methylmethanamine for treating neurological and psychiatric disorders |
Family Cites Families (13)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5294621A (en) | 1992-10-07 | 1994-03-15 | Ortho Pharmaceutical Corporation | Thieno tetrahydropyridines useful as class III antiarrhythmic agents |
| US5455258A (en) | 1993-01-06 | 1995-10-03 | Ciba-Geigy Corporation | Arylsulfonamido-substituted hydroxamic acids |
| AU7205894A (en) | 1993-06-08 | 1995-01-03 | Neogenix, Inc. | Purified natural and synthetic compounds for the treatment of osteoarthritis |
| US5863949A (en) | 1995-03-08 | 1999-01-26 | Pfizer Inc | Arylsulfonylamino hydroxamic acid derivatives |
| ES2153031T4 (es) * | 1995-04-20 | 2001-05-16 | Pfizer | Derivados del acido arilsulfonil hidroxamico como inhibidores de mmp y tnf. |
| US6207672B1 (en) | 1995-11-13 | 2001-03-27 | Aventis Pharma Deutschland Gmbh | Cyclic and heterocyclic N-substituted α-iminohydroxamic and carboxyclic acids |
| FR2748026B1 (fr) * | 1996-04-26 | 1998-06-05 | Adir | Nouveaux inhibiteurs de metalloproteases, leur procede de preparation et les compositions pharmaceutiques qui les contiennent |
| RU2203274C2 (ru) | 1996-08-28 | 2003-04-27 | Дзе Проктер Энд Гэмбл Компани | Спироциклические ингибиторы металлопротеаз |
| EP1003751A1 (en) * | 1997-08-04 | 2000-05-31 | Amgen Inc. | Hydroxamic acid substituted fused heterocyclic metalloproteinase inhibitors |
| FR2825705B1 (fr) | 2001-06-08 | 2005-05-20 | Aventis Pharma Sa | Nouveaux composes heterocycliques, leur preparation et leur utilisation comme medicaments, notamment comme anti-bacteriens |
| WO2003016248A2 (en) * | 2001-08-17 | 2003-02-27 | Bristol-Myers Squibb Company Patent Department | Bicyclic hydroxamates as inhibitors of matrix metalloproteinases and/or tnf-$g(a) converting enzyme (tace) |
| WO2003089416A1 (de) * | 2002-04-22 | 2003-10-30 | Ibfb Gmbh | Substituierte pyrimidin-2,4(1h,3h)-dione als matrix metalloproteinase (mmp) inhibitoren |
| CN1187332C (zh) * | 2002-04-26 | 2005-02-02 | 中国科学院上海有机化学研究所 | 四氢异喹啉羟肟酸磺酰胺类化合物、合成方法及其用途 |
-
2004
- 2004-01-31 DE DE102004004974A patent/DE102004004974A1/de not_active Withdrawn
-
2005
- 2005-01-18 EP EP05700992A patent/EP1723148A2/de not_active Withdrawn
- 2005-01-18 WO PCT/EP2005/000417 patent/WO2005073236A2/de not_active Ceased
- 2005-01-18 JP JP2006550004A patent/JP4733648B2/ja not_active Expired - Fee Related
-
2006
- 2006-07-31 US US11/461,189 patent/US7399770B2/en not_active Expired - Fee Related
Cited By (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE102004053982B4 (de) * | 2004-11-09 | 2011-07-21 | Koop, Daniel, 25337 | Verwendung von Reibhölzern und Verfahren zum Räuchern von Nahrungsmittelprodukten |
| DE102005015040A1 (de) * | 2005-03-31 | 2006-10-05 | Sanofi-Aventis Deutschland Gmbh | Substituierte Tetrahydroisochinoline als MMP-Inhibitoren, Verfahren zu ihrer Herstellung und ihre Verwendung als Medikament |
Also Published As
| Publication number | Publication date |
|---|---|
| WO2005073236A2 (de) | 2005-08-11 |
| WO2005073236A3 (de) | 2006-01-26 |
| JP4733648B2 (ja) | 2011-07-27 |
| EP1723148A2 (de) | 2006-11-22 |
| JP2007519654A (ja) | 2007-07-19 |
| US20070093482A1 (en) | 2007-04-26 |
| US7399770B2 (en) | 2008-07-15 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8127 | New person/name/address of the applicant |
Owner name: SANOFI-AVENTIS DEUTSCHLAND GMBH, 65929 FRANKFURT, |
|
| 8141 | Disposal/no request for examination | ||
| R005 | Application deemed withdrawn due to failure to request examination |
Effective date: 20110201 |