CL2020003272A1 - Nuevas formas cristalinas de 1-(4-{[6-amino-5-(4-fenoxi-fenil)-pirimidin-4-ilamino]-metil}-4-fluoro-piperidin-1-il)-propenona, formas de sal de la misma y procesos de obtención - Google Patents
Nuevas formas cristalinas de 1-(4-{[6-amino-5-(4-fenoxi-fenil)-pirimidin-4-ilamino]-metil}-4-fluoro-piperidin-1-il)-propenona, formas de sal de la misma y procesos de obtenciónInfo
- Publication number
- CL2020003272A1 CL2020003272A1 CL2020003272A CL2020003272A CL2020003272A1 CL 2020003272 A1 CL2020003272 A1 CL 2020003272A1 CL 2020003272 A CL2020003272 A CL 2020003272A CL 2020003272 A CL2020003272 A CL 2020003272A CL 2020003272 A1 CL2020003272 A1 CL 2020003272A1
- Authority
- CL
- Chile
- Prior art keywords
- forms
- propenone
- ylamino
- pyrimidin
- piperidin
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
- C07D401/12—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings linked by a chain containing hetero atoms as chain links
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Immunology (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines Containing Antibodies Or Antigens For Use As Internal Diagnostic Agents (AREA)
Abstract
La presente invención se refiere a una forma sólida de 1-(4-{[6-amino-5-(4-fenoxi-fenil)-pirimidin-4-ilamino]-metil}-4-fluoro-piperidin-1-il)-propenona (compuesto 1), o sales farmacéuticamente aceptables del mismo, útiles como inhibidores de BTK.
Applications Claiming Priority (1)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US201862686797P | 2018-06-19 | 2018-06-19 |
Publications (1)
Publication Number | Publication Date |
---|---|
CL2020003272A1 true CL2020003272A1 (es) | 2021-05-07 |
Family
ID=67003464
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CL2020003272A CL2020003272A1 (es) | 2018-06-19 | 2020-12-17 | Nuevas formas cristalinas de 1-(4-{[6-amino-5-(4-fenoxi-fenil)-pirimidin-4-ilamino]-metil}-4-fluoro-piperidin-1-il)-propenona, formas de sal de la misma y procesos de obtención |
Country Status (13)
Country | Link |
---|---|
US (2) | US11878967B2 (es) |
EP (1) | EP3810590A1 (es) |
JP (1) | JP2021527685A (es) |
KR (1) | KR20210022674A (es) |
CN (1) | CN112313214A (es) |
AU (1) | AU2019289628A1 (es) |
BR (1) | BR112020025881A2 (es) |
CA (1) | CA3104191A1 (es) |
CL (1) | CL2020003272A1 (es) |
IL (1) | IL279485A (es) |
MX (1) | MX2020013321A (es) |
SG (1) | SG11202012595PA (es) |
WO (1) | WO2019243223A1 (es) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20240024314A1 (en) * | 2020-01-08 | 2024-01-25 | Telios Pharma, Inc. | Methods of Treating Splenomegaly |
CR20220374A (es) * | 2020-01-08 | 2023-01-25 | Telios Pharma Inc | Métodos de tratamiento de la esplenomegalia |
EP4165730A1 (en) | 2020-06-10 | 2023-04-19 | Merck Patent GmbH | Steerable antenna and method for heating and/or tempering of a steerable antenna |
Family Cites Families (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
SG194219A1 (en) * | 2011-06-10 | 2013-11-29 | Merck Patent Gmbh | Compositions and methods for the production of pyrimidine and pyridine compounds with btk inhibitory activity |
CA3218491A1 (en) * | 2012-06-04 | 2013-12-12 | Pharmacyclics Llc | Crystalline forms of a bruton's tyrosine kinase inhibitor |
CN103694241A (zh) * | 2013-11-27 | 2014-04-02 | 苏州晶云药物科技有限公司 | Pci-32765的新晶型a及其制备方法 |
US20180051026A1 (en) | 2015-03-03 | 2018-02-22 | Dr. Reddy's Laboratories Limited | Polymorphs of ibrutinib |
CN107873029B (zh) * | 2015-04-02 | 2020-09-01 | 拉蒂奥法姆有限责任公司 | 依鲁替尼与羧酸的共晶体 |
DK3371165T3 (da) | 2015-11-04 | 2022-05-02 | Merck Patent Gmbh | Btk-inhibitor til anvendelse til behandling af kræft |
HUE064244T2 (hu) * | 2015-11-17 | 2024-02-28 | Merck Patent Gmbh | Módszerek szklerózis multiplex kezelésére BTK gátló aktivitású pirimidin- és piridin-származékokkal |
US10464923B2 (en) * | 2017-02-27 | 2019-11-05 | Merck Patent Gmbh | Crystalline forms of 1-(4-{[6-amino-5-(4-phenoxy-phenyl)-pyrimidin-4-ylamino]-methyl}-piperidin-1-yl)-propenone |
-
2019
- 2019-06-17 MX MX2020013321A patent/MX2020013321A/es unknown
- 2019-06-17 EP EP19732937.8A patent/EP3810590A1/en active Pending
- 2019-06-17 BR BR112020025881-4A patent/BR112020025881A2/pt unknown
- 2019-06-17 KR KR1020217001602A patent/KR20210022674A/ko unknown
- 2019-06-17 US US17/252,804 patent/US11878967B2/en active Active
- 2019-06-17 AU AU2019289628A patent/AU2019289628A1/en active Pending
- 2019-06-17 CA CA3104191A patent/CA3104191A1/en active Pending
- 2019-06-17 WO PCT/EP2019/065815 patent/WO2019243223A1/en unknown
- 2019-06-17 CN CN201980041020.4A patent/CN112313214A/zh active Pending
- 2019-06-17 SG SG11202012595PA patent/SG11202012595PA/en unknown
- 2019-06-17 JP JP2020570863A patent/JP2021527685A/ja active Pending
-
2020
- 2020-12-16 IL IL279485A patent/IL279485A/en unknown
- 2020-12-17 CL CL2020003272A patent/CL2020003272A1/es unknown
-
2023
- 2023-12-07 US US18/532,710 patent/US20240132472A1/en active Pending
Also Published As
Publication number | Publication date |
---|---|
BR112020025881A2 (pt) | 2021-03-23 |
IL279485A (en) | 2021-01-31 |
EP3810590A1 (en) | 2021-04-28 |
KR20210022674A (ko) | 2021-03-03 |
SG11202012595PA (en) | 2021-01-28 |
MX2020013321A (es) | 2021-02-22 |
JP2021527685A (ja) | 2021-10-14 |
US11878967B2 (en) | 2024-01-23 |
US20210261525A1 (en) | 2021-08-26 |
AU2019289628A1 (en) | 2021-02-04 |
CA3104191A1 (en) | 2019-12-26 |
US20240132472A1 (en) | 2024-04-25 |
WO2019243223A1 (en) | 2019-12-26 |
CN112313214A (zh) | 2021-02-02 |
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