CS193563B2 - Process for preparing steric uniform cis-and trans-5,6-alkylen-5,6-dihydropyrimidin-4/3h/-ones - Google Patents

Process for preparing steric uniform cis-and trans-5,6-alkylen-5,6-dihydropyrimidin-4/3h/-ones

Info

Publication number
CS193563B2
CS193563B2 CS766408A CS640876A CS193563B2 CS 193563 B2 CS193563 B2 CS 193563B2 CS 766408 A CS766408 A CS 766408A CS 640876 A CS640876 A CS 640876A CS 193563 B2 CS193563 B2 CS 193563B2
Authority
CS
Czechoslovakia
Prior art keywords
dihydropyrimidin
alkylen
trans
ones
cis
Prior art date
Application number
CS766408A
Other languages
Czech (cs)
English (en)
Inventor
Gabor Bernath
Lajos Gera
Gyoergy Goendoes
Zoltan Ecsery
Judit Hermann
Matyas Szentivanyi
Erzsebet Janvari
Original Assignee
Chinoin Gyogyszer Es Vegyeszet
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszet filed Critical Chinoin Gyogyszer Es Vegyeszet
Publication of CS193563B2 publication Critical patent/CS193563B2/cs

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/91—Oxygen atoms with aryl or aralkyl radicals attached in position 2 or 3
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P23/00—Anaesthetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C07D239/88—Oxygen atoms
    • C07D239/90—Oxygen atoms with acyclic radicals attached in position 2 or 3

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Anesthesiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
CS766408A 1975-10-03 1976-10-04 Process for preparing steric uniform cis-and trans-5,6-alkylen-5,6-dihydropyrimidin-4/3h/-ones CS193563B2 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU75CI00001614A HU172460B (hu) 1975-10-03 1975-10-03 Sposob poluchenija novykh proizvodnykh 5,6-digidro-3h-pirimidin-4-ona

Publications (1)

Publication Number Publication Date
CS193563B2 true CS193563B2 (en) 1979-10-31

Family

ID=10994582

Family Applications (1)

Application Number Title Priority Date Filing Date
CS766408A CS193563B2 (en) 1975-10-03 1976-10-04 Process for preparing steric uniform cis-and trans-5,6-alkylen-5,6-dihydropyrimidin-4/3h/-ones

Country Status (14)

Country Link
US (1) US4113868A (pm)
JP (1) JPS5257185A (pm)
AU (1) AU507798B2 (pm)
CH (2) CH626072A5 (pm)
CS (1) CS193563B2 (pm)
DD (1) DD127444A1 (pm)
DE (1) DE2643384A1 (pm)
FI (1) FI66603C (pm)
FR (1) FR2326193A1 (pm)
GB (1) GB1559985A (pm)
HU (1) HU172460B (pm)
IL (1) IL50577A (pm)
PL (2) PL110639B1 (pm)
SU (1) SU627752A3 (pm)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU179687B (en) * 1978-11-01 1982-11-29 Chinoin Gyogyszer Es Vegyeszet Process for producing 5,6,7,8-- etrahydro-4-bracket-3h-bracket closed-quinasolinones
US4814335A (en) * 1982-12-30 1989-03-21 Biomeasure, Incorporated Antiviral compounds
JPS59210071A (ja) * 1982-12-30 1984-11-28 バイオメジヤ−・インコ−ポレ−テツド 抗ウイルス作用を有する化合物
US5629264A (en) * 1995-03-23 1997-05-13 Rohm And Haas Company 2-aryl-5,6-dihydropyrimidinones and herbicidal use thereof
AU2004200A (en) * 1999-01-14 2000-08-01 Meiji Seika Kaisha Ltd. Poly(adp-ribose) polymerase inhibitors consisting of pyrimidine derivatives
DE10123163A1 (de) * 2001-05-09 2003-01-16 Gruenenthal Gmbh Substituierte Cyclohexan-1,4-diaminderivate
AUPS019702A0 (en) * 2002-01-29 2002-02-21 Fujisawa Pharmaceutical Co., Ltd. Condensed heterocyclic compounds

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3047462A (en) * 1959-03-06 1962-07-31 Lab Jacques Logeais Soc D Expl Quinazolone anti-inflammatory composition
GB1233943A (pm) * 1968-10-31 1971-06-03
US3696102A (en) * 1970-03-09 1972-10-03 Pfizer & Co C Process for the synthesis of substituted quinazolin-4-ones
US3996227A (en) * 1971-07-08 1976-12-07 Sandoz, Inc. 7-Methyl-1-isopropyl-4-phenyl-5,6,7,8-tetrahydro-2(1H)-quinazolinone
US3945960A (en) * 1973-07-26 1976-03-23 Sandoz, Inc. Antiinflammatory and analgesic cycloalkano-pyrimidin-2(1H)-ones
US3994894A (en) * 1975-01-08 1976-11-30 Sandoz, Inc. Cyclopentano[1,2-c]pyrimidin-2(1H)-ones

Also Published As

Publication number Publication date
AU1820376A (en) 1978-04-06
GB1559985A (en) 1980-01-30
CH626074A5 (pm) 1981-10-30
PL111251B1 (en) 1980-08-30
FR2326193A1 (fr) 1977-04-29
DD127444A1 (pm) 1977-09-21
FI762806A7 (pm) 1977-04-04
US4113868A (en) 1978-09-12
PL110639B1 (en) 1980-07-31
IL50577A (en) 1979-12-30
FI66603C (fi) 1984-11-12
DE2643384A1 (de) 1977-06-02
AU507798B2 (en) 1980-02-28
IL50577A0 (en) 1976-11-30
CH626072A5 (pm) 1981-10-30
JPS5257185A (en) 1977-05-11
HU172460B (hu) 1978-09-28
FI66603B (fi) 1984-07-31
SU627752A3 (ru) 1978-10-05
FR2326193B1 (pm) 1979-09-28

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