CA2739322A1 - Compounds for inflammation and immune-related uses - Google Patents

Compounds for inflammation and immune-related uses Download PDF

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Publication number
CA2739322A1
CA2739322A1 CA2739322A CA2739322A CA2739322A1 CA 2739322 A1 CA2739322 A1 CA 2739322A1 CA 2739322 A CA2739322 A CA 2739322A CA 2739322 A CA2739322 A CA 2739322A CA 2739322 A1 CA2739322 A1 CA 2739322A1
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Canada
Prior art keywords
alkyl
alkenyl
alkynyl
compound
heteroaryl
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Abandoned
Application number
CA2739322A
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English (en)
French (fr)
Inventor
Shoujun Chen
Junyi Zhang
Jun Jiang
Gary Bohnert
Nha Vo
Qinglin Che
Zhiqiang Xia
Lijun Sun
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Synta Phamaceuticals Corp
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Synta Phamaceuticals Corp
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Publication date
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Publication of CA2739322A1 publication Critical patent/CA2739322A1/en
Abandoned legal-status Critical Current

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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurology (AREA)
  • Diabetes (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Immunology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pulmonology (AREA)
  • Communicable Diseases (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Rheumatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Cardiology (AREA)
  • Dermatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Virology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Obesity (AREA)
  • Vascular Medicine (AREA)
  • Psychology (AREA)
  • Emergency Medicine (AREA)
CA2739322A 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses Abandoned CA2739322A1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US19483108P 2008-10-01 2008-10-01
US61/194,831 2008-10-01
PCT/US2009/005407 WO2010039237A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

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CA2739322A1 true CA2739322A1 (en) 2010-04-08

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CA2739322A Abandoned CA2739322A1 (en) 2008-10-01 2009-10-01 Compounds for inflammation and immune-related uses

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US (3) US8314130B2 (enExample)
EP (1) EP2350064A1 (enExample)
JP (1) JP2012504604A (enExample)
AU (1) AU2009300317A1 (enExample)
CA (1) CA2739322A1 (enExample)
TW (1) TW201026693A (enExample)
WO (1) WO2010039237A1 (enExample)

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CN102361869A (zh) 2009-01-23 2012-02-22 百时美施贵宝公司 在治疗自身免疫性疾病和炎性疾病中作为s1p激动剂的取代的噁二唑衍生物
JP2012515789A (ja) 2009-01-23 2012-07-12 ブリストル−マイヤーズ スクイブ カンパニー スフィンゴシン−１−リン酸アゴニストとしてのピラゾール−１，２，４−オキサジアゾール誘導体
US8993612B2 (en) 2009-10-08 2015-03-31 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel and methods for treatment of non-small cell lung cancer
US8377970B2 (en) 2009-10-08 2013-02-19 Rhizen Pharmaceuticals Sa Modulators of calcium release-activated calcium channel
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JP5985611B2 (ja) * 2011-05-03 2016-09-06 シンタ ファーマシューティカルズ コーポレーション 炎症および免疫関連用途のための化合物
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