CY1116085T1 - OXYGEN-SUBSTITUTED 3-HETEROYLAMINE-PROPIONIC ACID PRODUCERS AND THEIR USE AS PHARMACEUTICAL SUBSTANCES - Google Patents
OXYGEN-SUBSTITUTED 3-HETEROYLAMINE-PROPIONIC ACID PRODUCERS AND THEIR USE AS PHARMACEUTICAL SUBSTANCESInfo
- Publication number
- CY1116085T1 CY1116085T1 CY20151100142T CY151100142T CY1116085T1 CY 1116085 T1 CY1116085 T1 CY 1116085T1 CY 20151100142 T CY20151100142 T CY 20151100142T CY 151100142 T CY151100142 T CY 151100142T CY 1116085 T1 CY1116085 T1 CY 1116085T1
- Authority
- CY
- Cyprus
- Prior art keywords
- heteroylamine
- substituted
- oxygen
- propionic acid
- pharmaceutical substances
- Prior art date
Links
Abstract
Η παρούσα εφεύρεση αναφέρεται στις ενώσεις του χημικού τύπου I, όπου οι A, D, Ε, G, R10, R30, R40, R50 και R60 ορίζονται στις αξιώσεις, και είναι πολύτιμες, φαρμακευτικά δραστικές ενώσεις. Είναι αναστολείς της πρωτεάσης καθεψίνης Α, και μπορούν να χρησιμοποιηθούν για την αντιμετώπιση νοσημάτων όπως είναι παραδείγματος χάριν η αθηροσκλήρυνση, η καρδιακή ανεπάρκεια, οι νεφρικές παθήσεις, οι ηπατοπάθειες ή τα φλεγμονώδη νοσήματα. Η εφεύρεση αναφέρεται επίσης σε διαδικασίες παρασκευής των ενώσεων του χημικού τύπου I, στη χρήση αυτών και στις φαρμακευτικές συνθέσεις που τις περιέχουν.The present invention relates to the compounds of formula I, wherein A, D, E, G, R10, R30, R40, R50 and R60 are defined in the claims, and are valuable, pharmaceutically active compounds. They are inhibitors of cathepsin A protease, and can be used to treat diseases such as atherosclerosis, heart failure, kidney disease, liver disease or inflammatory diseases. The invention also relates to processes for the preparation of the compounds of formula I, their use and the pharmaceutical compositions containing them.
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP10305080 | 2010-01-26 | ||
US30911910A | 2010-03-01 | 2010-03-01 | |
EP11701123.9A EP2528902B1 (en) | 2010-01-26 | 2011-01-26 | Oxygen-substituted 3-heteroaroylamino-propionic acid derivatives and their use as pharmaceuticals |
Publications (1)
Publication Number | Publication Date |
---|---|
CY1116085T1 true CY1116085T1 (en) | 2017-02-08 |
Family
ID=58457908
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CY20151100142T CY1116085T1 (en) | 2010-01-26 | 2015-02-12 | OXYGEN-SUBSTITUTED 3-HETEROYLAMINE-PROPIONIC ACID PRODUCERS AND THEIR USE AS PHARMACEUTICAL SUBSTANCES |
Country Status (1)
Country | Link |
---|---|
CY (1) | CY1116085T1 (en) |
-
2015
- 2015-02-12 CY CY20151100142T patent/CY1116085T1/en unknown
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