CO2023012917A2 - Compuestos con propiedades de sensación refrescante - Google Patents
Compuestos con propiedades de sensación refrescanteInfo
- Publication number
- CO2023012917A2 CO2023012917A2 CONC2023/0012917A CO2023012917A CO2023012917A2 CO 2023012917 A2 CO2023012917 A2 CO 2023012917A2 CO 2023012917 A CO2023012917 A CO 2023012917A CO 2023012917 A2 CO2023012917 A2 CO 2023012917A2
- Authority
- CO
- Colombia
- Prior art keywords
- compounds
- cooling sensation
- sensation properties
- properties
- cooling
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 230000035597 cooling sensation Effects 0.000 title 1
- 102000003610 TRPM8 Human genes 0.000 abstract 1
- 101150111302 Trpm8 gene Proteins 0.000 abstract 1
- 238000001816 cooling Methods 0.000 abstract 1
- 210000004400 mucous membrane Anatomy 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K8/00—Cosmetics or similar toiletry preparations
- A61K8/18—Cosmetics or similar toiletry preparations characterised by the composition
- A61K8/30—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds
- A61K8/49—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds
- A61K8/494—Cosmetics or similar toiletry preparations characterised by the composition containing organic compounds containing heterocyclic compounds with more than one nitrogen as the only hetero atom
- A61K8/4946—Imidazoles or their condensed derivatives, e.g. benzimidazoles
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
- A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61Q—SPECIFIC USE OF COSMETICS OR SIMILAR TOILETRY PREPARATIONS
- A61Q11/00—Preparations for care of the teeth, of the oral cavity or of dentures; Dentifrices, e.g. toothpastes; Mouth rinses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K2800/00—Properties of cosmetic compositions or active ingredients thereof or formulation aids used therein and process related aspects
- A61K2800/20—Chemical, physico-chemical or functional or structural properties of the composition as a whole
- A61K2800/24—Thermal properties
- A61K2800/244—Endothermic; Cooling; Cooling sensation
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Epidemiology (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Oral & Maxillofacial Surgery (AREA)
- Birds (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Cosmetics (AREA)
Abstract
La presente invención se relaciona con moduladores de TRPM8 de fórmula (I) para lograr un efecto refrescante en la piel y las mucosas.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GBGB2105661.9A GB202105661D0 (en) | 2021-04-21 | 2021-04-21 | Organic compounds |
PCT/EP2022/060485 WO2022223661A1 (en) | 2021-04-21 | 2022-04-21 | Compounds with cooling sensation properties |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2023012917A2 true CO2023012917A2 (es) | 2023-10-19 |
Family
ID=76377639
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2023/0012917A CO2023012917A2 (es) | 2021-04-21 | 2023-09-28 | Compuestos con propiedades de sensación refrescante |
Country Status (7)
Country | Link |
---|---|
US (1) | US20240197604A1 (es) |
EP (1) | EP4326711A1 (es) |
BR (1) | BR112023018788A2 (es) |
CO (1) | CO2023012917A2 (es) |
GB (1) | GB202105661D0 (es) |
MX (1) | MX2023010891A (es) |
WO (1) | WO2022223661A1 (es) |
Family Cites Families (14)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US3988433A (en) | 1973-08-10 | 1976-10-26 | The Procter & Gamble Company | Oral compositions for preventing or removing stains from teeth |
US4083955A (en) | 1975-04-02 | 1978-04-11 | The Procter & Gamble Company | Processes and compositions for remineralization of dental enamel |
US4528180A (en) | 1983-03-01 | 1985-07-09 | Schaeffer Hans A | Dental preparation, article and method for storage and delivery thereof |
US4849213A (en) | 1983-03-01 | 1989-07-18 | Schaeffer Hans A | Dental preparation, article and method for storage and delivery therof |
US5198220A (en) | 1989-11-17 | 1993-03-30 | The Procter & Gamble Company | Sustained release compositions for treating periodontal disease |
US5213790A (en) | 1991-10-23 | 1993-05-25 | The Procter & Gamble Co. | Methods of reducing plaque and gingivitis with reduced staining |
US5145666A (en) | 1991-10-23 | 1992-09-08 | The Proctor & Gamble Co. | Methods of reducing plaque and gingivitis with reduced staining |
US5281410A (en) | 1991-10-23 | 1994-01-25 | The Proctor & Gamble Company | Methods of reducing plaque and gingivitis with reduced staining |
US5242910A (en) | 1992-10-13 | 1993-09-07 | The Procter & Gamble Company | Sustained release compositions for treating periodontal disease |
GB0704163D0 (en) | 2007-03-02 | 2007-04-11 | Quest Int Serv Bv | Compositions comprising a physiological coolant |
MX2011005374A (es) | 2008-11-20 | 2011-06-06 | Procter & Gamble | Composiciones para el cuidado personal que proporcionan una sensacion refrescante mejorada. |
ES2936608T3 (es) | 2017-12-21 | 2023-03-21 | Firmenich & Cie | Composiciones refrescantes y potenciadoras del sabor |
CN114555594A (zh) | 2019-10-17 | 2022-05-27 | 奇华顿股份有限公司 | 作为trmp8调节剂的取代的氮杂环 |
GB202013383D0 (en) * | 2020-08-26 | 2020-10-07 | Givaudan Sa | Process |
-
2021
- 2021-04-21 GB GBGB2105661.9A patent/GB202105661D0/en not_active Ceased
-
2022
- 2022-04-21 BR BR112023018788A patent/BR112023018788A2/pt unknown
- 2022-04-21 US US18/286,525 patent/US20240197604A1/en active Pending
- 2022-04-21 WO PCT/EP2022/060485 patent/WO2022223661A1/en active Application Filing
- 2022-04-21 MX MX2023010891A patent/MX2023010891A/es unknown
- 2022-04-21 EP EP22724058.7A patent/EP4326711A1/en active Pending
-
2023
- 2023-09-28 CO CONC2023/0012917A patent/CO2023012917A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
US20240197604A1 (en) | 2024-06-20 |
EP4326711A1 (en) | 2024-02-28 |
GB202105661D0 (en) | 2021-06-02 |
MX2023010891A (es) | 2023-09-27 |
WO2022223661A1 (en) | 2022-10-27 |
BR112023018788A2 (pt) | 2023-12-12 |
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