CN116832122A - 一种中药组合物、制剂及其制备方法、使用方法和应用 - Google Patents
一种中药组合物、制剂及其制备方法、使用方法和应用 Download PDFInfo
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Abstract
本发明公开了一种中药组合物、制剂及其制备方法、使用方法和应用,属于中药制备技术领域。所述组合物包括以下配方组分:大黄,龙胆草,白花藤,三丫苦叶,金银花,白鲜皮,金盏银盘,冰片,薄荷,冰蚕,黄莲,纯牛黄,冰醋酸氯己定,赤石脂,天麻子。本发明限定的中药组合物、制剂配方安全无毒,且通过药物组分之间的君臣佐使作用机理,按照五天一次,一共三次涂抹在患处,就能够在短时间内治愈痔疮,且该中药组合物还具有能够除去皮肤上的黑痣,老年斑和疣的作用功效,具有十分广阔的应用前景。
Description
技术领域
本发明涉及中药制备技术领域,更具体的说是涉及一种中药组合物、制剂及其制备方法、使用方法和应用。
背景技术
痔疮(Hemorrhoids),或称痔,是位于肛管的血管组织,是临床上一种最常见的肛门疾病。发病时痛苦难忍,给人们工作生活带来了很大的影响。目前治疗痔疮的方法很多,主要采用手术和非手术治疗。但是一方面,手术治疗具有痛苦大,安全系数低,费用高,伤口愈合时间长等缺点,大多数患者不愿接受;另一方面虽然也有中药治疗痔疮病的报道,但其疗效各有区别,有的效果不是十分理想。
因此,研究一种能够通过外涂抹不用手术就能治疗痔疮的中药组合物是本领域技术人员亟需解决的问题。
发明内容
有鉴于此,本发明提供了一种中药组合物、制剂及其制备方法、使用方法和应用,通过限定的中药组合物配方组分间的君臣佐使的配伍机理,能够激发人体自我排斥功能和自我修复功能达到消除痔疮的作用效果。
为了实现上述目的,本发明采用如下技术方案:
一种中药组合物,包括以下配方组分:大黄,龙胆草,白花藤,三丫苦叶,金银花,白鲜皮,金盏银盘,冰片,薄荷,冰蚕,黄莲,纯牛黄,冰醋酸氯己定,赤石脂,天麻子。
上述技术方案达到的有益效果为:通过本发明限定的上述组分的配伍,可以发挥各味中药的综合作用、以及所有组分的协同作用治愈痔疮。解决了现有痔疮需要手术流大量的血液和患者康复伤口短时间难以愈合,患者需要经历长时间的痛苦,影响患者的正常生活和行动的问题。且本发明原材料易得、成本低、无毒副作用、疗效快。
其中,本发明限定的中药组合物中各组分的功效为:
大黄(Rheum palmatum L.)别称将军、黄良、火参等,是多种蓼科大黄属的多年生植物的合称、中药材的名称。大黄能增加肠蠕动,抑制肠内水分吸收,促进排便;大黄有抗感染作用,对多种革兰阳性和阴性细菌均有抑制作用,其中最敏感的为葡萄球菌和链球菌,其次为白喉杆菌、伤寒和副伤寒杆菌、肺炎双球菌、痢疾杆菌等;对流感病毒也有抑制作用;由于鞣质所致,故泻后又有便秘现象;有利胆和健胃作用;此外,还有清热泻火,清血瘀、保肝、降压、降低血清胆固醇等作用。
龙胆草(学名:Gentiana scabraBunge,别名:草龙胆),捩花目龙胆科龙胆属植物。用于清热燥湿,泻肝胆火。用于湿热黄疸,阴肿阴痒,带下,湿疹瘙痒,肝火目赤,耳鸣耳聋,胁痛口苦,强中,惊风抽搐。
白花藤为豆科崖豆藤属植物滇桂崖豆藤MillettiabonatianaPamp.,具有清肝明目,清热,止痢的功效,还能治疗皮炎。
三丫苦叶,中药名。为芸香科植物三丫苦叶Evodialepta(spr.)Merr.的叶。具有清热解毒,散瘀止痛,祛风除湿的作用和功效,可用于咽喉肿痛,黄疸型肝炎,疮疡肿毒,虫蛇咬伤,风湿骨痛,湿疹,皮炎。
金银花(拉丁学名:Lonicerajaponica Thunb.,别名:子风藤),忍冬科忍冬属多年生半常绿缠绕灌木。金银花含有绿原酸、木犀草素苷等药理活性成分,对溶血性链球菌、金黄葡萄球菌等多种致病菌及上呼吸道感染致病病毒等有较强的抑制力,另外还可增强免疫力、抗早孕、护肝、抗肿瘤、清热解毒、疏风散热、止血(凝血)、抑制肠道吸收胆固醇等,其临床用途非常广泛,可与其它药物配伍用于治疗呼吸道感染、菌痢、急性泌尿系统感染、高血压等40余种病症。
白鲜皮,为芸香科白鲜属植物白鲜Dictamnus dasycarpus Turcz.的干燥根皮。具有清热燥湿,祛风解毒的功效,还能增强肌肉的收缩力和肠道的平滑肌收缩的作用与功效,其对出血消炎也有一定的帮助。
金盏银盘,中药名。为菊科植物三叶鬼针草或金盏银盘的干燥全草,春、夏季采收,鲜用或切段晒干。其味甘、微苦,性凉。有清热解毒,凉血止血,加快人体新陈代谢之功效。用于感冒发热,黄疸,泄泻,痢疾,血热吐血,血崩,跌打损伤,痈肿疮毒,鹤膝风,疥癞。
冰片(Borneol)是无色透明或白色半透明的片状松脆结晶,为龙脑香料植物龙脑香树的树脂中析出的天然结晶性化合物。可以固化伤口,消炎止痛,防止细菌进入。
薄荷(拉丁学名:Menthahaplocalyx Briq.),唇形科薄荷属多年生草本植物,是一种有特种经济价值的芳香作物。薄荷的作用是治外感风热,头痛,咽喉肿痛,温病初起,薄荷用药禁忌阴虚血燥,肝阳偏亢,表虚汗多者忌服薄荷;还能够治疗皮肤瘙痒,皮疹和湿疹,身热肿痛。
冰蚕:能够促进机体新陈代谢的作用,具有润肠,滑肌,生肌作用。
黄莲(拉丁学名:Coptis chinensis Franch),别名为南天竹。具有清热燥湿,泻火解毒的功效,还具有能止泻厚肠,热血排毒,抗病毒等作用。
纯牛黄(CowBzoar)是脊索动物门哺乳纲牛科动物牛胆囊的胆结石。其本身带有微毒性,具有阴寒特性,对人体有清热解毒,软化血管的作用,对血排毒效果很好。
冰醋酸氯己定:冰醋酸对葡萄球菌,变异链球菌,白色念珠菌,大肠杆菌,厌氧丙酸菌有抑制作用,一般粘膜的消毒,冲洗可外用于淋病,阴道炎,激发修复皮肤细胞。
赤石脂,中药名。为硅酸盐类多水高岭石族矿石多水高岭石与氧化物类赤铁矿或含氢氧化物类褐铁矿共同组成的细分散多矿物集合体,主含四水硅酸铝。具有涩肠止泻,收敛止血,敛疮生肌的功效。
天麻子(拉丁学名:Tetrapanaxpapyrifer(Hook.)K.Koch,别名:通脱木)。具有镇痛,抗惊厥,降血压,补虚定风的功效,也可以治疗失眠。
综上所述,本发明限定的原料组分之间君臣佐使的协同增效机理为:
君:白鲜皮冰片纯牛黄冰醋酸氯己定
臣:龙胆草白花藤金银花薄荷冰蚕天麻子
佐:大黄黄莲赤石脂
使:三丫苦叶金盏银盘
具体来讲,冰醋酸氯己定消除,杀灭痔疮感染的细菌,冰片,白鲜皮使痔疮达到固化和消炎,滑肌止痛的作用,冰蚕协助增强了痔疮的滑肌修复功能,纯牛黄有加快血液的排毒吸收,但是太短,为了加强牛黄的功能,大黄,黄莲,赤石脂起到了加强作用,薄荷,金银花,龙胆草,白花藤是为了减少冰醋酸氯己定的酸性对人体痛感时间,达到止痛消炎的作用,有冰凉的效果,三百苦,金盏银盘是辅助君药,臣药,防止固化出血,减少对人体的伤害,帮扶作用消除各种药物剩余的有害成分,起到了中和的关键性作用。因此,本发明通过修复静脉血管,可以根治痔疮。
优选的,按照重量份数计,包括以下配方组分:大黄20-40份,龙胆草10-30份,白花藤40-60份,三丫苦叶40-60份,金银花10-30份,白鲜皮10-30份,金盏银盘90-110份,冰片5-15份,薄荷15-25份,冰蚕15-25份,黄莲40-60份,纯牛黄1-2份,冰醋酸氯己定90-170份,赤石脂15-30份,天麻子5-10份。
优选的,按照重量份数计,包括以下配方组分:大黄30份,龙胆草20份,白花藤50份,三丫苦叶50份,金银花20份,白鲜皮20份,金盏银盘100份,冰片10份,薄荷20份,冰蚕20份,黄莲50份,纯牛黄1份,冰醋酸氯己定100份,赤石脂20份,天麻子10份。
一种中药制剂,包括上述中药组合物。
优选的,所述制剂为外敷液体制剂。
一种中药制剂的制备方法,包括以下步骤:
(1)根据上述中药制剂中各组分的用量份数,将所述纯牛黄,冰片,白鲜皮,冰蚕和赤石脂混合研磨,过筛成1000目的细浆,用冰醋酸反复冲洗,过滤,直到全部过滤用玻璃瓶密封装好,得药液1;
(2)将所述薄荷和金银花分别采用水蒸气蒸馏提取有效成分;
将所述龙胆草和天麻子分别采用乙醇蒸馏提取有效成分,其中所述乙醇体积浓度为50%(v/v),其用量为所述龙胆草或是天麻子重量的5倍;
再将上述得到的有效成分混合,得药液2;
(3)将所述大黄,白花藤,三丫苦叶,金盏银盘和黄莲,采用水煮法,得药液3;
(4)将所述药液1、2、3混匀,密封放在常温阴凉处保存,最终制得所述中药制剂,可保存两年。
优选的,步骤(1)所述过滤采用的过滤网为1000目。
优选的,步骤(3)所述水煮法具体步骤为:
将所述大黄,白花藤,三丫苦叶,金盏银盘和黄莲的混合物与水按照重量比为1:15慢火煮沸至1:2后过滤,再用慢火煮至所述混合物与水的重量比为1:1,密封装好放凉得所述药液3。
上述中药制剂在制备治疗痔疮药物中的应用。
一种上述中药制剂的使用方法,具体为:
在患者患有痔疮的位置,每五天涂抹所述中药制剂一次,连涂三次,经过第一次涂抹之后,患者30min以后就不会再痛,用洗脸纸巾包覆在痔疮上吸收人体排出来的静脉沉积蛋白,至所述洗脸纸巾不再吸附,再换新的洗脸纸巾,第25天就会感觉肛门发痒,第28天就没有液体排出,痔疮就治愈了,一般痒的感觉在七天左右。
优选的,当所述患有痔疮为内痔时,需要先采用扩肛器进行扩肛,然后涂抹,一小时后再取出扩肛器。
上述中药制剂在制备治疗除去皮肤上黑痣,老年斑和疣药物中的应用。
经由上述的技术方案可知,与现有技术相比,本发明公开提供了一种中药组合物、制剂及其制备方法、使用方法和应用,具有以下有益效果:
1.本发明制备的中药制剂仅仅通过外涂抹就可以治愈痔疮,无需手术,避免了流血和对生活和工作的严重影响;
2.本发明制备的中药制剂治疗痔疮周期短,每隔五天涂抹一次,共涂抹三次,治疗周期为35天就会完全康复;
3.本发明限定的中药组合物、制剂配方安全无毒,且制备方法简单,制备出的中药制剂具有疗效好,实用性高的特点;
4.该中药制剂还能够除去皮肤上的黑痣,老年斑和疣,具有广阔的应用前景。
附图说明
为了更清楚地说明本发明实施例或现有技术中的技术方案,下面将对实施例或现有技术描述中所需要使用的附图作简单地介绍,显而易见地,下面描述中的附图仅仅是本发明的实施例,对于本领域普通技术人员来讲,在不付出创造性劳动的前提下,还可以根据提供的附图获得其他的附图。
图1附图为本发明实施例4制备的中药制剂对痔疮患者1的治疗图片。
图2附图为本发明实施例4制备的中药制剂对痔疮患者2的治疗图片
具体实施方式
下面将结合本发明实施例中的附图,对本发明实施例中的技术方案进行清楚、完整地描述,显然,所描述的实施例仅仅是本发明一部分实施例,而不是全部的实施例。基于本发明中的实施例,本领域普通技术人员在没有做出创造性劳动前提下所获得的所有其他实施例,都属于本发明保护的范围。
实施例1
一种中药组合物,按照重量份数计,包括以下配方组分::大黄20份,龙胆草10份,白花藤40份,三丫苦叶40份,金银花10份,白鲜皮10份,金盏银盘90份,冰片5份,薄荷15份,冰蚕15份,黄莲40份,纯牛黄1份,冰醋酸氯己定90份,赤石脂15份,天麻子5份。
实施例2
一种中药组合物,按照重量份数计,包括以下配方组分:大黄30份,龙胆草20份,白花藤50份,三丫苦叶50份,金银花20份,白鲜皮20份,金盏银盘100份,冰片10份,薄荷20份,冰蚕20份,黄莲50份,纯牛黄1份,冰醋酸氯己定100份,赤石脂20份,天麻子10份。
实施例3
一种中药组合物,按照重量份数计,包括以下配方组分::大黄40份,龙胆草30份,白花藤60份,三丫苦叶60份,金银花30份,白鲜皮30份,金盏银盘110份,冰片15份,薄荷25份,冰蚕25份,黄莲60份,纯牛黄2份,冰醋酸氯己定170份,赤石脂30份,天麻子10份。
实施例4
一种中药制剂,按照以下步骤进行制备:
(1)按照上述实施例2中各组分的用量份数,将纯牛黄,冰片,白鲜皮,冰蚕,赤石脂混合研磨成1000目的细浆,用冰醋酸反复冲洗,过滤1000目的网,直到全部过滤用密封装好(玻璃瓶),得药液1;
(2)将薄荷和金银花分别采用水蒸气蒸馏提取有效成分;
将龙胆草和天麻子分别采用乙醇蒸馏提取有效成分,其中乙醇体积浓度为50%(v/v),乙醇用量为龙胆草或天麻子的5倍;
再将上述有效成分混合,得药液2;
(3)将大黄,白花藤,三丫苦叶,金盏银盘,黄莲采用水煮法得到药液3;其中,水煮法具体步骤为:将大黄,白花藤,三丫苦叶,金盏银盘和黄莲的混合物与水按照重量比为1:15慢火煮沸至1:2后过滤,再用慢火煮至混合物与水的重量比为1:1,密封装好放凉得药液3。
(4)将药液1、2、3混匀,得中药制剂。
效果验证
1.将实施例4制备的中药制剂,在患者患有痔疮的地方,每五天涂抹一次,连涂三次,治疗周期35天内便可痊愈。
现对两个患者利用上述使用方法进行治疗,具体治疗效果可见附图1和2。
从两个附图中可以看出,两位患者均患有严重的外痔,在本发明公开的中药制剂的涂抹治疗下,在35天的治疗周期内,痔疮在治疗过程中逐渐变小,最终完全消失,即痔疮彻底治愈。
2.将实施例4制备的中药制剂,用棉签蘸取,按照三天涂抹一次,涂覆在皮肤有黑痣,老年斑或疣的地方,七天就会脱落。
总结:通过本发明限定的中药组合物以及中药制剂,可以在短时间治愈痔疮,而且还能去除皮肤上的黑痣,老年斑和疣,具有很广阔的应用前景。
本说明书中各个实施例采用递进的方式描述,每个实施例重点说明的都是与其他实施例的不同之处,各个实施例之间相同相似部分互相参见即可。对于实施例公开的装置而言,由于其与实施例公开的方法相对应,所以描述的比较简单,相关之处参见方法部分说明即可。
对所公开的实施例的上述说明,使本领域专业技术人员能够实现或使用本发明。对这些实施例的多种修改对本领域的专业技术人员来说将是显而易见的,本文中所定义的一般原理可以在不脱离本发明的精神或范围的情况下,在其它实施例中实现。因此,本发明将不会被限制于本文所示的这些实施例,而是要符合与本文所公开的原理和新颖特点相一致的最宽的范围。
Claims (10)
1.一种中药组合物,其特征在于,包括以下组分:大黄,龙胆草,白花藤,三丫苦叶,金银花,白鲜皮,金盏银盘,冰片,薄荷,冰蚕,黄莲,纯牛黄,冰醋酸氯己定,赤石脂,天麻子。
2.根据权利要求1所述的中药组合物,其特征在于,按照重量份数计,包括以下组分:大黄20-40份,龙胆草10-30份,白花藤40-60份,三丫苦叶40-60份,金银花10-30份,白鲜皮10-30份,金盏银盘90-110份,冰片5-15份,薄荷15-25份,冰蚕15-25份,黄莲40-60份,纯牛黄1-2份,冰醋酸氯己定90-170份,赤石脂15-30份,天麻子5-10份。
3.根据权利要求2所述的中药组合物,其特征在于,按照重量份数计,包括以下组分:大黄30份,龙胆草20份,白花藤50份,三丫苦叶50份,金银花20份,白鲜皮20份,金盏银盘100份,冰片10份,薄荷20份,冰蚕20份,黄莲50份,纯牛黄1份,冰醋酸氯己定100份,赤石脂20份,天麻子10份。
4.一种中药制剂,其特征在于,包括权利要求1-3任一项所述中药组合物。
5.根据权利要求4所述的一种中药制剂,其特征在于,所述中药制剂为外敷液体制剂。
6.一种中药制剂的制备方法,其特征在于,包括以下步骤:
(1)根据权利要求4-5任一项所述中药制剂中各组分的用量份数,将所述纯牛黄、冰片、白鲜皮、冰蚕和赤石脂混合研磨,用所述冰醋酸氯己定冲洗,过滤,得药液1;
(2)将所述薄荷和金银花分别采用水蒸汽蒸馏提取有效成分;
将所述龙胆草和天麻子分别采用乙醇蒸馏提取有效成分;其中乙醇体积浓度为50%(v/v);
再将上述有效成分混合,得药液2;
(3)将所述大黄、白花藤、三丫苦叶、金盏银盘和黄莲混合,然后采用水煮法进行水煮,得到药液3;
(4)将所述药液1、2和3混匀,得所述中药制剂。
7.根据权利要求6所述的一种中药制剂的制备方法,其特征在于,步骤(1)所述过滤采用的是1000目过滤网。
8.根据权利要求6所述的一种中药制剂的制备方法,其特征在于,步骤(3)所述水煮法具体步骤为:
将所述大黄、白花藤、三丫苦叶、金盏银盘和黄莲的混合物与水按照重量比为1:15慢火煮沸至1:2后过滤,再用慢火煮至所述混合物与水的重量比为1:1,密封装好放凉得所述药液3。
9.根据权利要求4-5任一项所述中药制剂或权利要求6-8任一项所述制备方法制备的中药制剂在制备治疗痔疮药物中的应用。
10.根据权利要求4-5任一项所述中药制剂或权利要求6-8任一项所述制备方法制备的中药制剂的使用方法,其特征在于,将所述中药制剂在患者患处每5天涂抹一次,涂抹3次后便可治愈。
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