CS331491A3 - Cyclopeptides, process of their preparation and pharmaceuticals based thereon - Google Patents

Cyclopeptides, process of their preparation and pharmaceuticals based thereon

Info

Publication number
CS331491A3
CS331491A3 CS913314A CS331491A CS331491A3 CS 331491 A3 CS331491 A3 CS 331491A3 CS 913314 A CS913314 A CS 913314A CS 331491 A CS331491 A CS 331491A CS 331491 A3 CS331491 A3 CS 331491A3
Authority
CS
Czechoslovakia
Prior art keywords
cyclopeptides
preparation
pharmaceuticals based
pharmaceuticals
Prior art date
Application number
CS913314A
Other languages
Czech (cs)
Inventor
Gunter Dr Holzemann
Alfred Dr Jonczyk
Jurgen Harting
Hartmut Greiner
Original Assignee
Merck Patent Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merck Patent Gmbh filed Critical Merck Patent Gmbh
Publication of CS331491A3 publication Critical patent/CS331491A3/en

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/50Cyclic peptides containing at least one abnormal peptide link
    • C07K7/52Cyclic peptides containing at least one abnormal peptide link with only normal peptide links in the ring
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K7/00Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
    • C07K7/04Linear peptides containing only normal peptide links
    • C07K7/22Tachykinins, e.g. Eledoisins, Substance P; Related peptides
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/08Bronchodilators
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pain & Pain Management (AREA)
  • Biochemistry (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Biomedical Technology (AREA)
  • Pulmonology (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
CS913314A 1990-11-02 1991-11-01 Cyclopeptides, process of their preparation and pharmaceuticals based thereon CS331491A3 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4034829A DE4034829A1 (en) 1990-11-02 1990-11-02 CYCLOPEPTIDE

Publications (1)

Publication Number Publication Date
CS331491A3 true CS331491A3 (en) 1992-05-13

Family

ID=6417499

Family Applications (1)

Application Number Title Priority Date Filing Date
CS913314A CS331491A3 (en) 1990-11-02 1991-11-01 Cyclopeptides, process of their preparation and pharmaceuticals based thereon

Country Status (11)

Country Link
EP (1) EP0484719A3 (en)
JP (1) JPH04300895A (en)
KR (1) KR920009846A (en)
AU (1) AU8676291A (en)
CA (1) CA2054667A1 (en)
CS (1) CS331491A3 (en)
DE (1) DE4034829A1 (en)
HU (1) HUT61582A (en)
IE (1) IE913831A1 (en)
PT (1) PT99384A (en)
ZA (1) ZA918717B (en)

Families Citing this family (21)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE69231395T3 (en) 1991-09-20 2005-07-21 Glaxo Group Ltd., Greenford New medical indication for tachykinin antagonists
GB9702377D0 (en) * 1996-02-23 1997-03-26 Zeneca Ltd Peptide derivatives
GB9620819D0 (en) * 1996-10-05 1996-11-20 Zeneca Ltd Chemical compounds
TR199802537T2 (en) 1996-06-07 1999-03-22 Zeneca Limited Peptide tèrevleri.
GB9621836D0 (en) 1996-10-19 1996-12-11 Zeneca Ltd Peptide compounds
GB9624562D0 (en) 1996-11-27 1997-01-15 Zeneca Ltd Peptide derivatives
KR100408624B1 (en) * 2000-10-06 2003-12-06 엘지전선 주식회사 Poly vinyl chloride insulator composition for wire and cable
EP2117538A1 (en) 2007-01-24 2009-11-18 Glaxo Group Limited Pharmaceutical compositions comprising 2-methoxy-5- (5-trifluoromethyl-tetrazol-i-yl-benzyl) - (2s-phenyl-piperidin-3s-yl-)
UA105182C2 (en) 2008-07-03 2014-04-25 Ньюрексон, Інк. Benzoxazines, benzothiazines, and related compounds having nos inhibitory activity
US9446029B2 (en) 2010-07-27 2016-09-20 Colorado State University Research Foundation Use of NK-1 receptor antagonists in management of visceral pain
IN2014CN02806A (en) 2011-10-14 2015-07-03 Bristol Myers Squibb Co
IN2014CN02805A (en) 2011-10-14 2015-07-03 Bristol Myers Squibb Co
MY165742A (en) 2011-10-14 2018-04-23 Bristol Myers Squibb Co Substituted tetrahydroisoquinoline compounds as factor xia inhibitors
US9403774B2 (en) 2012-10-12 2016-08-02 Bristol-Myers Squibb Company Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors
EP2906551B1 (en) 2012-10-12 2018-02-28 Bristol-Myers Squibb Company Crystalline forms of a factor xia inhibitor
US9315519B2 (en) 2012-10-12 2016-04-19 Bristol-Myers Squibb Company Guanidine substituted tetrahydroisoquinoline compounds as factor XIa inhibitors
ES2712699T3 (en) 2013-03-25 2019-05-14 Bristol Myers Squibb Co Tetrahydroisoquinolines containing substituted azoles as inhibitors of factor XIa
UY35971A (en) 2014-01-31 2015-07-31 Bristol Myers Squibb Company Una Corporación Del Estado De Delaware MACROCICLOS WITH GROUPS P2? AROMATICS AS INHIBITORS OF THE XIA FACTOR
NO2760821T3 (en) 2014-01-31 2018-03-10
ES2714283T3 (en) 2014-09-04 2019-05-28 Bristol Myers Squibb Co Macrocycles of diamide that are inhibitors of FXIa
US9453018B2 (en) 2014-10-01 2016-09-27 Bristol-Myers Squibb Company Pyrimidinones as factor XIa inhibitors

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB8807246D0 (en) * 1988-03-25 1988-04-27 Merck Sharp & Dohme Therapeutic agents
AU638264B2 (en) * 1989-08-10 1993-06-24 Aventis Inc. Cyclic neurokinin a antagonists

Also Published As

Publication number Publication date
IE913831A1 (en) 1992-05-22
CA2054667A1 (en) 1992-05-03
HUT61582A (en) 1993-01-28
ZA918717B (en) 1992-08-26
EP0484719A2 (en) 1992-05-13
PT99384A (en) 1992-09-30
JPH04300895A (en) 1992-10-23
DE4034829A1 (en) 1992-05-07
KR920009846A (en) 1992-06-25
HU913450D0 (en) 1992-01-28
EP0484719A3 (en) 1993-05-19
AU8676291A (en) 1992-05-07

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