CA2247175A1 - Novel erythromycin derivatives, method for preparing same, and use thereof as drugs - Google Patents

Novel erythromycin derivatives, method for preparing same, and use thereof as drugs

Info

Publication number
CA2247175A1
CA2247175A1 CA002247175A CA2247175A CA2247175A1 CA 2247175 A1 CA2247175 A1 CA 2247175A1 CA 002247175 A CA002247175 A CA 002247175A CA 2247175 A CA2247175 A CA 2247175A CA 2247175 A1 CA2247175 A1 CA 2247175A1
Authority
CA
Canada
Prior art keywords
drugs
preparing same
erythromycin derivatives
novel erythromycin
radical
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002247175A
Other languages
French (fr)
Other versions
CA2247175C (en
Inventor
Constantin Agouridas
Jean-Francois Chantot
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Aventis Pharma SA
Original Assignee
Hoechst Marion Roussel
Constantin Agouridas
Jean-Francois Chantot
Aventis Pharma S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9602472A external-priority patent/FR2745290B1/en
Application filed by Hoechst Marion Roussel, Constantin Agouridas, Jean-Francois Chantot, Aventis Pharma S.A. filed Critical Hoechst Marion Roussel
Publication of CA2247175A1 publication Critical patent/CA2247175A1/en
Application granted granted Critical
Publication of CA2247175C publication Critical patent/CA2247175C/en
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

Links

Classifications

    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)

Abstract

L'invention a pour objet les composés de formule (I) dans lesquels: X représente un radical CH2 ou SO2 ou un atome d'oxygène, Y représente un radical (CH2)m-(CH=CH)n(CH2)o, avec m + n + o 8, n = 0 ou 1, Ar représente un radical aryle, W représente un atome d'hydrogène, ou le reste d'une fonction carbamate. Les composés de formule (I) présentent d'intéressantes propriétés antibiotiques.The subject of the invention is the compounds of formula (I) in which: X represents a CH2 or SO2 radical or an oxygen atom, Y represents a (CH2) m- (CH = CH) n (CH2) o radical, with m + n + o 8, n = 0 or 1, Ar represents an aryl radical, W represents a hydrogen atom, or the remainder of a carbamate function. The compounds of formula (I) have interesting antibiotic properties.

CA002247175A 1996-02-28 1997-02-27 Novel erythromycin derivatives, method for preparing same, and use thereof as drugs Expired - Lifetime CA2247175C (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR96/02472 1996-02-28
FR9602472A FR2745290B1 (en) 1996-02-28 1996-02-28 NOVEL ERYTHROMYCIN DERIVATIVES, THEIR PREPARATION PROCESS AND THEIR APPLICATION AS MEDICAMENTS
PCT/FR1997/000351 WO1997031929A1 (en) 1996-02-28 1997-02-27 Novel erythromycin derivatives, method for preparing same, and use thereof as drugs

Publications (2)

Publication Number Publication Date
CA2247175A1 true CA2247175A1 (en) 1997-09-04
CA2247175C CA2247175C (en) 2006-06-13

Family

ID=29422069

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002247175A Expired - Lifetime CA2247175C (en) 1996-02-28 1997-02-27 Novel erythromycin derivatives, method for preparing same, and use thereof as drugs

Country Status (1)

Country Link
CA (1) CA2247175C (en)

Also Published As

Publication number Publication date
CA2247175C (en) 2006-06-13

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Effective date: 20170227