CO5180549A1 - DERIVATIVES OF 1-AMINO ETHYLINDOL, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICS - Google Patents
DERIVATIVES OF 1-AMINO ETHYLINDOL, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICSInfo
- Publication number
- CO5180549A1 CO5180549A1 CO00026489A CO00026489A CO5180549A1 CO 5180549 A1 CO5180549 A1 CO 5180549A1 CO 00026489 A CO00026489 A CO 00026489A CO 00026489 A CO00026489 A CO 00026489A CO 5180549 A1 CO5180549 A1 CO 5180549A1
- Authority
- CO
- Colombia
- Prior art keywords
- hydrogen atom
- ethylindol
- therapeutics
- derivatives
- amino
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/08—Indoles; Hydrogenated indoles with only hydrogen atoms or radicals containing only hydrogen and carbon atoms, directly attached to carbon atoms of the hetero ring
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/10—Drugs for disorders of the urinary system of the bladder
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/06—Antimigraine agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/04—Indoles; Hydrogenated indoles
- C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- General Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Cardiology (AREA)
- Vascular Medicine (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Urology & Nephrology (AREA)
- Otolaryngology (AREA)
- Pulmonology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Indole Compounds (AREA)
Abstract
Compuesto de fórmula (I)<EMI FILE="00026489_1" ID="1" IMF=JPEG >en la cual:A representa un átomo de hidrógeno, un halógeno o un hidroxi,B y D representan, independientemente entre sí, un átomo de hidrógeno o un grupo C1-3 alquilo,R1 representa un átomo de hidrógeno, un grupo C1-4 alquilo, C1-2 fluoroalquilo o C1-2 perfluoroalquilo,R2 representa un átomo de hidrógeno, un halógeno, un grupo C1-6 alquilo, C3-6 cicloalquilo, C1-2 perfluoroalquilo, C1-2 perfluoroalquilo o un fenilo,R3 y R4 representan, independientemente entre sí, un átomo de hidrógeno, un halógeno o un grupo C1-6 alquilo,R5 y R6 representan, independientemente entre sí, un átomo de hidrógeno, un grupo C1-6; alquilo o C1-2 fluoroalquilo, o R5 y R6, juntos, forman una cadena C2-7alquileno, y sus sales.Compound of formula (I) <EMI FILE = "00026489_1" ID = "1" MFI = JPEG> in which: A represents a hydrogen atom, a halogen or a hydroxy, B and D represent, independently from each other, an atom of hydrogen or a C1-3 alkyl group, R1 represents a hydrogen atom, a C1-4 alkyl, C1-2 fluoroalkyl or C1-2 perfluoroalkyl group, R2 represents a hydrogen atom, a halogen, a C1-6 alkyl group , C3-6 cycloalkyl, C1-2 perfluoroalkyl, C1-2 perfluoroalkyl or a phenyl, R3 and R4 independently represent each other, a hydrogen atom, a halogen or a C1-6 alkyl group, R5 and R6 independently represent yes, a hydrogen atom, a C1-6 group; alkyl or C1-2 fluoroalkyl, or R5 and R6, together, form a C2-7alkylene chain, and salts thereof.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
FR9904577A FR2792316B1 (en) | 1999-04-13 | 1999-04-13 | 1-AMINOETHYLINDOLE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
Publications (1)
Publication Number | Publication Date |
---|---|
CO5180549A1 true CO5180549A1 (en) | 2002-07-30 |
Family
ID=9544316
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CO00026489A CO5180549A1 (en) | 1999-04-13 | 2000-04-11 | DERIVATIVES OF 1-AMINO ETHYLINDOL, ITS PREPARATION AND ITS APPLICATION IN THERAPEUTICS |
Country Status (7)
Country | Link |
---|---|
AR (1) | AR023451A1 (en) |
AU (1) | AU3971400A (en) |
CO (1) | CO5180549A1 (en) |
FR (1) | FR2792316B1 (en) |
PE (1) | PE20010041A1 (en) |
UY (1) | UY26102A1 (en) |
WO (1) | WO2000061554A1 (en) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
AR077405A1 (en) | 2009-07-10 | 2011-08-24 | Sanofi Aventis | DERIVATIVES OF INDOL INHIBITORS OF HSP90, COMPOSITIONS THAT CONTAIN THEM AND USE OF THE SAME FOR THE TREATMENT OF CANCER |
Family Cites Families (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
FR2752840A1 (en) * | 1996-08-29 | 1998-03-06 | Synthelabo | 7-Amino ethyl benzothiophene derivatives |
FR2752839B1 (en) * | 1996-08-29 | 1998-10-09 | Synthelabo | BENZOFURANE DERIVATIVES, THEIR PREPARATION AND THEIR THERAPEUTIC APPLICATION |
-
1999
- 1999-04-13 FR FR9904577A patent/FR2792316B1/en not_active Expired - Fee Related
-
2000
- 2000-04-10 UY UY26102A patent/UY26102A1/en not_active Application Discontinuation
- 2000-04-11 AU AU39714/00A patent/AU3971400A/en not_active Abandoned
- 2000-04-11 CO CO00026489A patent/CO5180549A1/en not_active Application Discontinuation
- 2000-04-11 WO PCT/FR2000/000922 patent/WO2000061554A1/en active Application Filing
- 2000-04-12 AR ARP000101669A patent/AR023451A1/en unknown
- 2000-04-13 PE PE2000000344A patent/PE20010041A1/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO2000061554A1 (en) | 2000-10-19 |
AU3971400A (en) | 2000-11-14 |
FR2792316B1 (en) | 2001-06-22 |
UY26102A1 (en) | 2000-10-31 |
AR023451A1 (en) | 2002-09-04 |
FR2792316A1 (en) | 2000-10-20 |
PE20010041A1 (en) | 2001-04-12 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FA | Application withdrawn |