CA2975072A1 - Method for producing pyrazinecarboxamide compound and synthetic intermediate thereof - Google Patents
Method for producing pyrazinecarboxamide compound and synthetic intermediate thereof Download PDFInfo
- Publication number
- CA2975072A1 CA2975072A1 CA2975072A CA2975072A CA2975072A1 CA 2975072 A1 CA2975072 A1 CA 2975072A1 CA 2975072 A CA2975072 A CA 2975072A CA 2975072 A CA2975072 A CA 2975072A CA 2975072 A1 CA2975072 A1 CA 2975072A1
- Authority
- CA
- Canada
- Prior art keywords
- compound
- salt
- formula
- production method
- methylpiperazin
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
- C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/4965—Non-condensed pyrazines
- A61K31/497—Non-condensed pyrazines containing further heterocyclic rings
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
JP2015-014533 | 2015-01-28 | ||
JP2015014533 | 2015-01-28 | ||
PCT/JP2016/052229 WO2016121777A1 (ja) | 2015-01-28 | 2016-01-27 | ピラジンカルボキサミド化合物の製造方法及びその合成中間体 |
Publications (1)
Publication Number | Publication Date |
---|---|
CA2975072A1 true CA2975072A1 (en) | 2016-08-04 |
Family
ID=56543388
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA2975072A Abandoned CA2975072A1 (en) | 2015-01-28 | 2016-01-27 | Method for producing pyrazinecarboxamide compound and synthetic intermediate thereof |
Country Status (6)
Country | Link |
---|---|
JP (1) | JPWO2016121777A1 (zh) |
KR (1) | KR20170105021A (zh) |
CN (1) | CN107207468A (zh) |
CA (1) | CA2975072A1 (zh) |
MX (1) | MX2017009714A (zh) |
WO (1) | WO2016121777A1 (zh) |
Families Citing this family (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US20190282569A1 (en) * | 2016-10-26 | 2019-09-19 | Astellas Pharma Inc. | Stable pharmaceutical composition |
JP2023528859A (ja) * | 2020-06-01 | 2023-07-06 | ウィゲン・バイオメディシン・テクノロジー・(シャンハイ)・カンパニー・リミテッド | 新規ピラジン化合物 |
IL313670A (en) | 2021-12-30 | 2024-08-01 | Biomea Fusion Inc | Pyrazine compounds as inhibitors of FLT3 |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
JPS5754177A (ja) * | 1980-09-19 | 1982-03-31 | Teikoku Hormone Mfg Co Ltd | Chikanchiazoorujudotai |
JP3534903B2 (ja) * | 1995-06-09 | 2004-06-07 | 鐘淵化学工業株式会社 | 1−[3−クロロ−(2s)−メチルプロピオニル]−ピロリジン−(2s)−カルボン酸の製造方法 |
CN104080774B (zh) * | 2012-01-17 | 2017-02-22 | 安斯泰来制药株式会社 | 吡嗪甲酰胺化合物 |
-
2016
- 2016-01-27 KR KR1020177020729A patent/KR20170105021A/ko unknown
- 2016-01-27 CN CN201680007743.9A patent/CN107207468A/zh active Pending
- 2016-01-27 MX MX2017009714A patent/MX2017009714A/es unknown
- 2016-01-27 CA CA2975072A patent/CA2975072A1/en not_active Abandoned
- 2016-01-27 WO PCT/JP2016/052229 patent/WO2016121777A1/ja active Application Filing
- 2016-01-27 JP JP2016572078A patent/JPWO2016121777A1/ja active Pending
Also Published As
Publication number | Publication date |
---|---|
KR20170105021A (ko) | 2017-09-18 |
JPWO2016121777A1 (ja) | 2017-11-02 |
MX2017009714A (es) | 2017-11-17 |
CN107207468A (zh) | 2017-09-26 |
WO2016121777A1 (ja) | 2016-08-04 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
FZDE | Dead |
Effective date: 20200128 |