CN102686574A - 作为具有治疗应用的受体调节剂的香豆素化合物 - Google Patents

作为具有治疗应用的受体调节剂的香豆素化合物 Download PDF

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Publication number
CN102686574A
CN102686574A CN2010800587171A CN201080058717A CN102686574A CN 102686574 A CN102686574 A CN 102686574A CN 2010800587171 A CN2010800587171 A CN 2010800587171A CN 201080058717 A CN201080058717 A CN 201080058717A CN 102686574 A CN102686574 A CN 102686574A
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oxo
chromene
methane amide
methoxyl group
propyl group
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CN2010800587171A
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Chinese (zh)
Inventor
T·M·海德尔堡
J·R·卡皮罗
P·阮
D·G·戈麦斯
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Allergan Inc
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Allergan Inc
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    • A61K31/365—Lactones
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  • Life Sciences & Earth Sciences (AREA)
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  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
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  • Dermatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pain & Pain Management (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
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  • Urology & Nephrology (AREA)
  • Surgery (AREA)
  • Vascular Medicine (AREA)
  • Communicable Diseases (AREA)
  • Transplantation (AREA)
  • Biochemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrane Compounds (AREA)
CN2010800587171A 2009-10-23 2010-10-20 作为具有治疗应用的受体调节剂的香豆素化合物 Pending CN102686574A (zh)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US25423609P 2009-10-23 2009-10-23
US61/254,236 2009-10-23
PCT/US2010/053363 WO2011050054A2 (en) 2009-10-23 2010-10-20 Coumarin compounds as receptor modulators with therapeutic utility

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CN102686574A true CN102686574A (zh) 2012-09-19

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CN2010800587171A Pending CN102686574A (zh) 2009-10-23 2010-10-20 作为具有治疗应用的受体调节剂的香豆素化合物

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US (2) US9073888B2 (https=)
EP (1) EP2491023B1 (https=)
JP (1) JP2013508385A (https=)
KR (1) KR20120075481A (https=)
CN (1) CN102686574A (https=)
BR (1) BR112012009670A2 (https=)
CA (1) CA2778611A1 (https=)
RU (1) RU2012119249A (https=)
WO (1) WO2011050054A2 (https=)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN107868069A (zh) * 2017-10-31 2018-04-03 山东新华制药股份有限公司 7‑羟基‑8‑甲基‑6‑硝基‑2‑氧‑2h‑苯并吡喃‑3‑羧酸的制备工艺
CN107935976A (zh) * 2017-11-13 2018-04-20 山东大学 香豆素酰胺衍生物及其应用
CN110713497A (zh) * 2019-10-30 2020-01-21 成都海杰亚医药科技有限公司 一种Brigatinib的中间体2-氨基苯基二甲基氧化膦制备方法
CN116478173A (zh) * 2023-04-20 2023-07-25 山西师范大学 一种靶向高尔基体监测极性的荧光探针及其制备与应用

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US12478503B2 (en) 2009-05-18 2025-11-25 Glaukos Corporation Implants with controlled drug delivery features and methods of using same
US10206813B2 (en) 2009-05-18 2019-02-19 Dose Medical Corporation Implants with controlled drug delivery features and methods of using same
CA2778611A1 (en) * 2009-10-23 2011-04-28 Allergan, Inc. Coumarin compounds as receptor modulators with therapeutic utility
JPWO2019151470A1 (ja) 2018-02-02 2021-02-25 国立大学法人京都大学 眼内血管新生及び／又は眼内血管透過性亢進を伴う眼科疾患の予防又は治療のための医薬
US12273086B2 (en) * 2022-08-31 2025-04-08 Apple Inc. Adjustable radio-frequency splitter-combiner

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KR20120075481A (ko) 2012-07-06
US9572792B2 (en) 2017-02-21
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US20120328661A1 (en) 2012-12-27
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RU2012119249A (ru) 2013-11-27
US9073888B2 (en) 2015-07-07

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