CU20160141A7 - Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular - Google Patents
Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascularInfo
- Publication number
- CU20160141A7 CU20160141A7 CUP2016000141A CU20160141A CU20160141A7 CU 20160141 A7 CU20160141 A7 CU 20160141A7 CU P2016000141 A CUP2016000141 A CU P2016000141A CU 20160141 A CU20160141 A CU 20160141A CU 20160141 A7 CU20160141 A7 CU 20160141A7
- Authority
- CU
- Cuba
- Prior art keywords
- central
- nervous system
- diseases
- benzodiazepina
- activity
- Prior art date
Links
- 210000000653 nervous system Anatomy 0.000 title abstract 2
- 230000002792 vascular Effects 0.000 title abstract 2
- 230000000694 effects Effects 0.000 title 1
- 201000010099 disease Diseases 0.000 abstract 4
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 4
- 208000028698 Cognitive impairment Diseases 0.000 abstract 1
- 208000037273 Pathologic Processes Diseases 0.000 abstract 1
- 230000032683 aging Effects 0.000 abstract 1
- 208000010877 cognitive disease Diseases 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 230000004065 mitochondrial dysfunction Effects 0.000 abstract 1
- 208000004296 neuralgia Diseases 0.000 abstract 1
- 208000015122 neurodegenerative disease Diseases 0.000 abstract 1
- 208000021722 neuropathic pain Diseases 0.000 abstract 1
- 230000036542 oxidative stress Effects 0.000 abstract 1
- 230000009054 pathological process Effects 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
- A61K31/551—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole having two nitrogen atoms, e.g. dilazep
- A61K31/5513—1,4-Benzodiazepines, e.g. diazepam or clozapine
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/08—Solutions
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2022—Organic macromolecular compounds
- A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
- A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Life Sciences & Earth Sciences (AREA)
- Veterinary Medicine (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Animal Behavior & Ethology (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Engineering & Computer Science (AREA)
- Oil, Petroleum & Natural Gas (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
<p>Compuesto de formula III, sus derivados y composiciones farmacéuticas que los contienen para el tratamiento de enfermedades del sistema nervioso central y vascular, especialmente trastornos neurodegenerativos, con deterioro cognitivo, enfermedades asociadas al estrés oxidativo, enfermedades que cursan con disfunción mitocondrial, enfermedad de Parkinson y dolor neuropático, así como procesos patológicos asociadas con el envejecimiento. ESPACIO PARA FÓRMULA</p>
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CUP2016000141A CU20160141A7 (es) | 2016-09-27 | 2016-09-27 | Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular |
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CUP2016000141A CU20160141A7 (es) | 2016-09-27 | 2016-09-27 | Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CU20160141A7 true CU20160141A7 (es) | 2018-05-08 |
Family
ID=62104051
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CUP2016000141A CU20160141A7 (es) | 2016-09-27 | 2016-09-27 | Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular |
Country Status (1)
| Country | Link |
|---|---|
| CU (1) | CU20160141A7 (es) |
-
2016
- 2016-09-27 CU CUP2016000141A patent/CU20160141A7/es unknown
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| CL2018002505A1 (es) | Inhibidores del envejecimiento proteico-proteico wdr5 | |
| CL2018003701A1 (es) | Compuestos heterocíclicos como inmunomoduladores. | |
| CL2018003050A1 (es) | Isoquinolin-3-il-carboxamidas, y preparación y uso de las mismas. | |
| CU20190073A7 (es) | 2-heteroaril-3-oxo-2,3-dihidropiridazin-4-carboxamidas | |
| NI201600164A (es) | Compuestos y composiciones como agonistas del receptor tipo toll 7 | |
| NI201800124A (es) | 3-oxo-2,6-difenil-2,3-dihidropiridazin-4-carboxamidas | |
| CL2018000375A1 (es) | 2-amino-3-fluoro-3-(fluorometil)-6-meti-6-fenil-3,4,5,6-tetrahidropiridinas como inhibidores de bace1. | |
| BR112016025048A2 (pt) | compostos e composições como agonistas do receptor tipo toll7 | |
| CO2019012767A2 (es) | Compuesto de fenil-2-hidroxi-acetilamino-2-metil-fenilo | |
| CO2017005959A2 (es) | 4-oxo-3,4-dihidro-1,2,3-benzotriazinas como moduladores de gpr139 | |
| CL2019002583A1 (es) | Inhibidores duales de magl y faah. | |
| CL2016002615A1 (es) | Heterociclil-sulfonas sustituidas con heteroarilo y su uso contra el dolor, accidente cerebrovascular, transtornos anímicos, epilepsia, esquizofrenia y trastornos neurodegenerativos. | |
| CL2021001198A1 (es) | Compuestos heteroaromáticos como inhibidores de vanina | |
| MX2020004666A (es) | Compuestos de pilocarpina con ácido lipoico para el tratamiento de trastornos oculares. | |
| ECSP19026702A (es) | Compuestos novedosos para el tratamiento de enfermedades parasitarias | |
| MX2018001592A (es) | Composiciones y metodos para el tratamiento y la prevencion de trastornos neurodegenerativos. | |
| CL2018001631A1 (es) | Compuestos de dihidroquinolinsulfonamida de alquilo | |
| CO2021007442A2 (es) | Compuesto de 1,3,4-oxadiazolona y fármaco | |
| CU20160058A7 (es) | Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular | |
| CU20160141A7 (es) | Derivado de benzodiazepina con actividad sobre el sistema nervioso central y vascular | |
| CO2020001375A2 (es) | Derivado de adamantilmetilamina y uso del mismo como producto farmacéutico | |
| EA201991835A1 (ru) | 2-гетероарил-3-оксо-2,3-дигидропиридазин-4-карбоксамиды для лечения злокачественного новообразования | |
| CR20190028A (es) | Compuestos heterocíclicos como inmunomoduladores | |
| BR112017014226A2 (pt) | derivados de heterociclilalquina e sua utilização como moduladores de receptores mglur5 |