CA2781063A1 - Combination - Google Patents
Combination Download PDFInfo
- Publication number
- CA2781063A1 CA2781063A1 CA2781063A CA2781063A CA2781063A1 CA 2781063 A1 CA2781063 A1 CA 2781063A1 CA 2781063 A CA2781063 A CA 2781063A CA 2781063 A CA2781063 A CA 2781063A CA 2781063 A1 CA2781063 A1 CA 2781063A1
- Authority
- CA
- Canada
- Prior art keywords
- administered
- cancer
- phenylamino
- pyrimidin
- fluoro
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
Links
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A61P35/02—Antineoplastic agents specific for leukemia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
Landscapes
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Molecular Biology (AREA)
- Biophysics (AREA)
- Urology & Nephrology (AREA)
- Inorganic Chemistry (AREA)
- Neurology (AREA)
- Physical Education & Sports Medicine (AREA)
- Endocrinology (AREA)
- Dermatology (AREA)
- Neurosurgery (AREA)
- Reproductive Health (AREA)
- Gastroenterology & Hepatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Pulmonology (AREA)
- Hematology (AREA)
- Biomedical Technology (AREA)
- Diabetes (AREA)
- Oncology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US26181309P | 2009-11-17 | 2009-11-17 | |
| US61/261,813 | 2009-11-17 | ||
| PCT/US2010/056931 WO2011062930A1 (en) | 2009-11-17 | 2010-11-17 | Combination |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2781063A1 true CA2781063A1 (en) | 2011-05-26 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA2781063A Abandoned CA2781063A1 (en) | 2009-11-17 | 2010-11-17 | Combination |
Country Status (17)
| Country | Link |
|---|---|
| US (4) | US20120283279A1 (enExample) |
| EP (1) | EP2501379B1 (enExample) |
| JP (1) | JP5834370B2 (enExample) |
| KR (1) | KR20120117779A (enExample) |
| CN (2) | CN104382906A (enExample) |
| AU (1) | AU2010322105B2 (enExample) |
| BR (1) | BR112012011677A8 (enExample) |
| CA (1) | CA2781063A1 (enExample) |
| EA (1) | EA022637B1 (enExample) |
| ES (1) | ES2578191T3 (enExample) |
| IL (1) | IL219786A (enExample) |
| MX (1) | MX2012005758A (enExample) |
| PL (1) | PL2501379T3 (enExample) |
| PT (1) | PT2501379E (enExample) |
| SG (1) | SG10201407558TA (enExample) |
| WO (1) | WO2011062930A1 (enExample) |
| ZA (1) | ZA201203444B (enExample) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP2640390A4 (en) * | 2010-11-17 | 2014-08-06 | Glaxosmithkline Ip No 2 Ltd | METHODS OF TREATING CANCER |
| TWI505828B (zh) | 2010-12-20 | 2015-11-01 | 葛蘭素史克智慧財產（第二）有限公司 | 新穎醫藥組成物 |
| US20140377285A1 (en) * | 2011-11-08 | 2014-12-25 | Intellikine, Llc | Treatment regimens using multiple pharmaceutical agents |
| WO2014059095A1 (en) * | 2012-10-12 | 2014-04-17 | Glaxosmithkline Llc | Combinations |
| CA2946759A1 (en) | 2014-04-25 | 2015-10-29 | Memorial Sloan-Kettering Cancer Center | Treatment of h-ras-driven tumors |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AU2003248813A1 (en) * | 2002-07-05 | 2004-01-23 | Beth Israel Deaconess Medical Center | Combination of mtor inhibitor and a tyrosine kinase inhibitor for the treatment of neoplasms |
| US7378423B2 (en) * | 2004-06-11 | 2008-05-27 | Japan Tobacco Inc. | Pyrimidine compound and medical use thereof |
| MXPA06014478A (es) * | 2004-06-11 | 2007-03-21 | Japan Tobacco Inc | Derivados de 5-amino-2, 4, 7-trioxo-3, 4, 7, 8-tetrahidro -2h-pirido[2, 3-d]pirimidina y compuestos relacionados para el tratamiento del cancer. |
| JP2011500657A (ja) * | 2007-10-15 | 2011-01-06 | アストラゼネカ アクチボラグ | 組合せ０５９ |
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2010
- 2010-11-17 KR KR1020127015509A patent/KR20120117779A/ko not_active Abandoned
- 2010-11-17 EA EA201290339A patent/EA022637B1/ru not_active IP Right Cessation
- 2010-11-17 US US13/509,955 patent/US20120283279A1/en not_active Abandoned
- 2010-11-17 EP EP10832068.0A patent/EP2501379B1/en active Active
- 2010-11-17 ES ES10832068.0T patent/ES2578191T3/es active Active
- 2010-11-17 SG SG10201407558TA patent/SG10201407558TA/en unknown
- 2010-11-17 PT PT108320680T patent/PT2501379E/pt unknown
- 2010-11-17 CA CA2781063A patent/CA2781063A1/en not_active Abandoned
- 2010-11-17 CN CN201410535441.1A patent/CN104382906A/zh active Pending
- 2010-11-17 CN CN2010800616827A patent/CN102724979A/zh active Pending
- 2010-11-17 WO PCT/US2010/056931 patent/WO2011062930A1/en not_active Ceased
- 2010-11-17 AU AU2010322105A patent/AU2010322105B2/en not_active Ceased
- 2010-11-17 MX MX2012005758A patent/MX2012005758A/es active IP Right Grant
- 2010-11-17 JP JP2012539983A patent/JP5834370B2/ja not_active Expired - Fee Related
- 2010-11-17 BR BR112012011677A patent/BR112012011677A8/pt not_active IP Right Cessation
- 2010-11-17 PL PL10832068.0T patent/PL2501379T3/pl unknown
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2012
- 2012-05-11 ZA ZA2012/03444A patent/ZA201203444B/en unknown
- 2012-05-14 IL IL219786A patent/IL219786A/en not_active IP Right Cessation
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2014
- 2014-06-19 US US14/309,262 patent/US20140303195A1/en not_active Abandoned
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2015
- 2015-09-24 US US14/863,709 patent/US20160008368A1/en not_active Abandoned
-
2016
- 2016-11-16 US US15/352,813 patent/US20170065593A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| KR20120117779A (ko) | 2012-10-24 |
| AU2010322105A1 (en) | 2012-05-31 |
| US20170065593A1 (en) | 2017-03-09 |
| WO2011062930A1 (en) | 2011-05-26 |
| EA201290339A1 (ru) | 2012-12-28 |
| CN102724979A (zh) | 2012-10-10 |
| JP2013511525A (ja) | 2013-04-04 |
| PT2501379E (pt) | 2016-06-09 |
| EP2501379B1 (en) | 2016-03-23 |
| IL219786A (en) | 2016-05-31 |
| EP2501379A4 (en) | 2013-07-31 |
| PL2501379T3 (pl) | 2016-10-31 |
| US20120283279A1 (en) | 2012-11-08 |
| MX2012005758A (es) | 2012-06-19 |
| JP5834370B2 (ja) | 2015-12-16 |
| EA022637B1 (ru) | 2016-02-29 |
| BR112012011677A8 (pt) | 2018-06-12 |
| CN104382906A (zh) | 2015-03-04 |
| US20140303195A1 (en) | 2014-10-09 |
| IL219786A0 (en) | 2012-07-31 |
| SG10201407558TA (en) | 2015-01-29 |
| US20160008368A1 (en) | 2016-01-14 |
| BR112012011677A2 (pt) | 2018-03-20 |
| EP2501379A1 (en) | 2012-09-26 |
| ZA201203444B (en) | 2013-01-31 |
| AU2010322105B2 (en) | 2014-05-08 |
| ES2578191T3 (es) | 2016-07-21 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request |
Effective date: 20151102 |
|
| FZDE | Discontinued |
Effective date: 20180925 |