CA2509374A1 - Glycogen synthase kinase-3 inhibitors - Google Patents
Glycogen synthase kinase-3 inhibitors Download PDFInfo
- Publication number
- CA2509374A1 CA2509374A1 CA002509374A CA2509374A CA2509374A1 CA 2509374 A1 CA2509374 A1 CA 2509374A1 CA 002509374 A CA002509374 A CA 002509374A CA 2509374 A CA2509374 A CA 2509374A CA 2509374 A1 CA2509374 A1 CA 2509374A1
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- acid
- amino acid
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- C—CHEMISTRY; METALLURGY
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- C07K—PEPTIDES
- C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
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- C07K14/46—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K7/00—Peptides having 5 to 20 amino acids in a fully defined sequence; Derivatives thereof
- C07K7/04—Linear peptides containing only normal peptide links
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- C—CHEMISTRY; METALLURGY
- C12—BIOCHEMISTRY; BEER; SPIRITS; WINE; VINEGAR; MICROBIOLOGY; ENZYMOLOGY; MUTATION OR GENETIC ENGINEERING
- C12Q—MEASURING OR TESTING PROCESSES INVOLVING ENZYMES, NUCLEIC ACIDS OR MICROORGANISMS; COMPOSITIONS OR TEST PAPERS THEREFOR; PROCESSES OF PREPARING SUCH COMPOSITIONS; CONDITION-RESPONSIVE CONTROL IN MICROBIOLOGICAL OR ENZYMOLOGICAL PROCESSES
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Landscapes
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| US48271903P | 2003-06-27 | 2003-06-27 | |
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| US7378432B2 (en) * | 2001-09-14 | 2008-05-27 | Tel Aviv University Future Technology Development L.P. | Glycogen synthase kinase-3 inhibitors |
| JP2006514104A (ja) * | 2002-12-12 | 2006-04-27 | テル アヴィヴ ユニヴァーシティ フューチャー テクノロジー ディヴェロップメント エル．ピー． | グリコーゲンシンターゼキナーゼ−３阻害剤 |
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| WO2009154697A2 (en) | 2008-05-28 | 2009-12-23 | Massachusetts Institute Of Technology | Disc-1 pathway activators in the control of neurogenesis |
| AU2008258150B1 (en) * | 2008-12-16 | 2009-03-19 | Jorge Miguel Pereira | An Improved Knee Pad |
| WO2010098888A1 (en) * | 2009-02-27 | 2010-09-02 | Massachusetts Institute Of Technology | Uses of chemicals to modulate gsk-3 signaling for treatment of bipolar disorder and other brain disorders |
| WO2012101599A2 (en) | 2011-01-27 | 2012-08-02 | Ramot At Tel-Aviv University Ltd. | Glycogen synthase kinase-3 inhibitors |
| WO2012101601A1 (en) | 2011-01-27 | 2012-08-02 | Ramot At Tel-Aviv University Ltd. | Glycogen synthase kinase-3 inhibitors |
| US9718859B2 (en) | 2013-06-24 | 2017-08-01 | Ramot At Tel-Aviv University Ltd. | Glycogen synthase kinase-3 inhibitors |
| WO2015155738A2 (en) | 2014-04-09 | 2015-10-15 | Christopher Rudd | Use of gsk-3 inhibitors or activators which modulate pd-1 or t-bet expression to modulate t cell immunity |
| SI3215518T1 (sl) | 2014-10-29 | 2021-08-31 | Bicyclerd Limited | Biciklični peptidni ligandi, značilni za MT1-MMP |
| JP2020502238A (ja) * | 2016-12-23 | 2020-01-23 | バイスクルアールディー・リミテッド | 新規連結構造を有するペプチド誘導体 |
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| CN111183147B (zh) | 2017-08-04 | 2024-07-05 | 拜斯科技术开发有限公司 | Cd137特异性的双环肽配体 |
| WO2019162682A1 (en) | 2018-02-23 | 2019-08-29 | Bicycletx Limited | Multimeric bicyclic peptide ligands |
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| WO2020128526A1 (en) | 2018-12-21 | 2020-06-25 | Bicycletx Limited | Bicyclic peptide ligands specific for pd-l1 |
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| AU2001280229B2 (en) | 2000-08-21 | 2006-12-07 | Pacific Corporation | Novel thiourea derivatives and the pharmaceutical compositions containing the same |
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- 2003-12-11 KR KR1020057010710A patent/KR20050091716A/ko not_active Ceased
- 2003-12-11 AU AU2003286411A patent/AU2003286411A1/en not_active Abandoned
- 2003-12-11 US US10/538,171 patent/US7446092B2/en not_active Expired - Lifetime
- 2003-12-11 EP EP03777156.5A patent/EP1569956B1/en not_active Expired - Lifetime
- 2003-12-11 CA CA002509374A patent/CA2509374A1/en not_active Abandoned
- 2003-12-11 WO PCT/IL2003/001057 patent/WO2004052404A2/en not_active Ceased
-
2008
- 2008-05-29 US US12/155,087 patent/US7833974B2/en not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| WO2004052404A3 (en) | 2004-07-29 |
| EP1569956B1 (en) | 2014-02-26 |
| US20090062180A1 (en) | 2009-03-05 |
| AU2003286411A1 (en) | 2004-06-30 |
| US7446092B2 (en) | 2008-11-04 |
| US20060135408A1 (en) | 2006-06-22 |
| EP1569956A2 (en) | 2005-09-07 |
| KR20050091716A (ko) | 2005-09-15 |
| WO2004052404A2 (en) | 2004-06-24 |
| JP2006514104A (ja) | 2006-04-27 |
| US7833974B2 (en) | 2010-11-16 |
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| FZDE | Discontinued |