CO4290359A1 - Metodo para tratar la alopecia androgenica con inhibidores 5-alfa-reductasa - Google Patents

Metodo para tratar la alopecia androgenica con inhibidores 5-alfa-reductasa

Info

Publication number
CO4290359A1
CO4290359A1 CO94046672A CO94046672A CO4290359A1 CO 4290359 A1 CO4290359 A1 CO 4290359A1 CO 94046672 A CO94046672 A CO 94046672A CO 94046672 A CO94046672 A CO 94046672A CO 4290359 A1 CO4290359 A1 CO 4290359A1
Authority
CO
Colombia
Prior art keywords
alpha
androgenic alopecia
reductase inhibitors
treating androgenic
treating
Prior art date
Application number
CO94046672A
Other languages
English (en)
Inventor
Glenn J Gormley
Keith D Kaufman
Elizabeth Stoner
Joanne Waldstricher
Original Assignee
Merck & Co Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22482390&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CO4290359(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Merck & Co Inc filed Critical Merck & Co Inc
Publication of CO4290359A1 publication Critical patent/CO4290359A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47Quinolines; Isoquinolines
    • A61K31/473Quinolines; Isoquinolines ortho- or peri-condensed with carbocyclic ring systems, e.g. acridines, phenanthridines
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K8/00Cosmetics or similar toiletry preparations
    • A61K8/18Cosmetics or similar toiletry preparations characterised by the composition
    • A61K8/30Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
    • A61K8/63Steroids; Derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00Preparations for care of the hair
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00Preparations for affecting hair growth
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q7/00Preparations for affecting hair growth
    • A61Q7/02Preparations for inhibiting or slowing hair growth
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/74Biological properties of particular ingredients
    • A61K2800/78Enzyme modulators, e.g. Enzyme agonists
    • A61K2800/782Enzyme inhibitors; Enzyme antagonists
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K2800/00Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
    • A61K2800/80Process related aspects concerning the preparation of the cosmetic composition or the storage or application thereof
    • A61K2800/92Oral administration
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q19/00Preparations for care of the skin
    • A61Q19/10Washing or bathing preparations
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61QSPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
    • A61Q5/00Preparations for care of the hair
    • A61Q5/02Preparations for cleaning the hair

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Dermatology (AREA)
  • Birds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Cosmetics (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Steroid Compounds (AREA)

Abstract

REIVINDICACION NUMERO UN METODO PARA TRATAR LA ALOPECIA ANDROGENICA, QUE SUPONE ADMINISTRAR A UNA PERSONA QUE NECESITA TAL TRATAMIENTO, UN INHIBIDOR 5-ALFA-REDUCTASA 2, EN UNA CANTIDAD DOSIFICIADA POR DEBAJO DE LOS 5.0 mg/ dia.
CO94046672A 1993-10-15 1994-10-12 Metodo para tratar la alopecia androgenica con inhibidores 5-alfa-reductasa CO4290359A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US13852093A 1993-10-15 1993-10-15
US08/214,905 US5547957A (en) 1993-10-15 1994-03-17 Method of treating androgenic alopecia with 5-α reductase inhibitors

Publications (1)

Publication Number Publication Date
CO4290359A1 true CO4290359A1 (es) 1996-04-17

Family

ID=22482390

Family Applications (1)

Application Number Title Priority Date Filing Date
CO94046672A CO4290359A1 (es) 1993-10-15 1994-10-12 Metodo para tratar la alopecia androgenica con inhibidores 5-alfa-reductasa

Country Status (8)

Country Link
US (4) US5547957A (es)
EP (1) EP0776664A2 (es)
KR (1) KR100375083B1 (es)
CO (1) CO4290359A1 (es)
HK (1) HK1000933A1 (es)
MY (2) MY123960A (es)
YU (1) YU49026B (es)
ZA (1) ZA948064B (es)

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TW382595B (en) * 1993-10-15 2000-02-21 Merck & Co Inc Pharmaceutical composition for use in arresting and reversing androgenic alopecia
US5547957A (en) * 1993-10-15 1996-08-20 Merck & Co., Inc. Method of treating androgenic alopecia with 5-α reductase inhibitors
US5739137A (en) * 1993-10-21 1998-04-14 Merck & Co., Inc. 16-substituted-4-aza-3-oxo-androstane as 5-alpha-reductase isozyme 1 inhibitors
USRE39056E1 (en) 1995-09-15 2006-04-04 Merck & Co, Inc. 4-Azasteroids for treatment of hyperandrogenic conditions
WO1997014418A1 (en) * 1995-10-19 1997-04-24 Merck & Co., Inc. 16-substituted-6-aza-steroid 5-alpha-reductase inhibitors
US5679378A (en) * 1995-12-18 1997-10-21 Olim Industries Of Israel, North America, Ltd. Method and material for hair therapy
US5935968A (en) 1997-03-17 1999-08-10 Merck & Co., Inc. Methods for treating polycystic ovary syndrome
US6348348B1 (en) * 1998-04-07 2002-02-19 The Carnegie Institution Of Washington Human hairless gene and protein
US6645974B2 (en) 2001-07-31 2003-11-11 Merck & Co., Inc. Androgen receptor modulators and methods for use thereof
EP1451144B1 (en) 2001-10-31 2010-09-01 Coreana Cosmetics Co., Ltd. Compositions for treating acne comprising phytandiol amine
GB0213745D0 (en) * 2002-06-14 2002-07-24 Univ Edinburgh Enzyme
US7790706B2 (en) * 2002-06-14 2010-09-07 The University Of Edinburgh Treatment of inflammation with 5α reduced metabolites
IL156670A0 (en) * 2003-06-26 2004-01-04 Zvi Zolotariov Aloe suppositories
ATE406376T1 (de) * 2003-07-03 2008-09-15 Cipla Ltd Verfahren zur herstellung von finasterid form i
US20050136015A1 (en) * 2003-12-17 2005-06-23 McKie Derrick B. Topical use of halosalicylic acid derivatives
JP2007522201A (ja) * 2004-02-12 2007-08-09 ワーナー−ランバート カンパニー リミテッド ライアビリティー カンパニー 毛成長の刺激方法
GB0407329D0 (en) * 2004-03-31 2004-05-05 Danisco Process
US7979110B1 (en) * 2004-09-23 2011-07-12 Orbital Research Inc. Method for accurate placement of electrodes
US7998970B2 (en) 2004-12-03 2011-08-16 Proteosys Ag Use of finasteride, dutasteride and related compounds for the prevention or treatment of neurologically-associated disorders
US20060263452A1 (en) * 2005-05-17 2006-11-23 Alwyn Dowell Topical composition containing essential oils
US20070167899A1 (en) * 2006-01-19 2007-07-19 Strom Randy A Compression apparatus and method for stimulating hair growth
US20090076058A1 (en) * 2007-09-17 2009-03-19 Protia, Llc Deuterium-enriched finasteride
US20090203628A1 (en) * 2008-02-12 2009-08-13 Jan Marini Composition, Method And Kit For Treating Skin Disorders And Improving Skin Condition
US20090233954A1 (en) * 2008-03-12 2009-09-17 Goren Andy Ofer Methods and systems for prognosis of a patient's response to treatment of androgenetic skin disorders
EP2378872A4 (en) 2008-12-18 2012-05-16 B Eugene Guthery TREATMENT PLAN FOR ACNE VULGARIS
FR2954124B1 (fr) * 2009-12-18 2012-04-06 Fabre Pierre Dermo Cosmetique Utilisation du 2,3-dihydroxypropyl dodecanoate pour le traitement de la seborrhee
BR112013002697A2 (pt) * 2010-08-05 2016-05-31 Legacy Healthcare Holding Ltd método para estimular o crescimento do cabelo
US8604047B2 (en) * 2010-08-10 2013-12-10 Elorac, Inc. Method and composition for treating nodulocystic and conglobate acne vulgaris
EP2782582A4 (en) * 2011-11-25 2016-09-28 Adrianna Janell Jackson OIL COMPOSITIONS AND METHODS FOR PROMOTING HAIR GROWTH AND / OR PREVENTING HAIR LOSS
KR102064488B1 (ko) * 2019-04-18 2020-01-13 주식회사 엠진 홍삼 추출물 등을 이용한 발모 촉진 또는 탈모 억제용 조성물
KR102221365B1 (ko) 2019-05-07 2021-03-02 (주)케어젠 트롤록스-펩타이드 결합체 및 그의 용도

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Also Published As

Publication number Publication date
US6174892B1 (en) 2001-01-16
YU58394A (en) 1999-11-22
MY123960A (en) 2006-06-30
HK1000933A1 (en) 1998-05-08
MY138240A (en) 2009-05-29
EP0776664A3 (es) 1997-06-11
KR960704555A (ko) 1996-10-09
US20020042425A1 (en) 2002-04-11
EP0776664A2 (en) 1997-06-04
US5547957A (en) 1996-08-20
US6355649B1 (en) 2002-03-12
ZA948064B (en) 1995-06-06
YU49026B (sh) 2003-07-07
KR100375083B1 (ko) 2003-06-09

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