CY1116607T1 - AZAIDOLI UNITS AND METHODS OF USE - Google Patents

AZAIDOLI UNITS AND METHODS OF USE

Info

Publication number
CY1116607T1
CY1116607T1 CY20151100676T CY151100676T CY1116607T1 CY 1116607 T1 CY1116607 T1 CY 1116607T1 CY 20151100676 T CY20151100676 T CY 20151100676T CY 151100676 T CY151100676 T CY 151100676T CY 1116607 T1 CY1116607 T1 CY 1116607T1
Authority
CY
Cyprus
Prior art keywords
methods
ccr1
azaidoli
units
compounds
Prior art date
Application number
CY20151100676T
Other languages
Greek (el)
Inventor
Penglie Zhang
Andrew M K Pennell
John J Kim Wright
Wei Chen
Manmohan R Leleti
Yandong Li
Lianfa Li
Yuan Xu
Original Assignee
Chemocentryx, Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP20060773773 external-priority patent/EP1906965B1/en
Application filed by Chemocentryx, Inc. filed Critical Chemocentryx, Inc.
Publication of CY1116607T1 publication Critical patent/CY1116607T1/en

Links

Abstract

Παρέχονται ενώσεις που δρουν ως ισχυροί ανταγωνιστές του υποδοχέα CCR1 και έχουν in vivo αντι-φλεγμονώδη δραστικότητα. Οι ενώσεις γενικώς είναι παράγωγα αρύλ πιπεραζίνης και είναι χρήσιμες σε φαρμακευτικές συνθέσεις, σε μεθόδους για την θεραπεία προκαλούμενων από CCR1 ασθενειών και ως δείγματα αναφοράς σε δοκιμασίες για πιστοποίηση ανταγωνιστικών ανταγωνιστών CCR1.Compounds that act as potent antagonists of the CCR1 receptor are provided and have in vivo anti-inflammatory activity. The compounds are generally aryl piperazine derivatives and are useful in pharmaceutical compositions, in methods for the treatment of CCR1-mediated diseases and as controls in tests for the identification of competitive CCR1 antagonists.

CY20151100676T 2005-06-22 2015-08-03 AZAIDOLI UNITS AND METHODS OF USE CY1116607T1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US69352505A 2005-06-22 2005-06-22
EP20060773773 EP1906965B1 (en) 2005-06-22 2006-06-22 Azaindazole compounds and methods of use

Publications (1)

Publication Number Publication Date
CY1116607T1 true CY1116607T1 (en) 2017-03-15

Family

ID=58459830

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20151100676T CY1116607T1 (en) 2005-06-22 2015-08-03 AZAIDOLI UNITS AND METHODS OF USE

Country Status (1)

Country Link
CY (1) CY1116607T1 (en)

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