CA2251353A1 - Dispositif pour administration transdermique de composes d'azapirone - Google Patents
Dispositif pour administration transdermique de composes d'azapironeInfo
- Publication number
- CA2251353A1 CA2251353A1 CA002251353A CA2251353A CA2251353A1 CA 2251353 A1 CA2251353 A1 CA 2251353A1 CA 002251353 A CA002251353 A CA 002251353A CA 2251353 A CA2251353 A CA 2251353A CA 2251353 A1 CA2251353 A1 CA 2251353A1
- Authority
- CA
- Canada
- Prior art keywords
- azapirone
- delivery device
- transdermal delivery
- transdermal
- compounds
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Granted
Links
- 150000001875 compounds Chemical class 0.000 title 1
- 230000037317 transdermal delivery Effects 0.000 title 1
- 239000008280 blood Substances 0.000 abstract 1
- 210000004369 blood Anatomy 0.000 abstract 1
- 230000002035 prolonged effect Effects 0.000 abstract 1
- 238000001953 recrystallisation Methods 0.000 abstract 1
- 239000003381 stabilizer Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/70—Web, sheet or filament bases ; Films; Fibres of the matrix type containing drug
- A61K9/7023—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms
- A61K9/703—Transdermal patches and similar drug-containing composite devices, e.g. cataplasms characterised by shape or structure; Details concerning release liner or backing; Refillable patches; User-activated patches
- A61K9/7038—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer
- A61K9/7046—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds
- A61K9/7053—Transdermal patches of the drug-in-adhesive type, i.e. comprising drug in the skin-adhesive layer the adhesive comprising macromolecular compounds obtained by reactions only involving carbon to carbon unsaturated bonds, e.g. polyvinyl, polyisobutylene, polystyrene
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/438—The ring being spiro-condensed with carbocyclic or heterocyclic ring systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
- A61K31/506—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Epidemiology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Dermatology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicinal Preparation (AREA)
Priority Applications (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US1996/004745 WO1997037659A1 (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
CA002251353A CA2251353C (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
EP96912595A EP0942727A1 (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
AU55363/96A AU5536396A (en) | 1996-04-08 | 1996-04-08 | Transdermal delivery device for azapirone compounds |
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
PCT/US1996/004745 WO1997037659A1 (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
CA002251353A CA2251353C (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
Publications (2)
Publication Number | Publication Date |
---|---|
CA2251353A1 true CA2251353A1 (fr) | 1997-10-16 |
CA2251353C CA2251353C (fr) | 2008-10-07 |
Family
ID=25680592
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
CA002251353A Expired - Fee Related CA2251353C (fr) | 1996-04-08 | 1996-04-08 | Dispositif pour administration transdermique de composes d'azapirone |
Country Status (3)
Country | Link |
---|---|
EP (1) | EP0942727A1 (fr) |
CA (1) | CA2251353C (fr) |
WO (1) | WO1997037659A1 (fr) |
Families Citing this family (2)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
GB0306859D0 (en) * | 2003-03-25 | 2003-04-30 | Arachnova Therapeutics Ltd | Topical formulation and use of buspirone |
JP6180520B2 (ja) * | 2012-07-05 | 2017-08-16 | エスケー ケミカルス カンパニー リミテッド | ロチゴチンを含有した経皮吸収製剤(Transdermalcompositioncomprisingrotigotine) |
Family Cites Families (4)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
IL91451A0 (en) * | 1988-08-30 | 1990-04-29 | Bristol Myers Co | Pharmaceutical compositions comprising azapiron compounds and their use in the treatment of addiction |
JPH06505712A (ja) * | 1990-11-28 | 1994-06-30 | サノ・コーポレーシヨン | タバコ中毒の処理方法および装置 |
CA2159091C (fr) * | 1993-03-26 | 2006-12-19 | Richard J. Sharpe | Application topique et systemique de la buspirone ou de derives de celle-ci pour le traitement de conditions pathologiques associees aux reponses immunitaires |
WO1995001167A2 (fr) * | 1993-06-25 | 1995-01-12 | Alza Corporation | Incorporation d'un amide poly-n-vinylique a un systeme transdermique |
-
1996
- 1996-04-08 EP EP96912595A patent/EP0942727A1/fr not_active Withdrawn
- 1996-04-08 CA CA002251353A patent/CA2251353C/fr not_active Expired - Fee Related
- 1996-04-08 WO PCT/US1996/004745 patent/WO1997037659A1/fr not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
WO1997037659A1 (fr) | 1997-10-16 |
EP0942727A1 (fr) | 1999-09-22 |
CA2251353C (fr) | 2008-10-07 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
EEER | Examination request | ||
MKLA | Lapsed |