CA2521776A1 - Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) - Google Patents
Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) Download PDFInfo
- Publication number
- CA2521776A1 CA2521776A1 CA002521776A CA2521776A CA2521776A1 CA 2521776 A1 CA2521776 A1 CA 2521776A1 CA 002521776 A CA002521776 A CA 002521776A CA 2521776 A CA2521776 A CA 2521776A CA 2521776 A1 CA2521776 A1 CA 2521776A1
- Authority
- CA
- Canada
- Prior art keywords
- phenylamino
- methylethyl
- fluorophenyl
- pyrrole
- dihydroxy
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- XUKUURHRXDUEBC-KAYWLYCHSA-N Atorvastatin Chemical compound C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CC[C@@H](O)C[C@@H](O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-KAYWLYCHSA-N 0.000 title abstract 3
- XUKUURHRXDUEBC-UHFFFAOYSA-N Atorvastatin Natural products C=1C=CC=CC=1C1=C(C=2C=CC(F)=CC=2)N(CCC(O)CC(O)CC(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 XUKUURHRXDUEBC-UHFFFAOYSA-N 0.000 title abstract 2
- 229960005370 atorvastatin Drugs 0.000 title abstract 2
- 229910052791 calcium Inorganic materials 0.000 title 1
- 239000011575 calcium Substances 0.000 title 1
- SAGAISAEDMDRFK-UHFFFAOYSA-N 2-hydroxy-7-[2-hydroxy-3-phenyl-4-(phenylcarbamoyl)-5-propan-2-ylpyrrol-1-yl]heptanoic acid Chemical compound C=1C=CC=CC=1C1=C(O)N(CCCCCC(O)C(O)=O)C(C(C)C)=C1C(=O)NC1=CC=CC=C1 SAGAISAEDMDRFK-UHFFFAOYSA-N 0.000 abstract 1
- 208000024827 Alzheimer disease Diseases 0.000 abstract 1
- 208000035150 Hypercholesterolemia Diseases 0.000 abstract 1
- 208000031226 Hyperlipidaemia Diseases 0.000 abstract 1
- 208000001132 Osteoporosis Diseases 0.000 abstract 1
- 238000001069 Raman spectroscopy Methods 0.000 abstract 1
- 159000000007 calcium salts Chemical class 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 239000008194 pharmaceutical composition Substances 0.000 abstract 1
- 238000000634 powder X-ray diffraction Methods 0.000 abstract 1
- 238000000371 solid-state nuclear magnetic resonance spectroscopy Methods 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Pyrrole Compounds (AREA)
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US30204901P | 2001-06-29 | 2001-06-29 | |
US60/302,049 | 2001-06-29 | ||
CA002450111A CA2450111C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
Related Parent Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002450111A Division CA2450111C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
Publications (2)
Publication Number | Publication Date |
---|---|
CA2521776A1 true CA2521776A1 (fr) | 2003-01-16 |
CA2521776C CA2521776C (fr) | 2006-04-25 |
Family
ID=35452260
Family Applications (14)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002521891A Expired - Fee Related CA2521891C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002522899A Expired - Fee Related CA2522899C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521953A Expired - Fee Related CA2521953C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521908A Expired - Fee Related CA2521908C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521958A Expired - Fee Related CA2521958C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521792A Expired - Fee Related CA2521792C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521933A Expired - Fee Related CA2521933C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521993A Abandoned CA2521993A1 (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide¬r-(r*,r*)|-2-(4-fluorop henyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-¬(phenylamino) carbonyl|-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521980A Expired - Fee Related CA2521980C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide[r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521828A Expired - Fee Related CA2521828C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521776A Expired - Fee Related CA2521776C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521956A Expired - Fee Related CA2521956C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521833A Expired - Fee Related CA2521833C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521887A Expired - Fee Related CA2521887C (fr) | 2001-06-29 | 2002-05-21 | Crystalline forms of [r-(r*,r*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid calcium salt(2:1)(atorvastatin) |
Family Applications Before (10)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002521891A Expired - Fee Related CA2521891C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002522899A Expired - Fee Related CA2522899C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521953A Expired - Fee Related CA2521953C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521908A Expired - Fee Related CA2521908C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521958A Expired - Fee Related CA2521958C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521792A Expired - Fee Related CA2521792C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521933A Expired - Fee Related CA2521933C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521993A Abandoned CA2521993A1 (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide¬r-(r*,r*)|-2-(4-fluorop henyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-¬(phenylamino) carbonyl|-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521980A Expired - Fee Related CA2521980C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide[r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521828A Expired - Fee Related CA2521828C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
Family Applications After (3)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002521956A Expired - Fee Related CA2521956C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521833A Expired - Fee Related CA2521833C (fr) | 2001-06-29 | 2002-05-21 | Formes cristallines de sel hemicalcique d'acide [r-(r*,r*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1h-pyrrole-1-heptanoique (2:1)(atorvastatine) |
CA002521887A Expired - Fee Related CA2521887C (fr) | 2001-06-29 | 2002-05-21 | Crystalline forms of [r-(r*,r*)]-2-(4-fluorophenyl)-beta, delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[phenylamino)carbonyl]-1h-pyrrole-1-heptanoic acid calcium salt(2:1)(atorvastatin) |
Country Status (1)
Country | Link |
---|---|
CA (14) | CA2521891C (fr) |
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8080672B2 (en) | 2005-12-13 | 2011-12-20 | Teva Pharmaceutical Industries Ltd. | Crystal form of atorvastatin hemi-calcium and processes for preparation thereof |
-
2002
- 2002-05-21 CA CA002521891A patent/CA2521891C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002522899A patent/CA2522899C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521953A patent/CA2521953C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521908A patent/CA2521908C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521958A patent/CA2521958C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521792A patent/CA2521792C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521933A patent/CA2521933C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521993A patent/CA2521993A1/fr not_active Abandoned
- 2002-05-21 CA CA002521980A patent/CA2521980C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521828A patent/CA2521828C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521776A patent/CA2521776C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521956A patent/CA2521956C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521833A patent/CA2521833C/fr not_active Expired - Fee Related
- 2002-05-21 CA CA002521887A patent/CA2521887C/fr not_active Expired - Fee Related
Cited By (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US8080672B2 (en) | 2005-12-13 | 2011-12-20 | Teva Pharmaceutical Industries Ltd. | Crystal form of atorvastatin hemi-calcium and processes for preparation thereof |
Also Published As
Publication number | Publication date |
---|---|
CA2521833A1 (fr) | 2003-01-16 |
CA2521887A1 (fr) | 2003-01-16 |
CA2521980A1 (fr) | 2003-01-16 |
CA2521828A1 (fr) | 2003-01-16 |
CA2521993A1 (fr) | 2003-01-16 |
CA2521956C (fr) | 2006-04-25 |
CA2521953C (fr) | 2006-03-14 |
CA2521958C (fr) | 2006-08-29 |
CA2521887C (fr) | 2006-04-25 |
CA2521953A1 (fr) | 2003-01-16 |
CA2521908A1 (fr) | 2003-01-16 |
CA2522899A1 (fr) | 2003-01-16 |
CA2521891C (fr) | 2006-04-25 |
CA2521792A1 (fr) | 2003-01-16 |
CA2521908C (fr) | 2006-04-25 |
CA2521956A1 (fr) | 2003-01-16 |
CA2522899C (fr) | 2006-04-25 |
CA2521776C (fr) | 2006-04-25 |
CA2521980C (fr) | 2006-08-29 |
CA2521933C (fr) | 2006-03-21 |
CA2521828C (fr) | 2006-04-25 |
CA2521833C (fr) | 2006-04-25 |
CA2521891A1 (fr) | 2003-01-16 |
CA2521933A1 (fr) | 2003-01-16 |
CA2521792C (fr) | 2006-04-25 |
CA2521958A1 (fr) | 2003-01-16 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
MKLA | Lapsed |
Effective date: 20190521 |