CO2022017895A2 - Cysteine protease inhibitors and their methods of use - Google Patents

Cysteine protease inhibitors and their methods of use

Info

Publication number
CO2022017895A2
CO2022017895A2 CONC2022/0017895A CO2022017895A CO2022017895A2 CO 2022017895 A2 CO2022017895 A2 CO 2022017895A2 CO 2022017895 A CO2022017895 A CO 2022017895A CO 2022017895 A2 CO2022017895 A2 CO 2022017895A2
Authority
CO
Colombia
Prior art keywords
methods
protease inhibitors
cysteine protease
compounds
active
Prior art date
Application number
CONC2022/0017895A
Other languages
Spanish (es)
Inventor
Lee D Arnold
Andy Jennings
Walter Keung
Original Assignee
Pardes Biosciences Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from PCT/US2021/036638 external-priority patent/WO2021252644A1/en
Application filed by Pardes Biosciences Inc filed Critical Pardes Biosciences Inc
Publication of CO2022017895A2 publication Critical patent/CO2022017895A2/en

Links

Landscapes

  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Peptides Or Proteins (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Se proveen compuestos de la Fórmula II con cargas activas (“warheads”) y su uso para el tratamiento de enfermedades y trastornos clínicos tales como las infecciones virales; también se proveen composiciones farmacéuticas y métodos para preparar distintos compuestos con carga activa; se observa que los compuestos inhiben proteasas tales como la proteasa tipo 3C, CL- o 3CL.Compounds of Formula II with active charges ("warheads") and their use for the treatment of diseases and clinical disorders such as viral infections are provided; Pharmaceutical compositions and methods for preparing various compounds with active charge are also provided; The compounds are shown to inhibit proteases such as type 3C, CL- or 3CL protease.

CONC2022/0017895A 2020-06-09 2022-12-09 Cysteine protease inhibitors and their methods of use CO2022017895A2 (en)

Applications Claiming Priority (11)

Application Number Priority Date Filing Date Title
US202063036866P 2020-06-09 2020-06-09
US202063039297P 2020-06-15 2020-06-15
US202063067669P 2020-08-19 2020-08-19
US202063091630P 2020-10-14 2020-10-14
US202063129018P 2020-12-22 2020-12-22
US202163171675P 2021-04-07 2021-04-07
US202163172478P 2021-04-08 2021-04-08
US202163172146P 2021-04-08 2021-04-08
US202163179128P 2021-04-23 2021-04-23
US202163195460P 2021-06-01 2021-06-01
PCT/US2021/036638 WO2021252644A1 (en) 2020-06-09 2021-06-09 Inhibitors of cysteine proteases and methods of use thereof

Publications (1)

Publication Number Publication Date
CO2022017895A2 true CO2022017895A2 (en) 2023-03-07

Family

ID=85382440

Family Applications (1)

Application Number Title Priority Date Filing Date
CONC2022/0017895A CO2022017895A2 (en) 2020-06-09 2022-12-09 Cysteine protease inhibitors and their methods of use

Country Status (1)

Country Link
CO (1) CO2022017895A2 (en)

Similar Documents

Publication Publication Date Title
DOP2022000278A (en) CYSTEINE PROTEASE INHIBITORS AND THEIR METHODS OF USE
ECSP20069418A (en) HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS
DOP2021000019A (en) INFLAMASOME INHIBITORS NLRP3
UY38979A (en) TETRAHYDROFURANS REPLACED AS SODIUM CHANNEL MODULATORS
CL2021000972A1 (en) Protein tyrosine phosphatase inhibitors
EA201800064A1 (en) 1,1,1-TRIFTOR-3-HYDROXYPROPAN-2-IL CARBAMATE DERIVATIVES AND 1,1,1-TRIFTOR-4-HYDROXYBUTAN-2-IL CARBAMATE DERIVATIVES AS MIGL INHIBITORS
EA202092490A1 (en) METHYL-MODIFYING ENZYMES MODULATORS, COMPOSITIONS AND THEIR APPLICATION
UY30617A1 (en) SUBSTITUTED CARBAMATE DERIVATIVES OF 1- (9 - {[(2R) -2- {4-HIDROXI-3 - [(METILSULFONIL) AMINO] FENIL} ETIL] AMINO} NONIL) PIPERIDIN-4-ILO, ITS SALTS AND SOLVATES PHARMACEUTICALLY ACCEPTABLE AND APPLICATIONS
ECSP21026485A (en) PYRIDAZINONES AND THEIR METHODS OF USE
DOP2019000076A (en) DERIVATIVES OF CHROMANO, ISOCROMANO AND DIHYDROISOBENZOFURANOS AS NEGATIVE ALOSTERIC MODULATORS OF mGluR2, COMPOSITIONS AND ITS USE
CO2022000749A2 (en) Heterocyclic monoacylglycerol lipase (MAGL) inhibitors
EA202191968A1 (en) NEW SUBSTITUTED SULFONYLUREA DERIVATIVES
EA202091604A1 (en) INHIBITION OF THE ION CHANNEL A1 WITH A TRANSITOR RECEPTOR POTENTIAL
BR112022010181A2 (en) TRIHETEROCYCLIC COMPOUND AS A JAK INHIBITOR AND USE OF IT
CL2022002386A1 (en) Fused amino pyrimidine compounds
ECSP23017158A (en) HETEROARYL-SUBSTITUTED SPIROPIPERIDINYL DERIVATIVES AND PHARMACEUTICAL USES THEREOF
CL2022001741A1 (en) Cyclic compounds and methods of using same
EA201891319A1 (en) COMPOUNDS OF ALKYDYDYDROCHINOLINSULPHONAMIDE
UY37745A (en) BICYCLIC COMPOUNDS 5.6 FUSIONATES AND COMPOSITIONS FOR THE TREATMENT OF PARASITARY DISEASES
CO2022017895A2 (en) Cysteine protease inhibitors and their methods of use
BR112022001866A2 (en) Hybrid amide derivatives of amphotericin b
EA202192111A1 (en) NEW TRITERPENE DERIVATIVES AS HIV INHIBITORS
EA201992436A1 (en) COMPOSITIONS WITH IMPROVED STABILITY AND BIOAVAILABILITY FOR THE INTRODUCTION OF (E) -2,6-DIALCOXY OF 4-SUBSTITUTED BENZENESULPHONES
AR114282A1 (en) PROTEIN SECRETION INHIBITORS BASED ON TRIAZACICLODODECANSULFONAMIDE ("TCD")
EA202092344A1 (en) HETEROCYCLIC COMPOUNDS AS IMMUNOMODULATORS