CY1111840T1 - Χρηση του 4-κυκλοπροπυλμεθοξυ-ν-(3,5-διχλωρο-1-οξειδο-πυριδιν-4-υλ)-5-(μεθοξυ)πυριδιν-2-καρβοξαμιδιου για τη θεραπεια κινητικων διαταραχων που σχετιζονται με τη νοσο toy parkinson - Google Patents

Χρηση του 4-κυκλοπροπυλμεθοξυ-ν-(3,5-διχλωρο-1-οξειδο-πυριδιν-4-υλ)-5-(μεθοξυ)πυριδιν-2-καρβοξαμιδιου για τη θεραπεια κινητικων διαταραχων που σχετιζονται με τη νοσο toy parkinson

Info

Publication number
CY1111840T1
CY1111840T1 CY20111100887T CY111100887T CY1111840T1 CY 1111840 T1 CY1111840 T1 CY 1111840T1 CY 20111100887 T CY20111100887 T CY 20111100887T CY 111100887 T CY111100887 T CY 111100887T CY 1111840 T1 CY1111840 T1 CY 1111840T1
Authority
CY
Cyprus
Prior art keywords
methoxy
carboxamide
pyridin
dichloro
pyridine
Prior art date
Application number
CY20111100887T
Other languages
Greek (el)
English (en)
Inventor
Philippe Delay-Goyet
Claire Delgorge
Christine Menet
Gilles Poughon
Christine Ravinet-Trillou
Original Assignee
Sanofi
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sanofi filed Critical Sanofi
Publication of CY1111840T1 publication Critical patent/CY1111840T1/el

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/14Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16Anti-Parkinson drugs

Landscapes

  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyridine Compounds (AREA)
CY20111100887T 2007-04-19 2011-09-15 Χρηση του 4-κυκλοπροπυλμεθοξυ-ν-(3,5-διχλωρο-1-οξειδο-πυριδιν-4-υλ)-5-(μεθοξυ)πυριδιν-2-καρβοξαμιδιου για τη θεραπεια κινητικων διαταραχων που σχετιζονται με τη νοσο toy parkinson CY1111840T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR0702853A FR2915100B1 (fr) 2007-04-19 2007-04-19 Utilisation du 4-cyclopropylmethoxy-n-(3,5-dichloro-1-oxydo- pyridin-4-yl)-5-(methoxy)pyridine-2-carboxalide pour le traitement des desordres moteurs lies a la maladie de parkinson
EP08787963A EP2146714B1 (fr) 2007-04-19 2008-04-16 Utilisation du 4-cyclopropylmethoxy-n-(3,5-dichloro-1 -oxydo- pyridin-4-yl)-5-(methoxy)pyridine-2-carboxamide pour le traitement des desordres moteurs lies a la maladie de parkinson

Publications (1)

Publication Number Publication Date
CY1111840T1 true CY1111840T1 (el) 2015-10-07

Family

ID=38712405

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20111100887T CY1111840T1 (el) 2007-04-19 2011-09-15 Χρηση του 4-κυκλοπροπυλμεθοξυ-ν-(3,5-διχλωρο-1-οξειδο-πυριδιν-4-υλ)-5-(μεθοξυ)πυριδιν-2-καρβοξαμιδιου για τη θεραπεια κινητικων διαταραχων που σχετιζονται με τη νοσο toy parkinson

Country Status (33)

Country Link
US (1) US20100130554A1 (https=)
EP (1) EP2146714B1 (https=)
JP (1) JP5386478B2 (https=)
KR (2) KR101503942B1 (https=)
CN (1) CN101663035B (https=)
AR (1) AR066108A1 (https=)
AT (1) ATE513548T1 (https=)
AU (1) AU2008257322B2 (https=)
BR (1) BRPI0810444A2 (https=)
CA (1) CA2684174C (https=)
CL (1) CL2008001136A1 (https=)
CY (1) CY1111840T1 (https=)
DK (1) DK2146714T3 (https=)
EA (1) EA019194B1 (https=)
ES (1) ES2367408T3 (https=)
FR (1) FR2915100B1 (https=)
HR (1) HRP20110666T1 (https=)
IL (1) IL201448A (https=)
JO (1) JO2678B1 (https=)
MA (1) MA31367B1 (https=)
ME (1) ME00935B (https=)
MX (1) MX2009011284A (https=)
MY (1) MY148092A (https=)
NZ (1) NZ580482A (https=)
PA (1) PA8776801A1 (https=)
PL (1) PL2146714T3 (https=)
PT (1) PT2146714E (https=)
RS (1) RS51869B (https=)
SI (1) SI2146714T1 (https=)
TW (1) TWI439269B (https=)
UY (1) UY31035A1 (https=)
WO (1) WO2008145841A1 (https=)
ZA (1) ZA200907251B (https=)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
BR112015011849A2 (pt) * 2012-11-28 2017-07-11 Sanofi Sa método de preparação de formas de cristal de 4 (ciclopropilmetoxi)-n-(3,5-dicloro-1-oxidopiridin-4-il)-5-metoxipiridina-2-carboxamida e formas de cristal da mesma
US9624100B2 (en) 2014-06-12 2017-04-18 Apple Inc. Micro pick up array pivot mount with integrated strain sensing elements
AU2024357688A1 (en) * 2023-10-12 2026-04-23 Alto Neuroscience, Inc. Treatment of neuropsychiatric disorders with tilivapram
WO2025079694A1 (ja) * 2023-10-12 2025-04-17 株式会社 メドレックス 経皮吸収組成物

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4193926A (en) * 1974-03-20 1980-03-18 Schering Aktiengesellschaft 4-(Polyalkoxy phenyl)-2-pyrrolidones
JP3775685B2 (ja) * 1993-07-28 2006-05-17 ローン−プーラン・ロレ・リミテツド Pde▲iv▼およびtnf抑制剤としての化合物
US6177077B1 (en) * 1999-02-24 2001-01-23 Edward L. Tobinick TNT inhibitors for the treatment of neurological disorders
PT1244649E (pt) * 1999-12-23 2005-06-30 Icos Corp Inibidores de fosfodiesterase especificos de mfa ciclica
EP1370211A4 (en) * 2001-03-02 2005-02-09 Bristol Myers Squibb Co SIMULTANEOUS ADMINISTRATION OF MELANOCORTIN RECEPTOR AGONISTS AND A PHOSPHODIESTERASE HEMMER FOR THE TREATMENT OF DISEASES RELATED TO CYCLIC AMP
AU2003281219A1 (en) * 2002-07-02 2004-01-23 Bernard Cote Di-aryl-substituted-ethane pyridone pde4 inhibitors
DE602004032522D1 (de) * 2003-03-12 2011-06-16 Celgene Corp Mit n-alkylhydroxamsäuren substituierte isoindolylverbindungen und deren pharmazeutische verwendung
JP2008543781A (ja) * 2005-06-10 2008-12-04 メモリー・ファーマシューティカルズ・コーポレイション ホスフオジエステラーゼ4阻害剤
US20070021451A1 (en) * 2005-07-20 2007-01-25 Hamamatsu University School Of Medicine Method for preventing or treating neurologic damage after spinal cord injury

Also Published As

Publication number Publication date
MX2009011284A (es) 2009-11-02
IL201448A0 (en) 2010-05-31
RS51869B (sr) 2012-02-29
SI2146714T1 (sl) 2011-10-28
US20100130554A1 (en) 2010-05-27
IL201448A (en) 2014-08-31
TW200911247A (en) 2009-03-16
WO2008145841A1 (fr) 2008-12-04
CL2008001136A1 (es) 2009-01-16
CN101663035B (zh) 2012-06-20
UY31035A1 (es) 2008-11-28
EP2146714A1 (fr) 2010-01-27
MY148092A (en) 2013-02-28
AU2008257322A1 (en) 2008-12-04
JO2678B1 (en) 2013-03-03
JP5386478B2 (ja) 2014-01-15
ATE513548T1 (de) 2011-07-15
PT2146714E (pt) 2011-09-02
HK1141725A1 (en) 2010-11-19
ZA200907251B (en) 2011-04-28
MA31367B1 (fr) 2010-05-03
TWI439269B (zh) 2014-06-01
BRPI0810444A2 (pt) 2016-05-31
DK2146714T3 (da) 2011-10-10
CA2684174C (fr) 2014-02-25
EP2146714B1 (fr) 2011-06-22
FR2915100B1 (fr) 2009-06-05
EA200970970A1 (ru) 2010-02-26
CN101663035A (zh) 2010-03-03
ES2367408T3 (es) 2011-11-03
NZ580482A (en) 2011-10-28
AU2008257322B2 (en) 2013-06-13
HRP20110666T1 (hr) 2011-10-31
PL2146714T3 (pl) 2011-10-31
KR101503942B1 (ko) 2015-03-18
CA2684174A1 (fr) 2008-12-04
JP2010524906A (ja) 2010-07-22
EA019194B1 (ru) 2014-01-30
KR20090130059A (ko) 2009-12-17
ME00935B (me) 2012-06-20
AR066108A1 (es) 2009-07-22
PA8776801A1 (es) 2008-11-19
KR20150004885A (ko) 2015-01-13
FR2915100A1 (fr) 2008-10-24

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