CA2403828A1 - Inhibiteurs de p38 - Google Patents
Inhibiteurs de p38 Download PDFInfo
- Publication number
- CA2403828A1 CA2403828A1 CA002403828A CA2403828A CA2403828A1 CA 2403828 A1 CA2403828 A1 CA 2403828A1 CA 002403828 A CA002403828 A CA 002403828A CA 2403828 A CA2403828 A CA 2403828A CA 2403828 A1 CA2403828 A1 CA 2403828A1
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- Prior art keywords
- optionally substituted
- compound
- disease
- treat
- prevent
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Abandoned
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Classifications
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- C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D213/60—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D489/00—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula:
- C07D489/02—Heterocyclic compounds containing 4aH-8, 9 c- Iminoethano-phenanthro [4, 5-b, c, d] furan ring systems, e.g. derivatives of [4, 5-epoxy]-morphinan of the formula: with oxygen atoms attached in positions 3 and 6, e.g. morphine, morphinone
- C07D489/04—Salts; Organic complexes
Landscapes
- Health & Medical Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Diabetes (AREA)
- Immunology (AREA)
- Neurology (AREA)
- Hematology (AREA)
- Physical Education & Sports Medicine (AREA)
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- Neurosurgery (AREA)
- Rheumatology (AREA)
- Orthopedic Medicine & Surgery (AREA)
- Cardiology (AREA)
- Pulmonology (AREA)
- Heart & Thoracic Surgery (AREA)
- Pain & Pain Management (AREA)
- Oncology (AREA)
- Urology & Nephrology (AREA)
- Dermatology (AREA)
- Communicable Diseases (AREA)
- Endocrinology (AREA)
- Hospice & Palliative Care (AREA)
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- Transplantation (AREA)
- Psychology (AREA)
- Psychiatry (AREA)
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- Gastroenterology & Hepatology (AREA)
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US19135800P | 2000-03-22 | 2000-03-22 | |
| US60/191,358 | 2000-03-22 | ||
| PCT/US2001/009256 WO2001070695A1 (fr) | 2000-03-22 | 2001-03-22 | Inhibiteurs de p38 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2403828A1 true CA2403828A1 (fr) | 2001-09-27 |
Family
ID=22705152
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002403828A Abandoned CA2403828A1 (fr) | 2000-03-22 | 2001-03-22 | Inhibiteurs de p38 |
Country Status (6)
| Country | Link |
|---|---|
| JP (1) | JP2003528084A (fr) |
| AU (1) | AU2001247700A1 (fr) |
| CA (1) | CA2403828A1 (fr) |
| MX (1) | MXPA02009319A (fr) |
| TW (1) | TWI282334B (fr) |
| WO (1) | WO2001070695A1 (fr) |
Families Citing this family (8)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| MXPA03001256A (es) | 2000-08-11 | 2004-12-06 | Vertex Pharma | Inhibidores de p38. |
| GB0124933D0 (en) | 2001-10-17 | 2001-12-05 | Glaxo Group Ltd | Chemical compounds |
| SI1474395T1 (sl) * | 2002-02-12 | 2008-02-29 | Smithkline Beecham Corp | Nikotinamidni derivati, uporabni kot inhibitorji p38 |
| GB0308201D0 (en) | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
| GB0308186D0 (en) | 2003-04-09 | 2003-05-14 | Smithkline Beecham Corp | Novel compounds |
| GB0318814D0 (en) * | 2003-08-11 | 2003-09-10 | Smithkline Beecham Corp | Novel compounds |
| GB0908317D0 (en) * | 2009-05-14 | 2009-06-24 | Argenta Discovery Ltd | Pharmaceutical compounds and compositions |
| WO2017151409A1 (fr) | 2016-02-29 | 2017-09-08 | University Of Florida Research Foundation, Incorporated | Méthodes de chimiothérapie |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US6147080A (en) * | 1996-12-18 | 2000-11-14 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
| US5945418A (en) * | 1996-12-18 | 1999-08-31 | Vertex Pharmaceuticals Incorporated | Inhibitors of p38 |
| JP2002502380A (ja) * | 1997-05-22 | 2002-01-22 | ジー．ディー．サール アンド カンパニー | ｐ３８キナーゼ阻害剤としてのピラゾール誘導体 |
| IL136768A0 (en) * | 1997-12-22 | 2001-06-14 | Bayer Ag | INHIBITION OF p38 KINASE ACTIVITY USING ARYL AND HETEROARYL SUBSTITUTED HETEROCYCLIC UREAS |
| MY132496A (en) * | 1998-05-11 | 2007-10-31 | Vertex Pharma | Inhibitors of p38 |
-
2001
- 2001-03-22 CA CA002403828A patent/CA2403828A1/fr not_active Abandoned
- 2001-03-22 MX MXPA02009319A patent/MXPA02009319A/es not_active Application Discontinuation
- 2001-03-22 WO PCT/US2001/009256 patent/WO2001070695A1/fr active Application Filing
- 2001-03-22 TW TWNOVELCOMA patent/TWI282334B/zh not_active IP Right Cessation
- 2001-03-22 AU AU2001247700A patent/AU2001247700A1/en not_active Abandoned
- 2001-03-22 JP JP2001568907A patent/JP2003528084A/ja not_active Withdrawn
Also Published As
| Publication number | Publication date |
|---|---|
| WO2001070695A8 (fr) | 2001-11-29 |
| AU2001247700A1 (en) | 2001-10-03 |
| TWI282334B (en) | 2007-06-11 |
| JP2003528084A (ja) | 2003-09-24 |
| WO2001070695A1 (fr) | 2001-09-27 |
| MXPA02009319A (es) | 2003-03-12 |
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