CA3072079A1 - Methods of treatment - Google Patents
Methods of treatment Download PDFInfo
- Publication number
- CA3072079A1 CA3072079A1 CA3072079A CA3072079A CA3072079A1 CA 3072079 A1 CA3072079 A1 CA 3072079A1 CA 3072079 A CA3072079 A CA 3072079A CA 3072079 A CA3072079 A CA 3072079A CA 3072079 A1 CA3072079 A1 CA 3072079A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- raynaud
- individual
- pharmaceutically acceptable
- hydrate
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Pending
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Classifications
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
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| US201862711369P | 2018-07-27 | 2018-07-27 | |
| US62/711,369 | 2018-07-27 | ||
| PCT/US2018/045683 WO2019032626A1 (en) | 2017-08-07 | 2018-08-07 | Methods of treatment |
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| EP2367797A1 (en) | 2008-11-26 | 2011-09-28 | Arena Pharmaceuticals, Inc. | Pyrazolyl substituted carbonic acid derivatives as modulators of the prostacyclin (pgi2) receptor useful for the treatment of disorders related thereto |
| US8940891B2 (en) | 2008-12-08 | 2015-01-27 | Arena Pharmaceuticals, Inc. | Modulators of the prostacyclin (PGI2) receptor useful for the treatment of disorders related thereto |
| AU2023222747A1 (en) | 2022-02-15 | 2024-08-22 | United Therapeutics Corporation | Crystalline prostacyclin (ip) receptor agonist and uses thereof |
| WO2025193579A1 (en) | 2024-03-11 | 2025-09-18 | United Therapeutics Corporation | Methods of making ip-receptor agonists |
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| EP2280696B9 (en) | 2008-03-18 | 2015-12-09 | Arena Pharmaceuticals, Inc. | Modulators of the prostacyclin (pgi2) receptor useful for the treatment of disorders related thereto |
| US10188648B2 (en) * | 2015-09-03 | 2019-01-29 | Teva Pharmaceuticals International Gmbh | Solid state forms of selexipag |
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- 2018-08-07 EP EP18759520.2A patent/EP3664792A1/en active Pending
- 2018-08-07 CA CA3072079A patent/CA3072079A1/en active Pending
- 2018-08-07 US US16/636,608 patent/US20200368190A1/en not_active Abandoned
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| US20200368190A1 (en) | 2020-11-26 |
| WO2019032626A1 (en) | 2019-02-14 |
| JP7343478B2 (ja) | 2023-09-12 |
| JP2020530447A (ja) | 2020-10-22 |
| EP3664792A1 (en) | 2020-06-17 |
| US20240122886A1 (en) | 2024-04-18 |
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