CA2380007A1 - Methods of inhibiting osteoclast activity - Google Patents
Methods of inhibiting osteoclast activity Download PDFInfo
- Publication number
- CA2380007A1 CA2380007A1 CA002380007A CA2380007A CA2380007A1 CA 2380007 A1 CA2380007 A1 CA 2380007A1 CA 002380007 A CA002380007 A CA 002380007A CA 2380007 A CA2380007 A CA 2380007A CA 2380007 A1 CA2380007 A1 CA 2380007A1
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- inhibitor
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- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
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- A61K38/1703—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans from vertebrates
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- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1005—Tetrapeptides with the first amino acid being neutral and aliphatic
- C07K5/1013—Tetrapeptides with the first amino acid being neutral and aliphatic the side chain containing O or S as heteroatoms, e.g. Cys, Ser
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
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- C07K5/1002—Tetrapeptides with the first amino acid being neutral
- C07K5/1016—Tetrapeptides with the first amino acid being neutral and aromatic or cycloaliphatic
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/10—Tetrapeptides
- C07K5/1021—Tetrapeptides with the first amino acid being acidic
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
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- Marine Sciences & Fisheries (AREA)
- Cell Biology (AREA)
- Toxicology (AREA)
- Emergency Medicine (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
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Priority Applications (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| CA002647796A CA2647796A1 (en) | 1999-07-28 | 2000-07-28 | Method of inhibiting osteoclast activity |
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US14609499P | 1999-07-28 | 1999-07-28 | |
| US60/146,094 | 1999-07-28 | ||
| PCT/US2000/020502 WO2001008677A1 (en) | 1999-07-28 | 2000-07-28 | Methods of inhibiting osteoclast activity |
Related Child Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| CA002647796A Division CA2647796A1 (en) | 1999-07-28 | 2000-07-28 | Method of inhibiting osteoclast activity |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| CA2380007A1 true CA2380007A1 (en) | 2001-02-08 |
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Family Applications (2)
| Application Number | Title | Priority Date | Filing Date |
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| CA002380007A Abandoned CA2380007A1 (en) | 1999-07-28 | 2000-07-28 | Methods of inhibiting osteoclast activity |
| CA002647796A Abandoned CA2647796A1 (en) | 1999-07-28 | 2000-07-28 | Method of inhibiting osteoclast activity |
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| CA002647796A Abandoned CA2647796A1 (en) | 1999-07-28 | 2000-07-28 | Method of inhibiting osteoclast activity |
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| JP (1) | JP4790179B2 (https=) |
| AT (1) | ATE448781T1 (https=) |
| AU (2) | AU778190B2 (https=) |
| CA (2) | CA2380007A1 (https=) |
| DE (1) | DE60043346D1 (https=) |
| WO (1) | WO2001008677A1 (https=) |
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| Publication number | Priority date | Publication date | Assignee | Title |
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| AU777634B2 (en) * | 1999-07-28 | 2004-10-28 | Kazuhiro Aoki | Methods of inhibiting osteoclastogenesis |
| WO2002024896A2 (en) | 2000-09-22 | 2002-03-28 | Immunex Corporation | Screening assays for agonists or antagonists of receptor activat or of nf-kb |
| ATE399790T1 (de) | 2001-07-03 | 2008-07-15 | Febit Biotech Gmbh | Zweistufige schutzgruppen für die synthese von biopolymeren |
| KR101560844B1 (ko) * | 2007-06-04 | 2015-10-15 | 벤-구리온 유니버시티 오브 더 네게브 리서치 앤드 디벨럽먼트 어쏘러티 | 트라이-아릴계 화합물 및 이를 포함하는 조성물 |
| US20100260680A1 (en) * | 2007-06-05 | 2010-10-14 | Oriental Yeast Co., Ltd. | Novel bone mass increasing agent |
| RU2010150688A (ru) * | 2008-05-13 | 2012-06-20 | Ашок Ранганат ШЕЛАР (IN) | Медицинские применения гидразонов бензойной кислоты, синтезированных на основе стероидного тигогенина |
| WO2013035852A1 (ja) | 2011-09-09 | 2013-03-14 | 住友電気工業株式会社 | 給電システム及び接続コネクタ |
| WO2014062625A1 (en) * | 2012-10-15 | 2014-04-24 | Iowa State University Research Foundation, Inc. | Tackifier compounds and methods of using the same |
| CN105209427B (zh) * | 2013-03-15 | 2018-05-25 | 特罗菲克斯制药股份有限公司 | 非肽bdnf神经营养蛋白模拟物 |
| CN105189449A (zh) | 2013-03-15 | 2015-12-23 | 特罗菲克斯制药股份有限公司 | 非肽bdnf神经营养蛋白模拟物 |
| US9321803B2 (en) * | 2013-07-12 | 2016-04-26 | Children's Hospital Medical Center | Compositions and methods for inhibiting norovirus infection |
| MX2016005995A (es) | 2013-11-05 | 2016-08-17 | Ben-Gurion Univ Of The Negev Res And Dev Authority | Compuestos para el tratamiento de diabetes y complicaciones de la enfermedad derivadas de la misma. |
| US10077257B2 (en) | 2015-04-06 | 2018-09-18 | Iowa State University Research Foundation, Inc. | Aziridinated triglycerides and polymers formed therefrom |
| US10392471B2 (en) | 2015-05-14 | 2019-08-27 | Iowa State University Research Foundation, Inc. | Polymers and methods of making the same |
| EP3299382B1 (en) * | 2015-05-20 | 2023-04-26 | Osaka University | Oligopeptide having proinflammatory cytokine secretion-inhibiting activity |
| EP3600397A4 (en) | 2017-03-28 | 2021-01-27 | Children's Hospital Medical Center | NOROVIRUS PARTICLE VACCINES AND THEIR MANUFACTURING AND USE PROCEDURES |
| CN110229118B (zh) | 2019-06-28 | 2021-03-02 | 深圳市三启药物开发有限公司 | 腙酰胺类衍生物及其在制备抗骨质疏松药物中的应用 |
| CN111686116B (zh) * | 2020-06-08 | 2021-05-04 | 广东省微生物研究所（广东省微生物分析检测中心） | 孕甾烷衍生物在制备破骨细胞分化抑制剂中的应用 |
Family Cites Families (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE69740107D1 (de) * | 1996-12-23 | 2011-03-10 | Immunex Corp | Rezeptor aktivator von nf-kappa b, rezeptor is mitglied der tnf rezeptor superfamilie |
| AU762574B2 (en) * | 1998-05-14 | 2003-06-26 | Immunex Corporation | Method of inhibiting osteoclast activity |
| WO2000001349A2 (en) * | 1998-07-01 | 2000-01-13 | The Trustees Of The University Of Pennsylvania | Cavity induced allosteric modification of intermolecular interactions and methods of identifying compounds that effect the same |
| HUP0103578A3 (en) * | 1998-09-15 | 2005-11-28 | Pharmexa As | Method for down-regulating osteoprotegerin ligand activity |
| AU777634B2 (en) * | 1999-07-28 | 2004-10-28 | Kazuhiro Aoki | Methods of inhibiting osteoclastogenesis |
-
2000
- 2000-07-28 AU AU63846/00A patent/AU778190B2/en not_active Ceased
- 2000-07-28 DE DE60043346T patent/DE60043346D1/de not_active Expired - Lifetime
- 2000-07-28 CA CA002380007A patent/CA2380007A1/en not_active Abandoned
- 2000-07-28 JP JP2001513407A patent/JP4790179B2/ja not_active Expired - Fee Related
- 2000-07-28 WO PCT/US2000/020502 patent/WO2001008677A1/en not_active Ceased
- 2000-07-28 AT AT00950797T patent/ATE448781T1/de not_active IP Right Cessation
- 2000-07-28 EP EP00950797A patent/EP1207873B1/en not_active Expired - Lifetime
- 2000-07-28 CA CA002647796A patent/CA2647796A1/en not_active Abandoned
-
2005
- 2005-02-14 AU AU2005200650A patent/AU2005200650B2/en not_active Ceased
Also Published As
| Publication number | Publication date |
|---|---|
| AU6384600A (en) | 2001-02-19 |
| JP2003505503A (ja) | 2003-02-12 |
| WO2001008677A1 (en) | 2001-02-08 |
| EP1207873B1 (en) | 2009-11-18 |
| AU778190B2 (en) | 2004-11-18 |
| ATE448781T1 (de) | 2009-12-15 |
| DE60043346D1 (de) | 2009-12-31 |
| WO2001008677A8 (en) | 2001-07-12 |
| AU2005200650B2 (en) | 2007-11-15 |
| AU2005200650A1 (en) | 2005-03-10 |
| JP4790179B2 (ja) | 2011-10-12 |
| CA2647796A1 (en) | 2001-02-08 |
| EP1207873A4 (en) | 2006-04-12 |
| EP1207873A1 (en) | 2002-05-29 |
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| Date | Code | Title | Description |
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| EEER | Examination request | ||
| FZDE | Discontinued |
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