CA2251353A1 - Dispositif pour administration transdermique de composes d'azapirone - Google Patents

Dispositif pour administration transdermique de composes d'azapirone

Info

Publication number
CA2251353A1
CA2251353A1 CA002251353A CA2251353A CA2251353A1 CA 2251353 A1 CA2251353 A1 CA 2251353A1 CA 002251353 A CA002251353 A CA 002251353A CA 2251353 A CA2251353 A CA 2251353A CA 2251353 A1 CA2251353 A1 CA 2251353A1
Authority
CA
Canada
Prior art keywords
azapirone
delivery device
transdermal delivery
transdermal
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002251353A
Other languages
English (en)
Other versions
CA2251353C (fr
Inventor
Cheryl M. Gentile
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aveva Drug Deliverty Systems Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Priority to PCT/US1996/004745 priority Critical patent/WO1997037659A1/fr
Priority to CA002251353A priority patent/CA2251353C/fr
Priority to EP96912595A priority patent/EP0942727A1/fr
Priority to AU55363/96A priority patent/AU5536396A/en
Publication of CA2251353A1 publication Critical patent/CA2251353A1/fr
Application granted granted Critical
Publication of CA2251353C publication Critical patent/CA2251353C/fr
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/70Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
    • A61K9/7023Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
    • A61K9/703Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
    • A61K9/7038Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
    • A61K9/7046Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
    • A61K9/7053Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/438The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Dermatology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
CA002251353A 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone Expired - Fee Related CA2251353C (fr)

Priority Applications (4)

Application Number Priority Date Filing Date Title
PCT/US1996/004745 WO1997037659A1 (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone
CA002251353A CA2251353C (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone
EP96912595A EP0942727A1 (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone
AU55363/96A AU5536396A (en) 1996-04-08 1996-04-08 Transdermal delivery device for azapirone compounds

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
PCT/US1996/004745 WO1997037659A1 (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone
CA002251353A CA2251353C (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone

Publications (2)

Publication Number Publication Date
CA2251353A1 true CA2251353A1 (fr) 1997-10-16
CA2251353C CA2251353C (fr) 2008-10-07

Family

ID=25680592

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002251353A Expired - Fee Related CA2251353C (fr) 1996-04-08 1996-04-08 Dispositif pour administration transdermique de composes d'azapirone

Country Status (3)

Country Link
EP (1) EP0942727A1 (fr)
CA (1) CA2251353C (fr)
WO (1) WO1997037659A1 (fr)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB0306859D0 (en) * 2003-03-25 2003-04-30 Arachnova Therapeutics Ltd Topical formulation and use of buspirone
JP6180520B2 (ja) * 2012-07-05 2017-08-16 エスケー ケミカルス カンパニー リミテッド ロチゴチンを含有した経皮吸収製剤(Transdermalcompositioncomprisingrotigotine)

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL91451A0 (en) * 1988-08-30 1990-04-29 Bristol Myers Co Pharmaceutical compositions comprising azapiron compounds and their use in the treatment of addiction
JPH06505712A (ja) * 1990-11-28 1994-06-30 サノ・コーポレーシヨン タバコ中毒の処理方法および装置
CA2159091C (fr) * 1993-03-26 2006-12-19 Richard J. Sharpe Application topique et systemique de la buspirone ou de derives de celle-ci pour le traitement de conditions pathologiques associees aux reponses immunitaires
WO1995001167A2 (fr) * 1993-06-25 1995-01-12 Alza Corporation Incorporation d'un amide poly-n-vinylique a un systeme transdermique

Also Published As

Publication number Publication date
WO1997037659A1 (fr) 1997-10-16
EP0942727A1 (fr) 1999-09-22
CA2251353C (fr) 2008-10-07

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Legal Events

Date Code Title Description
EEER Examination request
MKLA Lapsed