CO2018002046A2 - Nueva composición oral de libreación retardada dual de dexlansoprazol - Google Patents
Nueva composición oral de libreación retardada dual de dexlansoprazolInfo
- Publication number
- CO2018002046A2 CO2018002046A2 CONC2018/0002046A CO2018002046A CO2018002046A2 CO 2018002046 A2 CO2018002046 A2 CO 2018002046A2 CO 2018002046 A CO2018002046 A CO 2018002046A CO 2018002046 A2 CO2018002046 A2 CO 2018002046A2
- Authority
- CO
- Colombia
- Prior art keywords
- dexlansoprazole
- oral
- pharmaceutically acceptable
- new
- release layer
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5084—Mixtures of one or more drugs in different galenical forms, at least one of which being granules, microcapsules or (coated) microparticles according to A61K9/16 or A61K9/50, e.g. for obtaining a specific release pattern or for combining different drugs
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4427—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
- A61K31/4439—Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. omeprazole
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5026—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5005—Wall or coating material
- A61K9/5021—Organic macromolecular compounds
- A61K9/5036—Polysaccharides, e.g. gums, alginate; Cyclodextrin
- A61K9/5042—Cellulose; Cellulose derivatives, e.g. phthalate or acetate succinate esters of hydroxypropyl methylcellulose
- A61K9/5047—Cellulose ethers containing no ester groups, e.g. hydroxypropyl methylcellulose
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
Abstract
La presente descripción proporciona una composición farmacéutica oral de liberación retardada dual de Dexlansoprazol o sales farmacéuticamente aceptables o formas hidratadas del mismo. La composición farmacéutica de liberación retardada dual descrita puede incorporar dos formulaciones de liberación pulsátil (a) y (b), en donde la formulación (a) puede incluir: (i) una partícula de núcleo que comprende Dexlansoprazol o una sal farmacéuticamente aceptable o un hidrato del mismo, y (ii) una capa de liberación controlada dependiente del pH; y la formulación (b) puede incluir: (i) una partícula de núcleo que comprende Dexlansoprazol o una sal farmacéuticamente aceptable o un hidrato del mismo, (ii) una capa de liberación controlada independiente del pH, y (iii) una capa de liberación controlada dependiente del pH.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
IN2851MU2015 | 2015-07-28 | ||
PCT/IB2016/054467 WO2017017615A1 (en) | 2015-07-28 | 2016-07-27 | Novel dual delayed release oral composition of dexlansoprazole |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2018002046A2 true CO2018002046A2 (es) | 2018-02-28 |
Family
ID=57884420
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2018/0002046A CO2018002046A2 (es) | 2015-07-28 | 2018-02-26 | Nueva composición oral de libreación retardada dual de dexlansoprazol |
Country Status (6)
Country | Link |
---|---|
EP (1) | EP3328364A4 (es) |
BR (1) | BR112018001539A2 (es) |
CL (1) | CL2018000220A1 (es) |
CO (1) | CO2018002046A2 (es) |
PE (1) | PE20181012A1 (es) |
WO (1) | WO2017017615A1 (es) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
CN111991367A (zh) * | 2020-09-21 | 2020-11-27 | 青岛吉达巴尔国际贸易有限公司 | 一种埃索美拉唑镁脉冲微丸胶囊剂及制备方法 |
KR102471545B1 (ko) * | 2020-11-20 | 2022-11-29 | 서울대학교 산학협력단 | 덱스란소프라졸을 유효성분으로 포함하는 pH 의존성 타블렛-인-캡슐 복합제제 및 이의 제조방법 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
WO2010117756A2 (en) * | 2009-03-31 | 2010-10-14 | Dr. Reddy's Laboratories Ltd | Substituted benzimidazole pharmaceutical formulations |
US20120058194A1 (en) * | 2010-08-27 | 2012-03-08 | Navin Vaya | Pharmaceutical formulations comprising substituted benzimidazole derivatives |
WO2013111149A1 (en) * | 2011-12-21 | 2013-08-01 | Hetero Research Foundation | Controlled release solid oral compositions of dexlansoprazole |
-
2016
- 2016-07-27 EP EP16829940.2A patent/EP3328364A4/en not_active Withdrawn
- 2016-07-27 WO PCT/IB2016/054467 patent/WO2017017615A1/en active Application Filing
- 2016-07-27 PE PE2018000128A patent/PE20181012A1/es unknown
- 2016-07-27 BR BR112018001539A patent/BR112018001539A2/pt not_active IP Right Cessation
-
2018
- 2018-01-26 CL CL2018000220A patent/CL2018000220A1/es unknown
- 2018-02-26 CO CONC2018/0002046A patent/CO2018002046A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
BR112018001539A2 (pt) | 2018-09-18 |
EP3328364A1 (en) | 2018-06-06 |
WO2017017615A1 (en) | 2017-02-02 |
EP3328364A4 (en) | 2019-01-02 |
PE20181012A1 (es) | 2018-06-26 |
CL2018000220A1 (es) | 2018-07-20 |
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