CO2017001076A2 - Composiciones farmacéuticas antihiperalgésicas, antialodínicas y antiinflamatorias que contienen pregabalina y meloxicam - Google Patents
Composiciones farmacéuticas antihiperalgésicas, antialodínicas y antiinflamatorias que contienen pregabalina y meloxicamInfo
- Publication number
- CO2017001076A2 CO2017001076A2 CONC2017/0001076A CO2017001076A CO2017001076A2 CO 2017001076 A2 CO2017001076 A2 CO 2017001076A2 CO 2017001076 A CO2017001076 A CO 2017001076A CO 2017001076 A2 CO2017001076 A2 CO 2017001076A2
- Authority
- CO
- Colombia
- Prior art keywords
- antihyperalgesic
- pharmaceutical compositions
- meloxicam
- allodinic
- compositions containing
- Prior art date
Links
- 230000003070 anti-hyperalgesia Effects 0.000 title abstract 3
- 239000008194 pharmaceutical composition Substances 0.000 title abstract 3
- ZRVUJXDFFKFLMG-UHFFFAOYSA-N Meloxicam Chemical compound OC=1C2=CC=CC=C2S(=O)(=O)N(C)C=1C(=O)NC1=NC=C(C)S1 ZRVUJXDFFKFLMG-UHFFFAOYSA-N 0.000 title abstract 2
- 229960001929 meloxicam Drugs 0.000 title abstract 2
- AYXYPKUFHZROOJ-ZETCQYMHSA-N pregabalin Chemical compound CC(C)C[C@H](CN)CC(O)=O AYXYPKUFHZROOJ-ZETCQYMHSA-N 0.000 title abstract 2
- 229960001233 pregabalin Drugs 0.000 title abstract 2
- 230000003110 anti-inflammatory effect Effects 0.000 title 1
- 230000003574 anti-allodynic effect Effects 0.000 abstract 2
- 229940121363 anti-inflammatory agent Drugs 0.000 abstract 2
- 239000002260 anti-inflammatory agent Substances 0.000 abstract 2
- 239000003795 chemical substances by application Substances 0.000 abstract 2
- 208000004296 neuralgia Diseases 0.000 abstract 1
- 208000021722 neuropathic pain Diseases 0.000 abstract 1
- 230000002265 prevention Effects 0.000 abstract 1
- 230000002195 synergetic effect Effects 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
- A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/20—Pills, tablets, discs, rods
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4866—Organic macromolecular compounds
Landscapes
- Health & Medical Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Epidemiology (AREA)
- Biomedical Technology (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Rheumatology (AREA)
- Neurology (AREA)
- Neurosurgery (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Abstract
La presente invención se refiere a una novedosa combinación farmacéutica sinérgica de un agente antihiperalgésico, antialodínico y un agente antiinflamatorio, en donde el agente antihiperalgésico, antialodínico es Pregabalina, y el agente antiinflamatorio es Meloxicam. La presente invención además está dirigida a composiciones farmacéuticas que comprenden dicha combinación, y al uso de dicha combinación y composiciones farmacéuticas para la prevención y/o tratamiento del dolor neuropático ocasionado por diversas etiologías.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
MX2014008336A MX2014008336A (es) | 2014-07-07 | 2014-07-07 | Combinacion farmacologica antihiperalgesica, antialodinica y antiinflamatoria, composiciones farmaceuticas que la contienen, y su uso para el tratamiento del dolor neuropatico. |
PCT/IB2015/055127 WO2016005897A1 (en) | 2014-07-07 | 2015-07-07 | Combination of pregabalin and meloxicam for the treatment of neuropathic pain |
Publications (1)
Publication Number | Publication Date |
---|---|
CO2017001076A2 true CO2017001076A2 (es) | 2017-05-31 |
Family
ID=53938368
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CONC2017/0001076A CO2017001076A2 (es) | 2014-07-07 | 2017-02-06 | Composiciones farmacéuticas antihiperalgésicas, antialodínicas y antiinflamatorias que contienen pregabalina y meloxicam |
Country Status (5)
Country | Link |
---|---|
BR (1) | BR112017000359A2 (es) |
CO (1) | CO2017001076A2 (es) |
MX (1) | MX2014008336A (es) |
PE (1) | PE20171140A1 (es) |
WO (1) | WO2016005897A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US11590094B2 (en) | 2017-09-28 | 2023-02-28 | Nevakar Injectables Inc. | Fixed dose combination formulations for treating pain |
MX2019008467A (es) * | 2019-07-16 | 2019-11-07 | Federico Amezcua Amezcua | Combinacion sinergica de s-ketorolaco y pregabalina en una composicion farmaceutica para el tratamiento del dolor neuropatico. |
CN112353767A (zh) * | 2020-11-16 | 2021-02-12 | 海南锦瑞制药有限公司 | 一种盐酸地尔硫卓和普瑞巴林组合物及其制备方法及其应用 |
Family Cites Families (7)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US6129907A (en) | 1999-08-04 | 2000-10-10 | Colgate Palmolive Company | Stable hydrogenated lupulone antibacterial oral compositions |
WO2003066040A1 (fr) | 2002-02-05 | 2003-08-14 | Ajinomoto Co.,Inc. | Compositions medicinales contenant une gabapentine ou une pregabaline et antagoniste a canal de calcium de type n |
DE10331305A1 (de) | 2003-07-10 | 2005-02-17 | Siemens Ag | Kommunikationssystem, Peer-to-Peer-Nachrichten-Filter-Rechner und Verfahren zum Verarbeiten einer Peer-to-Peer-Nachricht |
BRPI0610316A2 (pt) | 2005-05-20 | 2010-06-15 | Pfizer Ltd | combinações sinergìsticas de medicamentos atiinflamatórios não estereoidais com alfa-delta-ligantes |
CA2701838A1 (en) | 2007-10-09 | 2009-04-16 | Merck Patent Gmbh | Pharmaceutical compositions containing benfotiamine and one or more pharmaceutically active agents for the treatment of pain conditions of neuropathic origin |
ES2619329T3 (es) | 2007-11-23 | 2017-06-26 | Grünenthal GmbH | Composiciones de tapentadol |
MX336979B (es) | 2011-12-16 | 2016-02-09 | Senosiain S A De C V Lab | Combinacion farmaceutica antineuritica y composiciones. |
-
2014
- 2014-07-07 MX MX2014008336A patent/MX2014008336A/es unknown
-
2015
- 2015-07-07 PE PE2017000033A patent/PE20171140A1/es unknown
- 2015-07-07 WO PCT/IB2015/055127 patent/WO2016005897A1/en active Application Filing
- 2015-07-07 BR BR112017000359-7A patent/BR112017000359A2/pt not_active Application Discontinuation
-
2017
- 2017-02-06 CO CONC2017/0001076A patent/CO2017001076A2/es unknown
Also Published As
Publication number | Publication date |
---|---|
WO2016005897A1 (en) | 2016-01-14 |
BR112017000359A2 (pt) | 2018-06-26 |
PE20171140A1 (es) | 2017-08-09 |
MX2014008336A (es) | 2016-01-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
SV2017005461A (es) | Benzamidas sustituidas con 1,3-tiazol-2-ilo | |
CL2020002032A1 (es) | Cristal de un compuesto derivado de 7,8-difluoro-6,11-dihidrodibenzotiepina, composición farmacéutica, útil en reducir el tiempo de alivio de los síntomas de la influenza para tratar y/o prevenir una infección provocada por el virus de la influenza. (divisional solicitud 201900325). | |
CL2018003588A1 (es) | Uso de inhibidores de miostatina y terapias de combinación. | |
SV2018005778A (es) | Derivados aromaticos de sulfonamida | |
BR112018004620A2 (pt) | moduladores da expressão de kras | |
CL2018001996A1 (es) | Composiciones y métodos para modular la expresión del factor b del complemento (divisional de solicitud 2764-16) | |
BR112017022089A2 (pt) | uso de uma composição, e, método para branqueamento de dentes | |
CR20160433A (es) | Nuevos compuestos | |
NI202100018A (es) | Moduladores de la expresión de pnpla3 | |
SV2017005466A (es) | Pirazolpiridinaminas como inhibidores de mknk1 y mknk2 | |
CL2019001996A1 (es) | Usos terapéuticos de un polvo de insectos. | |
GT201500247A (es) | Imidazopiridazinas sustituidas | |
CL2017002214A1 (es) | Formulación de combinación de tesofensina y betabloqueante | |
CR20190471A (es) | Moduladores de la expresión de pcsk9 | |
BR112016013754A2 (pt) | Recaptação de serotonina-norepinefrina inibidores (irsns) e combinações dos ligantes do receptor sigma | |
CL2019001746A1 (es) | Amidas aromáticas de ácido carboxílico | |
CO2017001076A2 (es) | Composiciones farmacéuticas antihiperalgésicas, antialodínicas y antiinflamatorias que contienen pregabalina y meloxicam | |
CL2019001618A1 (es) | Uso de compuestos de carbamato para prevención, alivio o tratamiento del trastorno bipolar. | |
DOP2016000251A (es) | Inhibidores de las vías de señalización de wnt | |
CO2020003134A2 (es) | Moduladores de la expresión de enac | |
AR106415A1 (es) | Composición farmacéutica para el tratamiento del dolor | |
CU20170134A7 (es) | 2-tiopirimidinonas | |
CO2019007261A2 (es) | Combinación de un inhibidor de mcl-1 y un compuesto taxano, usos y composiciones farmacéuticas de ésta | |
BR112019006591A2 (pt) | derivado de oxazina para uso no tratamento ou prevenção de angiopatia amiloide cerebral | |
AR102215A1 (es) | Compuesto de pirazol-4-carboxamida, composición farmacéutica que lo comprende y su uso para la fabricación de un medicamento |