CA3217168A1 - Crystalline form v of melanocortin receptor agonist compound, and method for preparing same - Google Patents
Crystalline form v of melanocortin receptor agonist compound, and method for preparing same Download PDFInfo
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- CA3217168A1 CA3217168A1 CA3217168A CA3217168A CA3217168A1 CA 3217168 A1 CA3217168 A1 CA 3217168A1 CA 3217168 A CA3217168 A CA 3217168A CA 3217168 A CA3217168 A CA 3217168A CA 3217168 A1 CA3217168 A1 CA 3217168A1
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- crystalline form
- ether
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Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/10—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/16—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07B—GENERAL METHODS OF ORGANIC CHEMISTRY; APPARATUS THEREFOR
- C07B2200/00—Indexing scheme relating to specific properties of organic compounds
- C07B2200/13—Crystalline forms, e.g. polymorphs
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Diabetes (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Endocrinology (AREA)
- Epidemiology (AREA)
- Child & Adolescent Psychology (AREA)
- Emergency Medicine (AREA)
- Pain & Pain Management (AREA)
- Rheumatology (AREA)
- Gynecology & Obstetrics (AREA)
- Reproductive Health (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| KR20210058701 | 2021-05-06 | ||
| KR10-2021-0058701 | 2021-05-06 | ||
| PCT/KR2022/006478 WO2022235104A1 (ko) | 2021-05-06 | 2022-05-06 | 멜라노코르틴 수용체 작용제 화합물의 결정형 v 및 이의 제조방법 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA3217168A1 true CA3217168A1 (en) | 2022-11-10 |
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ID=83932274
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA3217168A Pending CA3217168A1 (en) | 2021-05-06 | 2022-05-06 | Crystalline form v of melanocortin receptor agonist compound, and method for preparing same |
Country Status (9)
| Country | Link |
|---|---|
| US (1) | US20240228473A1 (de) |
| EP (1) | EP4317149A4 (de) |
| JP (1) | JP2024518055A (de) |
| KR (1) | KR20220151569A (de) |
| CN (1) | CN117242064A (de) |
| AU (1) | AU2022271119A1 (de) |
| CA (1) | CA3217168A1 (de) |
| MX (1) | MX2023013044A (de) |
| WO (1) | WO2022235104A1 (de) |
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| JP2003505435A (ja) * | 1999-06-04 | 2003-02-12 | メルク エンド カムパニー インコーポレーテッド | メラノコルチン−４受容体ゴニストとしての置換ピペリジン |
| WO2002059107A1 (en) * | 2001-01-23 | 2002-08-01 | Eli Lilly And Company | Substituted piperidines/piperazines as melanocortin receptor agonists |
| AR044510A1 (es) | 2003-04-14 | 2005-09-14 | Merck & Co Inc | Procedimiento e intermedios para preparar acidos carboxilicos de pirrolidina |
| US7989634B2 (en) * | 2003-11-12 | 2011-08-02 | Lg Life Sciences Ltd. | Melanocortin receptor agonists |
| TWI332501B (en) | 2006-07-14 | 2010-11-01 | Lg Life Sciences Ltd | Melanocortin receptor agonists |
| UA99555C2 (en) * | 2008-11-12 | 2012-08-27 | Элджи Лайф Саенсез Лтд. | Melanocortin receptor agonists |
| EP3580194A4 (de) | 2017-02-08 | 2020-12-30 | Tilray, Inc. | Verfahren und vorrichtung zur niederdruck-strahlungsenergieverarbeitung von cannabis |
| ES2970510T3 (es) * | 2019-11-07 | 2024-05-29 | Lg Chemical Ltd | Agonistas del receptor de melanocortina-4 |
| KR20210058701A (ko) | 2019-11-13 | 2021-05-24 | 서강대학교산학협력단 | 의존 구문 분석 시스템 및 이를 이용한 의존 구문 분석 방법 |
| KR102672626B1 (ko) * | 2020-10-29 | 2024-06-07 | 주식회사 엘지화학 | 멜라노코르틴 수용체 작용제 화합물의 결정형 ⅲ 및 이의 제조방법 |
| EP4219472A4 (de) * | 2020-10-29 | 2024-03-13 | Lg Chem, Ltd. | Kristalline form i einer melanocortinrezeptoragonistenverbindung und verfahren zur herstellung davon |
| AU2021371829B2 (en) * | 2020-10-29 | 2024-01-18 | Lg Chem, Ltd. | Crystalline form ii of melanocortin receptor agonist compound and preparation method therefor |
| MX2023004731A (es) * | 2020-10-29 | 2023-05-10 | Lg Chemical Ltd | Forma cristalina iv del compuesto agonista de receptor de melanocortina y metodo de preparacion para la misma. |
| US20240043407A1 (en) * | 2020-12-22 | 2024-02-08 | Lg Chem, Ltd. | Crystalline form i of melanocortin receptor agonist compound and method for preparing same |
| KR20220090455A (ko) * | 2020-12-22 | 2022-06-29 | 주식회사 엘지화학 | 무정형의 멜라노코르틴 수용체 작용제 및 이의 제조방법 |
| TWI814185B (zh) * | 2020-12-22 | 2023-09-01 | 南韓商Ｌｇ化學股份有限公司 | 黑皮質素受體促效劑化合物之晶型ii及其製備方法 |
-
2022
- 2022-05-06 EP EP22799147.8A patent/EP4317149A4/de active Pending
- 2022-05-06 WO PCT/KR2022/006478 patent/WO2022235104A1/ko active Application Filing
- 2022-05-06 JP JP2023568097A patent/JP2024518055A/ja active Pending
- 2022-05-06 MX MX2023013044A patent/MX2023013044A/es unknown
- 2022-05-06 AU AU2022271119A patent/AU2022271119A1/en active Pending
- 2022-05-06 CN CN202280032212.0A patent/CN117242064A/zh active Pending
- 2022-05-06 KR KR1020220055894A patent/KR20220151569A/ko not_active Application Discontinuation
- 2022-05-06 US US18/557,866 patent/US20240228473A1/en active Pending
- 2022-05-06 CA CA3217168A patent/CA3217168A1/en active Pending
Also Published As
| Publication number | Publication date |
|---|---|
| MX2023013044A (es) | 2023-11-15 |
| JP2024518055A (ja) | 2024-04-24 |
| CN117242064A (zh) | 2023-12-15 |
| US20240228473A1 (en) | 2024-07-11 |
| AU2022271119A1 (en) | 2023-11-02 |
| WO2022235104A1 (ko) | 2022-11-10 |
| KR20220151569A (ko) | 2022-11-15 |
| EP4317149A4 (de) | 2024-08-21 |
| EP4317149A1 (de) | 2024-02-07 |
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