CN102762210B - 2-醛肟-5-氟嘧啶衍生物 - Google Patents

2-醛肟-5-氟嘧啶衍生物 Download PDF

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Publication number
CN102762210B
CN102762210B CN201080063991.8A CN201080063991A CN102762210B CN 102762210 B CN102762210 B CN 102762210B CN 201080063991 A CN201080063991 A CN 201080063991A CN 102762210 B CN102762210 B CN 102762210B
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CN
China
Prior art keywords
herbicides
insecticides
compounds
plant
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Fee Related
Application number
CN201080063991.8A
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English (en)
Chinese (zh)
Other versions
CN102762210A (zh
Inventor
T.波伊贝尔
B.罗尔斯巴赫
T.马丁
W.欧文
M.苏伦伯格
姚成林
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Corteva Agriscience LLC
Original Assignee
Dow AgroSciences LLC
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Dow AgroSciences LLC filed Critical Dow AgroSciences LLC
Publication of CN102762210A publication Critical patent/CN102762210A/zh
Application granted granted Critical
Publication of CN102762210B publication Critical patent/CN102762210B/zh
Expired - Fee Related legal-status Critical Current
Anticipated expiration legal-status Critical

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
    • C07D239/46—Two or more oxygen, sulphur or nitrogen atoms
    • C07D239/47—One nitrogen atom and one oxygen or sulfur atom, e.g. cytosine
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/48—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with two nitrogen atoms as the only ring hetero atoms
    • A01N43/54—1,3-Diazines; Hydrogenated 1,3-diazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/10—Antimycotics

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Zoology (AREA)
  • Environmental Sciences (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Plant Pathology (AREA)
  • Pest Control & Pesticides (AREA)
  • Agronomy & Crop Science (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
CN201080063991.8A 2009-12-17 2010-12-16 2-醛肟-5-氟嘧啶衍生物 Expired - Fee Related CN102762210B (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US28734609P 2009-12-17 2009-12-17
US61/287,346 2009-12-17
PCT/US2010/060792 WO2011084611A1 (en) 2009-12-17 2010-12-16 2-aldoximino-5-fluoropyrimidine derivatives

Related Child Applications (1)

Application Number Title Priority Date Filing Date
CN201410396518.1A Division CN104211646A (zh) 2009-12-17 2010-12-16 2-醛肟-5-氟嘧啶衍生物

Publications (2)

Publication Number Publication Date
CN102762210A CN102762210A (zh) 2012-10-31
CN102762210B true CN102762210B (zh) 2014-09-17

Family

ID=44151954

Family Applications (2)

Application Number Title Priority Date Filing Date
CN201080063991.8A Expired - Fee Related CN102762210B (zh) 2009-12-17 2010-12-16 2-醛肟-5-氟嘧啶衍生物
CN201410396518.1A Pending CN104211646A (zh) 2009-12-17 2010-12-16 2-醛肟-5-氟嘧啶衍生物

Family Applications After (1)

Application Number Title Priority Date Filing Date
CN201410396518.1A Pending CN104211646A (zh) 2009-12-17 2010-12-16 2-醛肟-5-氟嘧啶衍生物

Country Status (17)

Country Link
US (1) US8912207B2 (enExample)
EP (1) EP2512482A4 (enExample)
KR (1) KR20120094140A (enExample)
CN (2) CN102762210B (enExample)
AU (1) AU2010339900A1 (enExample)
CA (1) CA2787488A1 (enExample)
CL (1) CL2012002070A1 (enExample)
CO (1) CO6561812A2 (enExample)
CR (1) CR20120380A (enExample)
EC (1) ECSP12012047A (enExample)
IN (1) IN2012DN06286A (enExample)
MA (1) MA33932B1 (enExample)
MY (1) MY159707A (enExample)
PH (1) PH12012501462A1 (enExample)
RU (1) RU2012130427A (enExample)
TN (1) TN2012000381A1 (enExample)
WO (1) WO2011084611A1 (enExample)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
PL2252594T3 (pl) * 2008-01-22 2016-01-29 Dow Agrosciences Llc Pochodne 4-amino-5-fluoropirymidyny jako fungicydy
CN110128354A (zh) * 2019-06-20 2019-08-16 大连大学 一种5-氟-2-甲磺酰基-4-氨基嘧啶的制备方法

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090203647A1 (en) * 2008-01-22 2009-08-13 Dow Agrosciences Llc 5-fluoro pyrimidine derivatives

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPH045279A (ja) * 1990-04-23 1992-01-09 Mitsubishi Petrochem Co Ltd 新規なオキシムエーテル誘導体およびそれを有効成分とする除草剤および農園芸用殺菌剤
MXPA04004583A (es) * 2001-11-19 2004-08-13 Basf Ag 5-fenilpirimidinas, agentes que comprenden las mismas, metodo de produccion y uso de la misma.
JP2005232081A (ja) 2004-02-19 2005-09-02 Bayer Cropscience Ag ベンジルピリミジン誘導体の農園芸用殺菌剤としての利用

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20090203647A1 (en) * 2008-01-22 2009-08-13 Dow Agrosciences Llc 5-fluoro pyrimidine derivatives

Non-Patent Citations (3)

* Cited by examiner, † Cited by third party
Title
嘧啶类化合物杀菌活性研究进展;薛伟等;《农药》;20070831;第46卷(第8期);第505-509,516页 *
嘧啶类化合物的合成及抗菌活性研究进展;吴琴等;《有机化学》;20090315;第29卷(第3期);第365-379页 *
张德志等.理化性质对药效的影响,官能团对药效的影响.《药学概论》.中国医药科技出版社,2008,356、359. *

Also Published As

Publication number Publication date
ECSP12012047A (es) 2012-08-31
EP2512482A4 (en) 2013-05-22
CN102762210A (zh) 2012-10-31
TN2012000381A1 (en) 2014-01-30
PH12012501462A1 (en) 2012-10-29
CO6561812A2 (es) 2012-11-15
MY159707A (en) 2017-01-13
IN2012DN06286A (enExample) 2015-09-25
AU2010339900A1 (en) 2012-08-09
US20110152300A1 (en) 2011-06-23
RU2012130427A (ru) 2014-01-27
CN104211646A (zh) 2014-12-17
CL2012002070A1 (es) 2013-03-08
CR20120380A (es) 2012-09-13
EP2512482A1 (en) 2012-10-24
WO2011084611A1 (en) 2011-07-14
MA33932B1 (fr) 2013-01-02
KR20120094140A (ko) 2012-08-23
US8912207B2 (en) 2014-12-16
CA2787488A1 (en) 2011-07-14

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