CA2739322A1 - Compounds for inflammation and immune-related uses - Google Patents

Compounds for inflammation and immune-related uses Download PDF

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Publication number
CA2739322A1
CA2739322A1 CA2739322A CA2739322A CA2739322A1 CA 2739322 A1 CA2739322 A1 CA 2739322A1 CA 2739322 A CA2739322 A CA 2739322A CA 2739322 A CA2739322 A CA 2739322A CA 2739322 A1 CA2739322 A1 CA 2739322A1
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CA
Canada
Prior art keywords
alkyl
alkenyl
alkynyl
compound
heteroaryl
Prior art date
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Abandoned
Application number
CA2739322A
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English (en)
French (fr)
Inventor
Shoujun Chen
Junyi Zhang
Jun Jiang
Gary Bohnert
Nha Vo
Qinglin Che
Zhiqiang Xia
Lijun Sun
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Synta Phamaceuticals Corp
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Synta Phamaceuticals Corp
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Filing date
Publication date
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Publication of CA2739322A1 publication Critical patent/CA2739322A1/en
Abandoned legal-status Critical Current

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Pain & Pain Management (AREA)
  • Urology & Nephrology (AREA)
  • Cardiology (AREA)
  • Rheumatology (AREA)
  • Endocrinology (AREA)
  • Dermatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Virology (AREA)
  • Psychology (AREA)
  • Vascular Medicine (AREA)
  • Obesity (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Transplantation (AREA)
CA2739322A 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses Abandoned CA2739322A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19483108P 2008-10-01 2008-10-01
US61/194,831 2008-10-01
PCT/US2009/005407 WO2010039237A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

Publications (1)

Publication Number Publication Date
CA2739322A1 true CA2739322A1 (en) 2010-04-08

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ID=41263687

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Application Number Title Priority Date Filing Date
CA2739322A Abandoned CA2739322A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

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US (3) US8314130B2 (enExample)
EP (1) EP2350064A1 (enExample)
JP (1) JP2012504604A (enExample)
AU (1) AU2009300317A1 (enExample)
CA (1) CA2739322A1 (enExample)
TW (1) TW201026693A (enExample)
WO (1) WO2010039237A1 (enExample)

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US8354398B2 (en) 2009-01-23 2013-01-15 Bristol-Myers Squibb Company Substituted isoxazole compounds
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
US10703722B2 (en) 2010-04-27 2020-07-07 Calcimedica, Inc. Compounds that modulate intracellular calcium
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WO2011139489A2 (en) 2010-04-27 2011-11-10 Calcimedica Inc. Compounds that modulate intracellular calcium
MX337711B (es) 2010-08-27 2016-03-15 Calcimedica Inc Compuestos que modulan el calcio intracelular.
SG192176A1 (en) * 2011-01-28 2013-08-30 4Sc Discovery Gmbh Il17 and ifn-gamma inhibition for the treatment of autoimmune inflammation
ES2660996T3 (es) * 2011-05-03 2018-03-27 PRCL Research Inc. Compuestos para la inflamación y usos relacionados con el sistema inmunitario
WO2012170931A2 (en) 2011-06-10 2012-12-13 Calcimedica, Inc. Compounds that modulate intracellular calcium
WO2013059677A1 (en) 2011-10-19 2013-04-25 Calcimedica, Inc. Compounds that modulate intracellular calcium
US9512116B2 (en) 2012-10-12 2016-12-06 Calcimedica, Inc. Compounds that modulate intracellular calcium
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US8314130B2 (en) 2012-11-20
EP2350064A1 (en) 2011-08-03
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US20130165451A9 (en) 2013-06-27
TW201026693A (en) 2010-07-16

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