CU24174B1 - TRIAZOLOPIRIDINS AS QUINASE INHIBITORS MPS-1 - Google Patents

TRIAZOLOPIRIDINS AS QUINASE INHIBITORS MPS-1

Info

Publication number
CU24174B1
CU24174B1 CUP2013000141A CU20130141A CU24174B1 CU 24174 B1 CU24174 B1 CU 24174B1 CU P2013000141 A CUP2013000141 A CU P2013000141A CU 20130141 A CU20130141 A CU 20130141A CU 24174 B1 CU24174 B1 CU 24174B1
Authority
CU
Cuba
Prior art keywords
compounds
triazolopiridins
mps
quinase
inhibitors
Prior art date
Application number
CUP2013000141A
Other languages
Spanish (es)
Other versions
CU20130141A7 (en
Inventor
Volker Schulze
Dirk Kosemund
Antje Margret Wengner
Gerhard Siemeister
Detlef Stöckigt
Philip Lienau
Hartmut Schirok
Hans Briem
Original Assignee
Bayer Ip Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ip Gmbh filed Critical Bayer Ip Gmbh
Priority claimed from PCT/EP2012/056914 external-priority patent/WO2012143329A1/en
Publication of CU20130141A7 publication Critical patent/CU20130141A7/en
Publication of CU24174B1 publication Critical patent/CU24174B1/en

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Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Compuestos de triazolopiridina de la fórmula general (I) Espacio para Fórmula donde R^1, R^2, R^3, R^4 y R^5 tienen los valores que se definen en la descripción y en las reinvindicaciones. Métodos para preparar dichos compuestos. Composiciones y combinaciones farmacéuticas que comprenden dichos compuestos. Uso de dichos compuestos para preparar una composición farmacéuticamente para el tratamiento o la profilaxis de una enfermedad. Compuestos intermediarios útiles para preparar dichos compuestos.Triazolopyridine compounds of the general formula (I) Space for Formula where R ^ 1, R ^ 2, R ^ 3, R ^ 4 and R ^ 5 have the values defined in the description and in the claims. Methods for preparing said compounds. Compositions and pharmaceutical combinations comprising said compounds. Use of said compounds to prepare a pharmaceutical composition for the treatment or prophylaxis of a disease. Intermediate compounds useful for preparing said compounds.

CUP2013000141A 2011-04-21 2012-04-16 TRIAZOLOPIRIDINS AS QUINASE INHIBITORS MPS-1 CU24174B1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP11163342 2011-04-21
EP11167872 2011-05-27
PCT/EP2012/056914 WO2012143329A1 (en) 2011-04-21 2012-04-16 Triazolopyridines

Publications (2)

Publication Number Publication Date
CU20130141A7 CU20130141A7 (en) 2014-03-26
CU24174B1 true CU24174B1 (en) 2016-04-25

Family

ID=52394781

Family Applications (1)

Application Number Title Priority Date Filing Date
CUP2013000141A CU24174B1 (en) 2011-04-21 2012-04-16 TRIAZOLOPIRIDINS AS QUINASE INHIBITORS MPS-1

Country Status (2)

Country Link
CU (1) CU24174B1 (en)
TN (1) TN2013000426A1 (en)

Also Published As

Publication number Publication date
TN2013000426A1 (en) 2015-03-30
CU20130141A7 (en) 2014-03-26

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Legal Events

Date Code Title Description
FG Grant of patent