CA2274022A1 - Processus combinatoire de preparation de bibliotheques de pyrimidines fondues - Google Patents

Processus combinatoire de preparation de bibliotheques de pyrimidines fondues Download PDF

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Publication number
CA2274022A1
CA2274022A1 CA002274022A CA2274022A CA2274022A1 CA 2274022 A1 CA2274022 A1 CA 2274022A1 CA 002274022 A CA002274022 A CA 002274022A CA 2274022 A CA2274022 A CA 2274022A CA 2274022 A1 CA2274022 A1 CA 2274022A1
Authority
CA
Canada
Prior art keywords
library
formula
compounds
compound
fused
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002274022A
Other languages
English (en)
Inventor
Gunnar Erik Junior Jagdmann
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2274022A1 publication Critical patent/CA2274022A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C07D239/72—Quinazolines; Hydrogenated quinazolines
    • C07D239/86—Quinazolines; Hydrogenated quinazolines with hetero atoms directly attached in position 4
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D239/00—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings
    • C07D239/70—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings condensed with carbocyclic rings or ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D473/00—Heterocyclic compounds containing purine ring systems
    • C07D473/26—Heterocyclic compounds containing purine ring systems with an oxygen, sulphur, or nitrogen atom directly attached in position 2 or 6, but not in both
    • C07D473/32—Nitrogen atom
    • C07D473/34—Nitrogen atom attached in position 6, e.g. adenine

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

La présente invention concerne une nouvelle échantillothèque combinatoire diversifiée de composés de pyrimidines fondues et un dispositif donnant facilement accès aux différents éléments de l'échantillothèque. Le dispositif peut s'utiliser pour des trousses d'essais et comme élément de remplacement dans des machines de dosage automatisé.
CA002274022A 1996-12-18 1997-12-15 Processus combinatoire de preparation de bibliotheques de pyrimidines fondues Abandoned CA2274022A1 (fr)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US3429596P 1996-12-18 1996-12-18
US60/034,295 1996-12-18
PCT/US1997/022839 WO1998027087A1 (fr) 1996-12-18 1997-12-15 Procede combinatoire de realisation d'echantillotheques de pyrimidines fondues

Publications (1)

Publication Number Publication Date
CA2274022A1 true CA2274022A1 (fr) 1998-06-25

Family

ID=21875516

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002274022A Abandoned CA2274022A1 (fr) 1996-12-18 1997-12-15 Processus combinatoire de preparation de bibliotheques de pyrimidines fondues

Country Status (5)

Country Link
EP (1) EP0946549A1 (fr)
JP (1) JP2001508049A (fr)
AU (1) AU5698398A (fr)
CA (1) CA2274022A1 (fr)
WO (1) WO1998027087A1 (fr)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6288234B1 (en) * 1998-06-08 2001-09-11 Advanced Medicine, Inc. Multibinding inhibitors of microsomal triglyceride transferase protein

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3948913A (en) * 1971-04-27 1976-04-06 Ciba-Geigy Corporation New 5-nitrofuryl derivatives
US4044130A (en) * 1974-07-03 1977-08-23 Ciba-Geigy Corporation Compositions for the control of microorganisms
GB1570494A (en) * 1975-11-28 1980-07-02 Ici Ltd Thienopyrimidine derivatives and their use as pesticides
US4053474A (en) * 1976-04-21 1977-10-11 E. R. Squibb & Sons, Inc. Pyrazolo[4,3-e][1,2,4]triazolo[4,3-c]pyrimidine
ZA781457B (en) * 1977-03-23 1979-03-28 Ici Ltd Pesticidal compounds,compositions and processes
US4196207A (en) * 1977-05-23 1980-04-01 Ici Australia Limited Process for controlling eradicating or preventing infestations of animals by Ixodid ticks
JPS5942387A (ja) * 1982-07-21 1984-03-08 Sankyo Co Ltd チエノピリミジン誘導体および殺虫、殺ダニ剤
GB8422916D0 (en) * 1984-09-11 1984-10-17 May & Baker Ltd Compositions of matter

Also Published As

Publication number Publication date
AU5698398A (en) 1998-07-15
JP2001508049A (ja) 2001-06-19
WO1998027087A1 (fr) 1998-06-25
EP0946549A1 (fr) 1999-10-06

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Legal Events

Date Code Title Description
FZDE Discontinued