CY1114324T1 - ΜΗ ΚΡΥΣΤΑΛΛΙΚΗ ΜΟΡΦΗ Ν-{2-ΦΘΟΡΟ-5-[3-(ΘΕΙΟΦΑΙΝΟ-2-ΚΑΡΒΟΝΥΛ)-ΠΥΡΑΖΟΛΟ[1,5-a]ΠΥΡΙΜΙΔΙΝ-7-ΥΛ]-ΦΑΙΝΥΛ}-Ν-ΜΕΘΥΛ-ΑΚΕΤΑΜΙΔΙΟΥ - Google Patents

ΜΗ ΚΡΥΣΤΑΛΛΙΚΗ ΜΟΡΦΗ Ν-{2-ΦΘΟΡΟ-5-[3-(ΘΕΙΟΦΑΙΝΟ-2-ΚΑΡΒΟΝΥΛ)-ΠΥΡΑΖΟΛΟ[1,5-a]ΠΥΡΙΜΙΔΙΝ-7-ΥΛ]-ΦΑΙΝΥΛ}-Ν-ΜΕΘΥΛ-ΑΚΕΤΑΜΙΔΙΟΥ

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Publication number
CY1114324T1
CY1114324T1 CY20131100320T CY131100320T CY1114324T1 CY 1114324 T1 CY1114324 T1 CY 1114324T1 CY 20131100320 T CY20131100320 T CY 20131100320T CY 131100320 T CY131100320 T CY 131100320T CY 1114324 T1 CY1114324 T1 CY 1114324T1
Authority
CY
Cyprus
Prior art keywords
pyrazolo
pyrimidin
fluoro
carbonyl
methyl
Prior art date
Application number
CY20131100320T
Other languages
English (en)
Inventor
Luis Anglada
Albert Palomer
Antonio Guglietta
Original Assignee
Ferrer Internacional, S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP06123652A external-priority patent/EP1921079A1/en
Application filed by Ferrer Internacional, S.A. filed Critical Ferrer Internacional, S.A.
Publication of CY1114324T1 publication Critical patent/CY1114324T1/el

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Abstract

Η παρούσα εφεύρεση αναφέρεται σε μια μη κρυσταλλική μορφή Ν-{2-φθορο-5-[3-(θειοφαινο-2-καρβονυλ)-πυραζολο[1,5-a]πυριμιδιν-7-υλ]-φαινυλ}-Ν-μεθυλ-ακεταμιδίου, σε μεθόδους για την παρασκευή της, στη χρήση της ως ένας θεραπευτικός δραστικός παράγοντας και σε φαρμακευτικές συνθέσεις περιέχουσες τη νέα μορφή.
CY20131100320T 2006-11-08 2013-04-19 ΜΗ ΚΡΥΣΤΑΛΛΙΚΗ ΜΟΡΦΗ Ν-{2-ΦΘΟΡΟ-5-[3-(ΘΕΙΟΦΑΙΝΟ-2-ΚΑΡΒΟΝΥΛ)-ΠΥΡΑΖΟΛΟ[1,5-a]ΠΥΡΙΜΙΔΙΝ-7-ΥΛ]-ΦΑΙΝΥΛ}-Ν-ΜΕΘΥΛ-ΑΚΕΤΑΜΙΔΙΟΥ CY1114324T1 (el)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US86481406A 2006-11-08 2006-11-08
EP06123652A EP1921079A1 (en) 2006-11-08 2006-11-08 Amorphous form of N-{2-Fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo[1,5-a] pyrimidin-7-yl]-phenyl}-N-methyl-acetamide
EP07822324A EP2086978B1 (en) 2006-11-08 2007-11-07 Amorphous form of n-{2-fluoro-5-[3-(thiophene-2-carbonyl)-pyrazolo [1,5-a]pyrimidin-7-yl]-phenyl-n-methyl-acetamide

Publications (1)

Publication Number Publication Date
CY1114324T1 true CY1114324T1 (el) 2016-08-31

Family

ID=58436471

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20131100320T CY1114324T1 (el) 2006-11-08 2013-04-19 ΜΗ ΚΡΥΣΤΑΛΛΙΚΗ ΜΟΡΦΗ Ν-{2-ΦΘΟΡΟ-5-[3-(ΘΕΙΟΦΑΙΝΟ-2-ΚΑΡΒΟΝΥΛ)-ΠΥΡΑΖΟΛΟ[1,5-a]ΠΥΡΙΜΙΔΙΝ-7-ΥΛ]-ΦΑΙΝΥΛ}-Ν-ΜΕΘΥΛ-ΑΚΕΤΑΜΙΔΙΟΥ

Country Status (1)

Country Link
CY (1) CY1114324T1 (el)

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