CS331491A3 - Cyclopeptides, process of their preparation and pharmaceuticals based thereon - Google Patents
Cyclopeptides, process of their preparation and pharmaceuticals based thereonInfo
- Publication number
- CS331491A3 CS331491A3 CS913314A CS331491A CS331491A3 CS 331491 A3 CS331491 A3 CS 331491A3 CS 913314 A CS913314 A CS 913314A CS 331491 A CS331491 A CS 331491A CS 331491 A3 CS331491 A3 CS 331491A3
- Authority
- CS
- Czechoslovakia
- Prior art keywords
- cyclopeptides
- preparation
- pharmaceuticals based
- pharmaceuticals
- Prior art date
Links
- 102000001189 Cyclic Peptides Human genes 0.000 title 1
- 108010069514 Cyclic Peptides Proteins 0.000 title 1
- 239000003814 drug Substances 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/50—Cyclic peptides containing at least one abnormal peptide link
- C07K7/52—Cyclic peptides containing at least one abnormal peptide link with only normal peptide links in the ring
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
- C07K7/22—Tachykinins, e.g. Eledoisins, Substance P; Related peptides
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/08—Bronchodilators
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Chemical & Material Sciences (AREA)
- Public Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Pain & Pain Management (AREA)
- Biochemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Molecular Biology (AREA)
- Genetics & Genomics (AREA)
- Biophysics (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Rheumatology (AREA)
- Neurosurgery (AREA)
- Cardiology (AREA)
- Biomedical Technology (AREA)
- Heart & Thoracic Surgery (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4034829A DE4034829A1 (en) | 1990-11-02 | 1990-11-02 | CYCLOPEPTIDE |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CS331491A3 true CS331491A3 (en) | 1992-05-13 |
Family
ID=6417499
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CS913314A CS331491A3 (en) | 1990-11-02 | 1991-11-01 | Cyclopeptides, process of their preparation and pharmaceuticals based thereon |
Country Status (11)
| Country | Link |
|---|---|
| EP (1) | EP0484719A3 (en) |
| JP (1) | JPH04300895A (en) |
| KR (1) | KR920009846A (en) |
| AU (1) | AU8676291A (en) |
| CA (1) | CA2054667A1 (en) |
| CS (1) | CS331491A3 (en) |
| DE (1) | DE4034829A1 (en) |
| HU (1) | HUT61582A (en) |
| IE (1) | IE913831A1 (en) |
| PT (1) | PT99384A (en) |
| ZA (1) | ZA918717B (en) |
Families Citing this family (21)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| ATE195867T1 (en) | 1991-09-20 | 2000-09-15 | Glaxo Group Ltd | NEW MEDICAL INDICATION FOR TACHYKININ ANTAGONISTS |
| GB9620819D0 (en) * | 1996-10-05 | 1996-11-20 | Zeneca Ltd | Chemical compounds |
| GB9702377D0 (en) * | 1996-02-23 | 1997-03-26 | Zeneca Ltd | Peptide derivatives |
| WO1997046578A1 (en) | 1996-06-07 | 1997-12-11 | Zeneca Limited | Peptide derivatives |
| GB9621836D0 (en) | 1996-10-19 | 1996-12-11 | Zeneca Ltd | Peptide compounds |
| GB9624562D0 (en) | 1996-11-27 | 1997-01-15 | Zeneca Ltd | Peptide derivatives |
| KR100408624B1 (en) * | 2000-10-06 | 2003-12-06 | 엘지전선 주식회사 | Poly vinyl chloride insulator composition for wire and cable |
| JP2010516734A (en) | 2007-01-24 | 2010-05-20 | グラクソ グループ リミテッド | 3,5-diamino-6- (2,3-dichlorophenyl) -1,2,4-triazine or R (-)-2,4-diamino-5- (2,3-dichlorophenyl) -6-fluoromethylpyrimidine A pharmaceutical composition comprising |
| UA105182C2 (en) | 2008-07-03 | 2014-04-25 | Ньюрексон, Інк. | Benzoxazines, benzothiazines, and related compounds having nos inhibitory activity |
| US9446029B2 (en) | 2010-07-27 | 2016-09-20 | Colorado State University Research Foundation | Use of NK-1 receptor antagonists in management of visceral pain |
| IN2014CN02805A (en) | 2011-10-14 | 2015-07-03 | Bristol Myers Squibb Co | |
| CN103974938B (en) | 2011-10-14 | 2016-11-09 | 百时美施贵宝公司 | The tetrahydro isoquinoline compound being substituted as factor XI, plasma thromboplastin antecedent A inhibitor |
| ES2699226T3 (en) | 2011-10-14 | 2019-02-08 | Bristol Myers Squibb Co | Substituted tetrahydroisoquinoline compounds as inhibitors of factor XIa |
| WO2014059214A1 (en) | 2012-10-12 | 2014-04-17 | Bristol-Myers Squibb Company | Guanidine and amine substituted tetrahydroisoquinoline compounds as factor xia inhibitors |
| US9315519B2 (en) | 2012-10-12 | 2016-04-19 | Bristol-Myers Squibb Company | Guanidine substituted tetrahydroisoquinoline compounds as factor XIa inhibitors |
| JP6154473B2 (en) | 2012-10-12 | 2017-06-28 | ブリストル−マイヤーズ スクイブ カンパニーＢｒｉｓｔｏｌ−Ｍｙｅｒｓ Ｓｑｕｉｂｂ Ｃｏｍｐａｎｙ | Crystal form of factor XIa inhibitor |
| ES2712699T3 (en) | 2013-03-25 | 2019-05-14 | Bristol Myers Squibb Co | Tetrahydroisoquinolines containing substituted azoles as inhibitors of factor XIa |
| TWI688564B (en) | 2014-01-31 | 2020-03-21 | 美商必治妥美雅史谷比公司 | Macrocycles with hetrocyclic p2' groups as factor xia inhibitors |
| NO2760821T3 (en) | 2014-01-31 | 2018-03-10 | ||
| WO2016036893A1 (en) | 2014-09-04 | 2016-03-10 | Bristol-Myers Squibb Company | Diamide macrocycles that are fxia inhibitors |
| US9453018B2 (en) | 2014-10-01 | 2016-09-27 | Bristol-Myers Squibb Company | Pyrimidinones as factor XIa inhibitors |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB8807246D0 (en) * | 1988-03-25 | 1988-04-27 | Merck Sharp & Dohme | Therapeutic agents |
| AU638264B2 (en) * | 1989-08-10 | 1993-06-24 | Aventis Inc. | Cyclic neurokinin a antagonists |
-
1990
- 1990-11-02 DE DE4034829A patent/DE4034829A1/en not_active Withdrawn
-
1991
- 1991-10-19 EP EP19910117864 patent/EP0484719A3/en not_active Withdrawn
- 1991-10-25 AU AU86762/91A patent/AU8676291A/en not_active Abandoned
- 1991-10-29 KR KR1019910019015A patent/KR920009846A/en not_active Withdrawn
- 1991-10-30 PT PT99384A patent/PT99384A/en not_active Application Discontinuation
- 1991-10-31 CA CA002054667A patent/CA2054667A1/en not_active Abandoned
- 1991-11-01 JP JP3349287A patent/JPH04300895A/en active Pending
- 1991-11-01 HU HU913450A patent/HUT61582A/en unknown
- 1991-11-01 ZA ZA918717A patent/ZA918717B/en unknown
- 1991-11-01 CS CS913314A patent/CS331491A3/en unknown
- 1991-11-01 IE IE383191A patent/IE913831A1/en not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| ZA918717B (en) | 1992-08-26 |
| AU8676291A (en) | 1992-05-07 |
| JPH04300895A (en) | 1992-10-23 |
| EP0484719A2 (en) | 1992-05-13 |
| EP0484719A3 (en) | 1993-05-19 |
| KR920009846A (en) | 1992-06-25 |
| HU913450D0 (en) | 1992-01-28 |
| CA2054667A1 (en) | 1992-05-03 |
| HUT61582A (en) | 1993-01-28 |
| DE4034829A1 (en) | 1992-05-07 |
| PT99384A (en) | 1992-09-30 |
| IE913831A1 (en) | 1992-05-22 |
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