CA2652339A1 - Cdki pathway inhibitors as selective inhibitors of tumor cell growth - Google Patents
Cdki pathway inhibitors as selective inhibitors of tumor cell growth Download PDFInfo
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- CA2652339A1 CA2652339A1 CA002652339A CA2652339A CA2652339A1 CA 2652339 A1 CA2652339 A1 CA 2652339A1 CA 002652339 A CA002652339 A CA 002652339A CA 2652339 A CA2652339 A CA 2652339A CA 2652339 A1 CA2652339 A1 CA 2652339A1
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- alkyl
- hydrogen
- cdk3
- snx9
- halogen
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- A61K31/403—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with carbocyclic rings, e.g. carbazole
- A61K31/404—Indoles, e.g. pindolol
- A61K31/4045—Indole-alkylamines; Amides thereof, e.g. serotonin, melatonin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
Landscapes
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Epidemiology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines Containing Material From Animals Or Micro-Organisms (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US74722006P | 2006-05-15 | 2006-05-15 | |
| US60/747,220 | 2006-05-15 | ||
| US84996806P | 2006-10-06 | 2006-10-06 | |
| US60/849,968 | 2006-10-06 | ||
| PCT/US2007/011622 WO2007133772A2 (en) | 2006-05-15 | 2007-05-15 | Cdki pathway inhibitors as selective inhibitors of tumor cell growth |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2652339A1 true CA2652339A1 (en) | 2007-11-22 |
Family
ID=38694543
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002652339A Abandoned CA2652339A1 (en) | 2006-05-15 | 2007-05-15 | Cdki pathway inhibitors as selective inhibitors of tumor cell growth |
Country Status (6)
| Country | Link |
|---|---|
| US (1) | US20080200531A1 (enExample) |
| EP (1) | EP2023925A4 (enExample) |
| JP (1) | JP2009537532A (enExample) |
| AU (1) | AU2007249761A1 (enExample) |
| CA (1) | CA2652339A1 (enExample) |
| WO (1) | WO2007133772A2 (enExample) |
Families Citing this family (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| JP6245983B2 (ja) | 2010-08-11 | 2017-12-13 | ドレクセル ユニバーシティ | パーキンソン病におけるジスキネジアを治療するための新規ｄ３ドーパミン受容体アゴニスト |
| US9073851B2 (en) | 2011-10-28 | 2015-07-07 | Board Of Regents, The University Of Texas System | Compositions and methods for treating cancer |
| CN103468786B (zh) * | 2012-06-06 | 2017-06-13 | 上海吉凯基因化学技术有限公司 | 人cdkl3基因的用途及其相关药物 |
| WO2014089450A1 (en) * | 2012-12-06 | 2014-06-12 | Senex Biotechnology, Inc. | Specific inhibitors of cdk3 |
| US10584369B2 (en) * | 2013-01-11 | 2020-03-10 | Senex Biotechnology, Inc. | Cell-based methods for measuring activity of a protein inhibitor |
| ES2769780T3 (es) | 2013-10-28 | 2020-06-29 | Univ Drexel | Tratamientos novedosos para los trastornos de atención y cognitivos y para la demencia asociada a un trastorno neurodegenerativo |
| WO2018186366A1 (ja) | 2017-04-03 | 2018-10-11 | 京都薬品工業株式会社 | 新規サイクリン依存性キナーゼ８及び／又は１９阻害剤 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3915990A (en) * | 1973-03-13 | 1975-10-28 | Nelson Res & Dev | Tryptamines |
| US5849733A (en) * | 1996-05-10 | 1998-12-15 | Bristol-Myers Squibb Co. | 2-thio or 2-oxo flavopiridol analogs |
| DE69912808T2 (de) * | 1999-12-08 | 2004-09-30 | Centre National De La Recherche Scientifique (C.N.R.S.) | Verwendung von Hymenialdisin und dessen Derivaten zur Herstellung therapeutischer Mittel |
| EP1667720A1 (en) * | 2003-09-18 | 2006-06-14 | Novartis AG | Combination of a histone deacetylase inhibitor with a death receptor ligand |
| WO2006122546A1 (de) * | 2005-05-18 | 2006-11-23 | Forschungsverbund Berlin E.V. | Nicht-peptidische inhibitoren der akap-pka-wechselwirkung |
-
2007
- 2007-05-15 CA CA002652339A patent/CA2652339A1/en not_active Abandoned
- 2007-05-15 JP JP2009511024A patent/JP2009537532A/ja active Pending
- 2007-05-15 EP EP07809083A patent/EP2023925A4/en not_active Withdrawn
- 2007-05-15 WO PCT/US2007/011622 patent/WO2007133772A2/en not_active Ceased
- 2007-05-15 US US11/803,739 patent/US20080200531A1/en not_active Abandoned
- 2007-05-15 AU AU2007249761A patent/AU2007249761A1/en not_active Abandoned
Also Published As
| Publication number | Publication date |
|---|---|
| EP2023925A4 (en) | 2011-02-16 |
| JP2009537532A (ja) | 2009-10-29 |
| EP2023925A2 (en) | 2009-02-18 |
| US20080200531A1 (en) | 2008-08-21 |
| WO2007133772A2 (en) | 2007-11-22 |
| WO2007133772A3 (en) | 2008-11-20 |
| AU2007249761A1 (en) | 2007-11-22 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued |
Effective date: 20140515 |