CL2008001112A1 - Uses of compounds derived from pyrido [2,3-d] pyrimidin-4-one to treat itching or a disorder related to itching; combination of the compounds with another drug; and use of the combination to treat itching or a disorder related to itching. - Google Patents

Uses of compounds derived from pyrido [2,3-d] pyrimidin-4-one to treat itching or a disorder related to itching; combination of the compounds with another drug; and use of the combination to treat itching or a disorder related to itching.

Info

Publication number
CL2008001112A1
CL2008001112A1 CL2008001112A CL2008001112A CL2008001112A1 CL 2008001112 A1 CL2008001112 A1 CL 2008001112A1 CL 2008001112 A CL2008001112 A CL 2008001112A CL 2008001112 A CL2008001112 A CL 2008001112A CL 2008001112 A1 CL2008001112 A1 CL 2008001112A1
Authority
CL
Chile
Prior art keywords
itching
combination
disorder related
treat
compounds
Prior art date
Application number
CL2008001112A
Other languages
Spanish (es)
Inventor
Thomas Meingassner Josef Gottfried Jung
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38038626&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CL2008001112(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CL2008001112A1 publication Critical patent/CL2008001112A1/en

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4427Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems
    • A61K31/444Non condensed pyridines; Hydrogenated derivatives thereof containing further heterocyclic ring systems containing a six-membered ring with nitrogen as a ring heteroatom, e.g. amrinone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K45/00Medicinal preparations containing active ingredients not provided for in groups A61K31/00 - A61K41/00
    • A61K45/06Mixtures of active ingredients without chemical characterisation, e.g. antiphlogistics and cardiaca
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/04Antipruritics

Abstract

Usos de compuestos derivados de piridina, antagonistas del receptor vanilloide, para el tratamiento de comezón o de un trastorno o enfermedad relacionada con comezón; combinación farmacéutica que comprende al compuesto derivado de piridina.Uses of pyridine-derived compounds, vanilloid receptor antagonists, for the treatment of itching or of a disorder or disease related to itching; pharmaceutical combination comprising the pyridine derivative compound.

CL2008001112A 2007-04-20 2008-04-18 Uses of compounds derived from pyrido [2,3-d] pyrimidin-4-one to treat itching or a disorder related to itching; combination of the compounds with another drug; and use of the combination to treat itching or a disorder related to itching. CL2008001112A1 (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
EP07106648 2007-04-20

Publications (1)

Publication Number Publication Date
CL2008001112A1 true CL2008001112A1 (en) 2008-12-19

Family

ID=38038626

Family Applications (1)

Application Number Title Priority Date Filing Date
CL2008001112A CL2008001112A1 (en) 2007-04-20 2008-04-18 Uses of compounds derived from pyrido [2,3-d] pyrimidin-4-one to treat itching or a disorder related to itching; combination of the compounds with another drug; and use of the combination to treat itching or a disorder related to itching.

Country Status (3)

Country Link
CL (1) CL2008001112A1 (en)
TW (1) TW200902014A (en)
WO (1) WO2008129000A1 (en)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US20140179727A1 (en) 2012-12-14 2014-06-26 Trevi Therapeutics, Inc. Methods for treating pruritus
US8987289B2 (en) * 2012-12-14 2015-03-24 Trevi Therapeutics, Inc. Methods for treating pruritus
WO2015112588A1 (en) 2014-01-22 2015-07-30 Biomimetix Jv, Llc Methods of treating skin disorders
US10080759B2 (en) 2014-01-22 2018-09-25 Duke University Methods of treating pruritus
WO2020023486A1 (en) 2018-07-23 2020-01-30 Trevi Therapeutics, Inc. Treatment of chronic cough, breathlessness and dyspnea
CN114605408B (en) * 2022-03-30 2023-06-16 沈阳药科大学 5-hydroxy-1, 3-disubstituted phenylpyrido [2,3-d ] pyrimidine compound and preparation method and application thereof

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP4205430B2 (en) * 2001-03-26 2009-01-07 ノバルティス アクチエンゲゼルシャフト Condensed pyridine derivatives for use as vanilloid receptor antagonists to treat pain
WO2005023807A2 (en) * 2003-09-09 2005-03-17 Neurogen Corporation 4 - heterobicyclyamino - substituted quinazolines and analogues therof as capsaicin - antagonists

Also Published As

Publication number Publication date
TW200902014A (en) 2009-01-16
WO2008129000A1 (en) 2008-10-30

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