CA2487073A1 - Methods for using jnk inhibitors for treating or preventing disease-related wasting - Google Patents
Methods for using jnk inhibitors for treating or preventing disease-related wasting Download PDFInfo
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- CA2487073A1 CA2487073A1 CA002487073A CA2487073A CA2487073A1 CA 2487073 A1 CA2487073 A1 CA 2487073A1 CA 002487073 A CA002487073 A CA 002487073A CA 2487073 A CA2487073 A CA 2487073A CA 2487073 A1 CA2487073 A1 CA 2487073A1
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- heterocycle
- alkyl
- aryl
- disease
- arylalkyl
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Landscapes
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- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Medicinal Chemistry (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
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- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
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- Physical Education & Sports Medicine (AREA)
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- Tropical Medicine & Parasitology (AREA)
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- Dermatology (AREA)
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Thiazole And Isothizaole Compounds (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38320202P | 2002-05-24 | 2002-05-24 | |
| US60/383,202 | 2002-05-24 | ||
| US10/443,263 | 2003-05-22 | ||
| US10/443,263 US20040034084A1 (en) | 2002-05-24 | 2003-05-22 | Methods for using JNK inhibitors for treating or preventing disease-related wasting |
| PCT/US2003/016333 WO2003099221A2 (en) | 2002-05-24 | 2003-05-23 | Methods for using jnk inhibitors for treating or preventing disease-related wasting |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2487073A1 true CA2487073A1 (en) | 2003-12-04 |
Family
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Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002487073A Abandoned CA2487073A1 (en) | 2002-05-24 | 2003-05-23 | Methods for using jnk inhibitors for treating or preventing disease-related wasting |
Country Status (10)
| Country | Link |
|---|---|
| US (1) | US20040034084A1 (enExample) |
| EP (1) | EP1507528A4 (enExample) |
| JP (1) | JP2005535594A (enExample) |
| CN (1) | CN1668299A (enExample) |
| AU (1) | AU2003256259A1 (enExample) |
| CA (1) | CA2487073A1 (enExample) |
| IL (1) | IL165359A0 (enExample) |
| MX (1) | MXPA04011599A (enExample) |
| NZ (1) | NZ537055A (enExample) |
| WO (1) | WO2003099221A2 (enExample) |
Families Citing this family (18)
| Publication number | Priority date | Publication date | Assignee | Title |
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| JP4219289B2 (ja) * | 2004-03-10 | 2009-02-04 | 独立行政法人科学技術振興機構 | 多環性ケトン化合物及びその製造方法 |
| US20110008327A1 (en) | 2004-03-29 | 2011-01-13 | Cheng Jin Q | Compositions including triciribine and epidermal growth factor receptor inhibitor compounds or salts thereof and methods of use thereof |
| US20100028339A1 (en) | 2004-03-29 | 2010-02-04 | Cheng Jin Q | Compositions including triciribine and trastuzumab and methods of use thereof |
| US20100009928A1 (en) | 2004-03-29 | 2010-01-14 | Cheng Jin Q | Compositions including triciribine and taxanes and methods of use thereof |
| US20100173864A1 (en) | 2004-03-29 | 2010-07-08 | Cheng Jin Q | Compositions including triciribine and one or more platinum compounds and methods of use thereof |
| LT2574341T (lt) | 2004-03-29 | 2017-09-11 | University Of South Florida | Navikų ir vėžio efektyvus gydymas triciribino fosfatu |
| US20100009929A1 (en) | 2004-03-29 | 2010-01-14 | Cheng Jin Q | Compositions including triciribine and bortezomib and derivatives thereof and methods of use thereof |
| PE20060373A1 (es) * | 2004-06-24 | 2006-04-29 | Smithkline Beecham Corp | Derivados 3-piperidinil-7-carboxamida-indazol como inhibidores de la actividad cinasa de ikk2 |
| KR20070038565A (ko) * | 2004-07-27 | 2007-04-10 | 노파르티스 아게 | Hsp90의 억제제 |
| MX2007001155A (es) * | 2004-07-29 | 2007-08-14 | Creabilis Therapeutics Spa | Uso de inhibidores de k-252a y de quinasa para la prevencion o el tratamiento de patologias asociadas con hmgb1. |
| EP1676574A3 (en) | 2004-12-30 | 2006-07-26 | Johnson & Johnson Vision Care, Inc. | Methods for promoting survival of transplanted tissues and cells |
| NZ590283A (en) | 2008-07-14 | 2012-11-30 | Gilead Sciences Inc | Imidazolylpyrimidine compounds as hdac and / or cdk inhibitors |
| AU2009271019A1 (en) | 2008-07-14 | 2010-01-21 | Gilead Sciences, Inc. | Fused heterocyclyc inhibitors of histone deacetylase and/or cyclin-dependent kinases |
| EP2303841A1 (en) | 2008-07-14 | 2011-04-06 | Gilead Sciences, Inc. | Oxindolyl inhibitor compounds |
| CA2731323A1 (en) | 2008-07-28 | 2010-02-04 | Gilead Sciences, Inc. | Cycloalkylidene and heterocycloalkylidene histone deacetylase inhibitor compounds |
| CA2763167A1 (en) | 2009-06-08 | 2010-12-16 | Gilead Sciences, Inc. | Cycloalkylcarbamate benzamide aniline hdac inhibitor compounds |
| EP2440519A1 (en) | 2009-06-08 | 2012-04-18 | Gilead Sciences, Inc. | Alkanoylamino benzamide aniline hdac inihibitor compounds |
| US10624948B2 (en) * | 2013-06-26 | 2020-04-21 | Xigen Inflammation Ltd. | Use of cell-permeable peptide inhibitors of the JNK signal transduction pathway for the treatment of various diseases |
Family Cites Families (16)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3994890A (en) * | 1974-01-31 | 1976-11-30 | Chugai Seiyaku Kabushiki Kaisha | 1-Aminoalkyl, 3-phenyl indazoles |
| US4198518A (en) * | 1977-09-02 | 1980-04-15 | Ciba-Geigy Corporation | Process for the production of 3-substituted pyrazolanthrones |
| JPS57109787A (en) * | 1980-12-26 | 1982-07-08 | Chugai Pharmaceut Co Ltd | Pyrazoloindazole derivative |
| US4788195A (en) * | 1986-01-13 | 1988-11-29 | American Cyanamid Company | 4,5,6-substituted-N-(substituted-phenyl)-2-pyrimidinamines |
| US4973690A (en) * | 1988-04-12 | 1990-11-27 | Ciba-Geigy Corporation | Novel ureas |
| US4966622A (en) * | 1988-04-12 | 1990-10-30 | Ciba-Geigy Corporation | N-phenyl-N-pyrimidin-2-ylureas |
| JP2515162B2 (ja) * | 1990-02-23 | 1996-07-10 | 富士写真フイルム株式会社 | メチン化合物 |
| GB9016449D0 (en) * | 1990-07-26 | 1990-09-12 | Ici Plc | Anionic compounds |
| DE69230387T2 (de) * | 1991-04-22 | 2000-06-29 | Fuji Photo Film Co., Ltd. | Photographische Silberhalogenidmaterialien und Verfahren zu ihrer Verarbeitung |
| JP2692021B2 (ja) * | 1991-09-13 | 1997-12-17 | 富士写真フイルム株式会社 | ハロゲン化銀感光材料 |
| US5516775A (en) * | 1992-08-31 | 1996-05-14 | Ciba-Geigy Corporation | Further use of pyrimidine derivatives |
| WO1996004909A1 (en) * | 1994-08-12 | 1996-02-22 | Takeda Chemical Industries, Ltd. | Use of quinone and hydroquinone derivatives for the teatment of cachexia |
| AP1147A (en) * | 1996-05-03 | 2003-02-25 | Pfizer | Substituted indazole derivatives and related compounds. |
| US6162613A (en) * | 1998-02-18 | 2000-12-19 | Vertex Pharmaceuticals, Inc. | Methods for designing inhibitors of serine/threonine-kinases and tyrosine kinases |
| US6897231B2 (en) * | 2000-07-31 | 2005-05-24 | Signal Pharmaceuticals, Inc. | Indazole derivatives as JNK inhibitors and compositions and methods related thereto |
| US6987184B2 (en) * | 2001-02-15 | 2006-01-17 | Signal Pharmaceuticals, Llc | Isothiazoloanthrones, isoxazoloanthrones, isoindolanthrones and derivatives thereof as JNK inhibitors and compositions and methods related |
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2003
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- 2003-05-23 IL IL16535903A patent/IL165359A0/xx unknown
- 2003-05-23 CA CA002487073A patent/CA2487073A1/en not_active Abandoned
- 2003-05-23 JP JP2004506748A patent/JP2005535594A/ja active Pending
- 2003-05-23 WO PCT/US2003/016333 patent/WO2003099221A2/en not_active Ceased
- 2003-05-23 MX MXPA04011599A patent/MXPA04011599A/es not_active Application Discontinuation
- 2003-05-23 CN CNA038166992A patent/CN1668299A/zh active Pending
- 2003-05-23 AU AU2003256259A patent/AU2003256259A1/en not_active Abandoned
- 2003-05-23 NZ NZ537055A patent/NZ537055A/en unknown
- 2003-05-23 EP EP03755458A patent/EP1507528A4/en not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| CN1668299A (zh) | 2005-09-14 |
| IL165359A0 (en) | 2006-01-15 |
| EP1507528A2 (en) | 2005-02-23 |
| WO2003099221A2 (en) | 2003-12-04 |
| JP2005535594A (ja) | 2005-11-24 |
| EP1507528A4 (en) | 2009-12-30 |
| NZ537055A (en) | 2006-07-28 |
| MXPA04011599A (es) | 2005-07-27 |
| WO2003099221A3 (en) | 2004-06-24 |
| AU2003256259A1 (en) | 2003-12-12 |
| US20040034084A1 (en) | 2004-02-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| EEER | Examination request | ||
| FZDE | Discontinued | ||
| FZDE | Discontinued |
Effective date: 20100525 |