CY1114923T1 - 6-Substituted isokinolines and isokinolines - Google Patents

6-Substituted isokinolines and isokinolines

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Publication number
CY1114923T1
CY1114923T1 CY20131101086T CY131101086T CY1114923T1 CY 1114923 T1 CY1114923 T1 CY 1114923T1 CY 20131101086 T CY20131101086 T CY 20131101086T CY 131101086 T CY131101086 T CY 131101086T CY 1114923 T1 CY1114923 T1 CY 1114923T1
Authority
CY
Cyprus
Prior art keywords
isokinolines
substituted
rho
kinase
isoquinolones
Prior art date
Application number
CY20131101086T
Other languages
Greek (el)
Inventor
Oliver Plettenburg
Katrin Lorenz
Matthias Loehn
John Weston
Heinz-Werner Kleemann
Original Assignee
Sanofi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP09768948.3A external-priority patent/EP2313374B1/en
Application filed by Sanofi filed Critical Sanofi
Publication of CY1114923T1 publication Critical patent/CY1114923T1/en

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Abstract

Η εφεύρεση σχετίζεται με 6-υποκατεστημένα παράγωγα ισοκινολινών και ισοκινολινονών με τον τύπο (Ι) τα οποία είναι χρήσιμα για τη θεραπευτική αντιμετώπιση ή/και την πρόληψη νόσων οι οποίες συνδέονται με τη Rho-κινάση ή/και τη φωσφορυλίωση της φωσφατάσης της ελαφράς αλυσίδας της μυοσίνης στη οποία διαμεσολαβεί η Rho-κινάση, και με συνθέσεις οι οποίες περιέχουν τις ενώσεις αυτές.The invention relates to 6-substituted isoquinolines and isoquinolones derivatives of formula (I) which are useful for the treatment and / or prevention of diseases associated with Rho-kinase and / or phosphorylation of its light chain phosphatase. myosin mediated by Rho-kinase, and with compositions containing these compounds.

CY20131101086T 2008-06-24 2013-12-03 6-Substituted isokinolines and isokinolines CY1114923T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP08290605 2008-06-24
US15314509A 2009-02-17 2009-02-17
EP09768948.3A EP2313374B1 (en) 2008-06-24 2009-06-19 6-substituted isoquinolines and isoquinolinones

Publications (1)

Publication Number Publication Date
CY1114923T1 true CY1114923T1 (en) 2016-12-14

Family

ID=58464065

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20131101086T CY1114923T1 (en) 2008-06-24 2013-12-03 6-Substituted isokinolines and isokinolines

Country Status (1)

Country Link
CY (1) CY1114923T1 (en)

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