CA3181292A1 - Methods and compositions for preventing and treating myopia with levocabastine, a selective histamine h1-receptor antagonist, and derivatives thereof - Google Patents
Methods and compositions for preventing and treating myopia with levocabastine, a selective histamine h1-receptor antagonist, and derivatives thereof Download PDFInfo
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- CA3181292A1 CA3181292A1 CA3181292A CA3181292A CA3181292A1 CA 3181292 A1 CA3181292 A1 CA 3181292A1 CA 3181292 A CA3181292 A CA 3181292A CA 3181292 A CA3181292 A CA 3181292A CA 3181292 A1 CA3181292 A1 CA 3181292A1
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- myopia
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- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/445—Non condensed piperidines, e.g. piperocaine
- A61K31/451—Non condensed piperidines, e.g. piperocaine having a carbocyclic group directly attached to the heterocyclic ring, e.g. glutethimide, meperidine, loperamide, phencyclidine, piminodine
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0048—Eye, e.g. artificial tears
- A61K9/0051—Ocular inserts, ocular implants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/10—Ophthalmic agents for accommodation disorders, e.g. myopia
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- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Medicinal Chemistry (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
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- Bioinformatics & Cheminformatics (AREA)
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- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nutrition Science (AREA)
- Physiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicinal Preparation (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
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| US202063033291P | 2020-06-02 | 2020-06-02 | |
| US63/033,291 | 2020-06-02 | ||
| PCT/US2021/035344 WO2021247635A1 (en) | 2020-06-02 | 2021-06-02 | Methods and compositions for preventing and treating myopia with levocabastine, a selective histamine h1-receptor antagonist, and derivatives thereof |
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| CA3181292A1 true CA3181292A1 (en) | 2021-12-09 |
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| IL (1) | IL298796A (ko) |
| WO (1) | WO2021247635A1 (ko) |
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| CN116270442A (zh) * | 2021-12-21 | 2023-06-23 | 浙江瑞瞳生物科技有限公司 | 一种用于矫正近距离视力的眼用制剂 |
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| EP2399555B1 (en) * | 2009-02-20 | 2016-12-07 | Seed Co., Ltd. | Sustainedly drug-releasing hydrogel contact lens, and drug releasing method using sustainedly drug-releasing hydrogel contact lens |
| US9827250B2 (en) * | 2012-07-31 | 2017-11-28 | Johnson & Johnson Vision Care, Inc. | Lens incorporating myopia control optics and muscarinic agents |
| ITUB20160876A1 (it) * | 2016-02-19 | 2017-08-19 | Dambrosio Enzo Maria | Combinazione di un agente antiallergico con un antagonista muscarinico e/o un agonista dopaminergico per l'uso in prevenzione/ arresto di miopia assiale nell’uomo |
| US10945980B2 (en) * | 2016-06-21 | 2021-03-16 | The University Of Newcastle | Treatment for myopia |
| SG11201907701YA (en) * | 2017-02-21 | 2019-09-27 | Singapore Health Serv Pte Ltd | Composition and method for preventing or delaying onset of myopia comprising atropine |
| AU2018371787A1 (en) * | 2017-11-21 | 2020-11-05 | Sydnexis, Inc. | Ophthalmic composition and delivery device thereof |
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2021
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- 2021-06-02 CN CN202180049465.4A patent/CN115835905A/zh active Pending
- 2021-06-02 EP EP21816939.9A patent/EP4157453A4/en active Pending
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- 2021-06-02 CA CA3181292A patent/CA3181292A1/en active Pending
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| IL298796A (en) | 2023-02-01 |
| EP4157453A1 (en) | 2023-04-05 |
| JP2023529374A (ja) | 2023-07-10 |
| WO2021247635A1 (en) | 2021-12-09 |
| CN115835905A (zh) | 2023-03-21 |
| KR20230051130A (ko) | 2023-04-17 |
| EP4157453A4 (en) | 2024-06-19 |
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