CH519519A - 2 3 1-diazaborine derivs - Google Patents
2 3 1-diazaborine derivsInfo
- Publication number
- CH519519A CH519519A CH1784167A CH1784167A CH519519A CH 519519 A CH519519 A CH 519519A CH 1784167 A CH1784167 A CH 1784167A CH 1784167 A CH1784167 A CH 1784167A CH 519519 A CH519519 A CH 519519A
- Authority
- CH
- Switzerland
- Prior art keywords
- alkyl
- derivs
- subst
- opt
- mercapto
- Prior art date
Links
- 125000000217 alkyl group Chemical group 0.000 abstract 3
- 229910052736 halogen Inorganic materials 0.000 abstract 2
- 150000002367 halogens Chemical class 0.000 abstract 2
- 125000002887 hydroxy group Chemical group [H]O* 0.000 abstract 2
- 125000000449 nitro group Chemical group [O-][N+](*)=O 0.000 abstract 2
- 125000002030 1,2-phenylene group Chemical group [H]C1=C([H])C([*:1])=C([*:2])C([H])=C1[H] 0.000 abstract 1
- 125000000175 2-thienyl group Chemical group S1C([*])=C([H])C([H])=C1[H] 0.000 abstract 1
- 241000588724 Escherichia coli Species 0.000 abstract 1
- 101000835998 Homo sapiens SRA stem-loop-interacting RNA-binding protein, mitochondrial Proteins 0.000 abstract 1
- 241000699666 Mus <mouse, genus> Species 0.000 abstract 1
- 241000699670 Mus sp. Species 0.000 abstract 1
- 102100025491 SRA stem-loop-interacting RNA-binding protein, mitochondrial Human genes 0.000 abstract 1
- 125000004442 acylamino group Chemical group 0.000 abstract 1
- 230000000845 anti-microbial effect Effects 0.000 abstract 1
- 230000001741 anti-phlogistic effect Effects 0.000 abstract 1
- 230000000842 anti-protozoal effect Effects 0.000 abstract 1
- 125000003118 aryl group Chemical group 0.000 abstract 1
- 125000004391 aryl sulfonyl group Chemical group 0.000 abstract 1
- 150000001768 cations Chemical class 0.000 abstract 1
- 239000000824 cytostatic agent Substances 0.000 abstract 1
- 230000001085 cytostatic effect Effects 0.000 abstract 1
- 125000000623 heterocyclic group Chemical group 0.000 abstract 1
- -1 mercapto, amino Chemical group 0.000 abstract 1
- 125000004957 naphthylene group Chemical group 0.000 abstract 1
- 125000001997 phenyl group Chemical group [H]C1=C([H])C([H])=C(*)C([H])=C1[H] 0.000 abstract 1
- 125000005556 thienylene group Chemical group 0.000 abstract 1
- 125000003396 thiol group Chemical class [H]S* 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F5/00—Compounds containing elements of Groups 3 or 13 of the Periodic Table
- C07F5/02—Boron compounds
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
Abstract
derivs. of formula: (I) where Z = o-phenylene, naphthylene or thienylene, opt. subst. by one or more halogen, alkyl, etherified hydroxy or mercapto, alkyl-, aralkyl- or aryl-sulphonyl, or nitro; R1= mono- or polynuclear aromatic or heterocyclic gp., opt. subst. by halogen, alkyl, etherified hydroxy or mercapto, amino, acylamino or nitro; R2= H, monovalent cation or Antimicrobial, eg. DC50 determined by oral administration to mice infected with E. coli is about 0.5 mg/20 g mouse for cpd. I(Z-o-phenylene; R1 = phenyl or 2-thienyl). Some cpds. I have antiprotozoal effect, esp. on trypanosomes and plasmodia. Some also have cytostatic or antiphlogistic activity.
Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CH1784167A CH519519A (en) | 1966-04-30 | 1967-12-20 | 2 3 1-diazaborine derivs |
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DEC0038925 | 1966-04-30 | ||
| CH1784167A CH519519A (en) | 1966-04-30 | 1967-12-20 | 2 3 1-diazaborine derivs |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CH519519A true CH519519A (en) | 1972-02-29 |
Family
ID=25720118
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CH1784167A CH519519A (en) | 1966-04-30 | 1967-12-20 | 2 3 1-diazaborine derivs |
Country Status (1)
| Country | Link |
|---|---|
| CH (1) | CH519519A (en) |
-
1967
- 1967-12-20 CH CH1784167A patent/CH519519A/en not_active IP Right Cessation
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| FR2337554A1 (en) | (1)-Substd. (2)-phenyl-(4)-butyl-pyrazolidine dione salts - analgesics and antiinflammatories with little ulcerogenic action | |
| CH519519A (en) | 2 3 1-diazaborine derivs | |
| CH288866A (en) | Ceramic, magnetic molded body with the properties of an insulator. | |
| FR2071171A6 (en) | 1,1-diphenyl-azaborolidines - with insecticidal acaricidal - herbicidal and fungicidal activity | |
| ES346192A1 (en) | 6-chloro-2-(5-nitro-2-furyl) cinchoninic acid | |
| FR1602619A (en) | Antibiotic cephalosporin cpds | |
| FR2104634A1 (en) | 1-hydroxycarbonyl-2-aminobenzimidazoles - and their thio derivs antifungal agents | |
| GB1070183A (en) | Silver mercaptides and their use in sensitive photographic materials | |
| FR2205525A1 (en) | Alkyl 2,2-dichlorovinyl phosphates - prepd. by reaction of corresp. halo-phosphate with opt. substd. cyclic hydroxy cpds | |
| FR1072948A (en) | Luminous body | |
| NL7416673A (en) | 3-(4-Ureido-2-acylphenoxy)-2-hydroxy-propylamines - cardioselective beta-adrenergic blocking agents | |
| CA506002A (en) | Controlled oxidation of branched chain organic compounds | |
| FR1100820A (en) | Mechanical toy, especially tank | |
| NL7309456A (en) | Compsns. contg. 5-(1,1-disubstd. alkyl) pyrimidines - with pesticidal and/or plant-growth regulating activity | |
| ES28894U (en) | Pacifier with surprise (Machine-translation by Google Translate, not legally binding) | |
| FR2018246A1 (en) | 4,5-dihydro-3h-1,3-benzodiazepine-4-ones as psycho - sedatives, hypnotics and muscle relaxants | |
| FR2171939A2 (en) | 2,2-dichlorovinyl - pyridyl alkyl phosphates - with antiparasitic activity | |
| GR10545B (en) | MOVING ANIMAL MODEL - CHILDREN'S TOY. | |
| FR1102573A (en) | Pump, especially for agricultural applications | |
| ES39990U (en) | Sprayer or pocket nebulizer (Machine-translation by Google Translate, not legally binding) | |
| CH291059A (en) | Amplifier with conditionally stable negative feedback. | |
| AU166943B2 (en) | IMPROVEMENTS INTHE PURIFICATION OF 1, 1, i TRICHLORO 2, 2-BIS(4-CHLOROPHENYL)ETHANE | |
| NL189334B (en) | THERAPEUTIC PREPARATION CONTAINING CATECHOL DERIVATIVES. | |
| ES17720U (en) | Cigarette case. (Machine-translation by Google Translate, not legally binding) | |
| FI40535C (en) | Staining to 5- (gamma-sec. |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PFA | Name/firm changed |
Owner name: GRUENENTHAL GMBH |
|
| PL | Patent ceased |