CU23698B7 -
PROCEDURE FOR THE PREPARATION OF THE CRISTALINA DELTA D FORM OF IVABRADINE CHLORHYDRATE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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PROCEDURE FOR THE PREPARATION OF THE CRISTALINA DELTA D FORM OF IVABRADINE CHLORHYDRATE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
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CU23698B7
CU23698B7CU20060195ACU20060195ACU23698B7CU 23698 B7CU23698 B7CU 23698B7CU 20060195 ACU20060195 ACU 20060195ACU 20060195 ACU20060195 ACU 20060195ACU 23698 B7CU23698 B7CU 23698B7
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Priority to CU20060195ApriorityCriticalpatent/CU23698B7/en
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Publication of CU23698B7publicationCriticalpatent/CU23698B7/en
Pharmaceuticals Containing Other Organic And Inorganic Compounds
(AREA)
Abstract
La presente invención se refiere a un procedimiento de preparación de la forma cristalina delta d del clorhidrato de ivabradina de fórmula (I) (ESPACIO PARA FÓRMULA) consistiendo en el precalentamientio del acetonitrilo o una mezcla de acetonitrilo y agua, seguidamente se anade el clorhidrato de ivabradina y se enfría la solución obtenida a temperatura ambiente, y se mantiene a esta temperatura hasta la completa cristalización, luego se deshidratan los cristales obtenidos.The present invention relates to a process for preparing the delta d crystalline form of the ivabradine hydrochloride of formula (I) (SPACE FOR FORMULA) consisting of the preheating of acetonitrile or a mixture of acetonitrile and water, then the hydrochloride of Ivabradine and the solution obtained is cooled to room temperature, and is maintained at this temperature until complete crystallization, then the crystals obtained are dehydrated.
CU20060195A2006-10-112006-10-11
PROCEDURE FOR THE PREPARATION OF THE CRISTALINA DELTA D FORM OF IVABRADINE CHLORHYDRATE AND THE PHARMACEUTICAL COMPOSITIONS CONTAINING THEM
CU23698B7
(en)
Compounds derived from dihydropyrimidine-2,4- (1h, 3h) -dione; crystalline forms, intermediate compounds; process for preparing intermediate compounds, pharmaceutical composition; and its useful use to treat hepatitis C in a mammal.
SUBSTITUTED DERIVATIVES OF N- (3,4-DIHIDRO-2H-CROMEN-3-IL) FORMAMIDA AND N- (1, 2,3, 4-TETRAHIDRONAFTALEN-2-IL) FORMAMIDA, SALTS OF THE SAME, COMPOSITIONS THAT CONTAIN THEM , PROCEDURES FOR PREPARATION AND APPLICATIONS
DERIVATIVES OF AZAESPIRODECANONA, PHARMACEUTICAL COMPOSITIONS THAT CONTAIN THEM, PROCEDURE TO PREPARE THEM AND USE OF THEM FOR THE TREATMENT OF DIABETES, OBESITY AND CARDIOVASCULAR DISEASES, BETWEEN OTHER