CY1124940T1 - Αλας διμεθυλαμινοαιθανολης ενος ρυθμιστη του υποδοχεα glp-1 - Google Patents

Αλας διμεθυλαμινοαιθανολης ενος ρυθμιστη του υποδοχεα glp-1

Info

Publication number
CY1124940T1
CY1124940T1 CY20211101089T CY211101089T CY1124940T1 CY 1124940 T1 CY1124940 T1 CY 1124940T1 CY 20211101089 T CY20211101089 T CY 20211101089T CY 211101089 T CY211101089 T CY 211101089T CY 1124940 T1 CY1124940 T1 CY 1124940T1
Authority
CY
Cyprus
Prior art keywords
glp
receptor regulator
dimethylaminoethanol salt
salt
dimethylaminoethanol
Prior art date
Application number
CY20211101089T
Other languages
English (en)
Inventor
Ephraim Vidal
Roger Bakale
Philip TURNBULL
David Moser
Andrew Robbins
Craig Grant
Original Assignee
Receptos Llc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Receptos Llc filed Critical Receptos Llc
Publication of CY1124940T1 publication Critical patent/CY1124940T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D409/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms
    • C07D409/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
    • C07B2200/00—Indexing scheme relating to specific properties of organic compounds
    • C07B2200/13—Crystalline forms, e.g. polymorphs

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Diabetes (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Obesity (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Κρυσταλλικό άλας 1-(2-(5-(tert-βουτυλο)-θειοφαινο-2-καρβοξαμιδο)-3-(4-(5-( 4'-αιθυλο-[1,1'-δι(κυκλοεξαν)]-3-εν-4-υλο)πυριμιδιν-2-υλο)φαινυλο)προπανοϋλο)αζετιδινο-3-καρβοξυλικού 2-υδροξυ-Ν,Ν-διμεθυλαιθαναμινίου και μέθοδοι που σχετίζονται με τη σύνθεση και τη θεραπευτική χρήση αυτού.
CY20211101089T 2016-09-30 2021-12-10 Αλας διμεθυλαμινοαιθανολης ενος ρυθμιστη του υποδοχεα glp-1 CY1124940T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US201662402565P 2016-09-30 2016-09-30
PCT/US2017/054298 WO2018064476A1 (en) 2016-09-30 2017-09-29 Dimethylaminoethanol salt of a glp-1 receptor modulator

Publications (1)

Publication Number Publication Date
CY1124940T1 true CY1124940T1 (el) 2023-01-05

Family

ID=60043396

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20211101089T CY1124940T1 (el) 2016-09-30 2021-12-10 Αλας διμεθυλαμινοαιθανολης ενος ρυθμιστη του υποδοχεα glp-1

Country Status (12)

Country Link
US (1) US11066395B2 (el)
EP (1) EP3519407B1 (el)
CY (1) CY1124940T1 (el)
ES (1) ES2901599T3 (el)
HR (1) HRP20211938T1 (el)
HU (1) HUE056805T2 (el)
LT (1) LT3519407T (el)
PL (1) PL3519407T3 (el)
PT (1) PT3519407T (el)
RS (1) RS62814B1 (el)
SI (1) SI3519407T1 (el)
WO (1) WO2018064476A1 (el)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN113166056A (zh) * 2018-11-28 2021-07-23 罗欣药业(上海)有限公司 一种雌激素受体下调剂的盐型、晶型及其制备方法

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107074820B (zh) * 2014-07-25 2021-05-18 赛尔基因第二国际有限公司 Glp-1受体调节剂

Also Published As

Publication number Publication date
HRP20211938T1 (hr) 2022-03-18
PT3519407T (pt) 2021-12-10
ES2901599T3 (es) 2022-03-23
LT3519407T (lt) 2022-01-10
US20200131164A1 (en) 2020-04-30
HUE056805T2 (hu) 2022-03-28
WO2018064476A1 (en) 2018-04-05
US11066395B2 (en) 2021-07-20
EP3519407A1 (en) 2019-08-07
PL3519407T3 (pl) 2022-02-14
RS62814B1 (sr) 2022-02-28
EP3519407B1 (en) 2021-09-22
SI3519407T1 (sl) 2022-01-31

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