CA2692160A1 - Salts of potassium atp channel openers and uses thereof - Google Patents

Salts of potassium atp channel openers and uses thereof Download PDF

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Publication number
CA2692160A1
CA2692160A1 CA002692160A CA2692160A CA2692160A1 CA 2692160 A1 CA2692160 A1 CA 2692160A1 CA 002692160 A CA002692160 A CA 002692160A CA 2692160 A CA2692160 A CA 2692160A CA 2692160 A1 CA2692160 A1 CA 2692160A1
Authority
CA
Canada
Prior art keywords
formula
formulation
group
salt
subject
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002692160A
Other languages
English (en)
French (fr)
Inventor
Neil M. Cowen
Lain Dukes
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Essentialis Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2692160A1 publication Critical patent/CA2692160A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/18—Drugs for disorders of the alimentary tract or the digestive system for pancreatic disorders, e.g. pancreatic enzymes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00—Drugs for genital or sexual disorders; Contraceptives
    • A61P15/08—Drugs for genital or sexual disorders; Contraceptives for gonadal disorders or for enhancing fertility, e.g. inducers of ovulation or of spermatogenesis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives
CA002692160A 2007-07-02 2008-07-01 Salts of potassium atp channel openers and uses thereof Abandoned CA2692160A1 (en)

Applications Claiming Priority (9)

Application Number Priority Date Filing Date Title
US94762807P 2007-07-02 2007-07-02
US60/947,628 2007-07-02
US94920707P 2007-07-11 2007-07-11
US60/949,207 2007-07-11
US95085407P 2007-07-19 2007-07-19
US60/950,854 2007-07-19
US98625107P 2007-11-07 2007-11-07
US60/986,251 2007-11-07
PCT/US2008/068936 WO2009006483A1 (en) 2007-07-02 2008-07-01 Salts of potassium atp channel openers and uses thereof

Publications (1)

Publication Number Publication Date
CA2692160A1 true CA2692160A1 (en) 2009-01-08

Family

ID=40226526

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002692160A Abandoned CA2692160A1 (en) 2007-07-02 2008-07-01 Salts of potassium atp channel openers and uses thereof

Country Status (7)

Country Link
US (2) US20090062264A1 (enIt)
EP (1) EP2170341A4 (enIt)
JP (1) JP2010532383A (enIt)
CN (1) CN101795691A (enIt)
AU (1) AU2008272923A1 (enIt)
CA (1) CA2692160A1 (enIt)
WO (1) WO2009006483A1 (enIt)

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CA2578224A1 (en) * 2004-08-25 2006-03-09 Essentialis, Inc. Pharmaceutical formulations of potassium atp channel openers and uses thereof
US9757384B2 (en) 2005-04-06 2017-09-12 Essentialis, Inc. Methods for treating subjects with Prader-Willi syndrome or Smith-Magenis syndrome
AU2006335153B2 (en) * 2006-01-05 2012-03-15 Essentialis, Inc. Salts of potassium ATP channel openers and uses thereof
EP2343075A1 (en) * 2010-01-04 2011-07-13 Neurotec Pharma, S.L. Diazoxide for use in the treatment a central nervous system (CNS) autoimmune demyelinating disease
EP2612669A4 (en) 2010-08-31 2014-05-14 Snu R&Db Foundation USING THE FÖTAL REPROGRAMMING OF A PPAR AGONIST
EP2819675A4 (en) 2012-02-27 2015-07-22 Essentialis Inc SALTS OF KALIUM ATP CHANNEL OPENERS AND USES THEREOF
US20140364367A1 (en) * 2013-06-08 2014-12-11 Sedogen, Llc Methods of treating prader willi syndrome and conditions associated with low basal metabolic rate or hyperphagia using a katp channel opener
US20170189429A1 (en) * 2014-07-10 2017-07-06 Rhode Island Hospital Treating Arrhythmia with Mitochondrial-Targeted Antioxidants
WO2016077629A1 (en) 2014-11-14 2016-05-19 Essentialis, Inc. Methods for treating subjects with prader-willi syndrome or smith-magenis syndrome
CN107408694B (zh) * 2015-03-26 2020-12-29 太平洋水泥株式会社 二次电池用正极活性物质和其制造方法
CN106518804A (zh) * 2016-07-31 2017-03-22 北京梅尔森医药技术开发有限公司 一种二氮嗪新晶型及其制备方法
CN115877018A (zh) * 2022-08-05 2023-03-31 四川大学华西医院 一种孔蛋白在制备检测去氢表雄酮硫酸酯的试剂盒中的应用

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Also Published As

Publication number Publication date
WO2009006483A1 (en) 2009-01-08
EP2170341A4 (en) 2010-12-01
US20130040942A1 (en) 2013-02-14
EP2170341A1 (en) 2010-04-07
CN101795691A (zh) 2010-08-04
US20090062264A1 (en) 2009-03-05
AU2008272923A1 (en) 2009-01-08
JP2010532383A (ja) 2010-10-07

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Legal Events

Date Code Title Description
FZDE Discontinued

Effective date: 20140702