CY1118181T1 - Αναβραζοντα δισκια για χρηση σε εισπνοες - Google Patents

Αναβραζοντα δισκια για χρηση σε εισπνοες

Info

Publication number
CY1118181T1
CY1118181T1 CY20161101120T CY161101120T CY1118181T1 CY 1118181 T1 CY1118181 T1 CY 1118181T1 CY 20161101120 T CY20161101120 T CY 20161101120T CY 161101120 T CY161101120 T CY 161101120T CY 1118181 T1 CY1118181 T1 CY 1118181T1
Authority
CY
Cyprus
Prior art keywords
suspension
restoreable
discs
drug
particle size
Prior art date
Application number
CY20161101120T
Other languages
English (en)
Inventor
Marco Gentile
Marco Cantarini
Original Assignee
Dompé Farmaceutici S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dompé Farmaceutici S.P.A. filed Critical Dompé Farmaceutici S.P.A.
Publication of CY1118181T1 publication Critical patent/CY1118181T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/57Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone
    • A61K31/573Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids substituted in position 17 beta by a chain of two carbon atoms, e.g. pregnane or progesterone substituted in position 21, e.g. cortisone, dexamethasone, prednisone or aldosterone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0002Galenical forms characterised by the drug release technique; Application systems commanded by energy
    • A61K9/0007Effervescent
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/0012Galenical forms characterised by the site of application
    • A61K9/007Pulmonary tract; Aromatherapy
    • A61K9/0073Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy
    • A61K9/0078Sprays or powders for inhalation; Aerolised or nebulised preparations generated by other means than thermal energy for inhalation via a nebulizer such as a jet nebulizer, ultrasonic nebulizer, e.g. in the form of aqueous drug solutions or dispersions
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/20Pills, tablets, discs, rods
    • A61K9/2004Excipients; Inactive ingredients
    • A61K9/2009Inorganic compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dispersion Chemistry (AREA)
  • Otolaryngology (AREA)
  • Pulmonology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Η παρούσα εφεύρεση αναφέρεται στη χρήση αναβραζόντων δισκίων τα οποία περιέχουν αδιάλυτα δραστικά συστατικά για την παρασκευή εναιωρήματος για χρήση σε εισπνοές τα οποία διατηρούν το πρωτογενές μέγεθος σωματιδίων της φαρμακευτικής ουσίας. Τα δισκία διαλύονται στο διάλυμα έως ότου σχηματιστεί ένα εναιώρημα. Το εναιώρημα διατηρεί την αρχική κατανομή μεγέθους σωματιδίων της φαρμακευτικής ουσίας, εξασφαλίζοντας την επίτευξη του θεραπευτικού παραθύρου του εισπνεόμενου κλάσματος.
CY20161101120T 2007-06-22 2016-11-03 Αναβραζοντα δισκια για χρηση σε εισπνοες CY1118181T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP07110896 2007-06-22
EP08784529.3A EP2170348B1 (en) 2007-06-22 2008-06-20 Effervescent tablets for inhalatory use
PCT/EP2008/004993 WO2009000473A2 (en) 2007-06-22 2008-06-20 Effervescent tablets for inhalatory use

Publications (1)

Publication Number Publication Date
CY1118181T1 true CY1118181T1 (el) 2017-06-28

Family

ID=40186078

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20161101120T CY1118181T1 (el) 2007-06-22 2016-11-03 Αναβραζοντα δισκια για χρηση σε εισπνοες

Country Status (13)

Country Link
EP (1) EP2170348B1 (el)
BR (1) BRPI0814716A2 (el)
CY (1) CY1118181T1 (el)
DK (1) DK2170348T3 (el)
EA (1) EA021148B1 (el)
ES (1) ES2601860T3 (el)
HR (1) HRP20161388T1 (el)
HU (1) HUE030605T2 (el)
LT (1) LT2170348T (el)
PL (1) PL2170348T3 (el)
PT (1) PT2170348T (el)
SI (1) SI2170348T1 (el)
WO (1) WO2009000473A2 (el)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1921919B1 (en) 2005-07-14 2012-04-04 Lithera, Inc. Sustained release enhanced lipolytic formulation for regional adipose tissue treatment
ATE498396T1 (de) * 2008-07-21 2011-03-15 Falk Pharma Gmbh Pharmazeutische formulierung zur behandlung des oberen verdauungstraktes
US9132084B2 (en) 2009-05-27 2015-09-15 Neothetics, Inc. Methods for administration and formulations for the treatment of regional adipose tissue
GB2477030A (en) * 2010-01-15 2011-07-20 Lithera Inc Lyophilised forms of fluticasone, salmeterol and combinations thereof
CN105832681A (zh) 2010-11-24 2016-08-10 纽赛蒂克斯公司 选择性、亲脂性及长效型β激动剂单一治疗调配物和用于肥胖及外形凸起的美容治疗的方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP1438019A1 (en) * 2001-10-24 2004-07-21 PARI GmbH Spezialisten für effektive Inhalation Kit for the preparation of a pharmaceutical composition
ITMI20020808A1 (it) * 2002-04-17 2003-10-17 Chiesi Farma Spa Procedimento per la preparazione di una sospensione sterile di particelle di beclometasone dipropionato da somministrare per inalazione
US20040045546A1 (en) * 2002-09-05 2004-03-11 Peirce Management, Llc Pharmaceutical delivery system for oral inhalation through nebulization consisting of inert substrate impregnated with substance (S) to be solubilized or suspended prior to use
ITFI20030194A1 (it) * 2003-07-17 2005-01-18 Menarini Int Operations Lu Sa Composizione farmaceutiche effervescenti contenenti

Also Published As

Publication number Publication date
DK2170348T3 (en) 2016-11-07
EP2170348B1 (en) 2016-08-10
EA021148B1 (ru) 2015-04-30
PT2170348T (pt) 2016-11-02
EP2170348A2 (en) 2010-04-07
SI2170348T1 (sl) 2016-12-30
WO2009000473A3 (en) 2009-07-30
ES2601860T3 (es) 2017-02-16
HRP20161388T1 (hr) 2016-12-02
EA200971113A1 (ru) 2010-04-30
HUE030605T2 (hu) 2017-05-29
BRPI0814716A2 (pt) 2015-02-24
LT2170348T (lt) 2016-11-25
PL2170348T3 (pl) 2017-01-31
WO2009000473A2 (en) 2008-12-31

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