CA2067540A1 - Analogue de la rapamycine comme immunosuppresseurs et antifongiques - Google Patents

Analogue de la rapamycine comme immunosuppresseurs et antifongiques

Info

Publication number
CA2067540A1
CA2067540A1 CA002067540A CA2067540A CA2067540A1 CA 2067540 A1 CA2067540 A1 CA 2067540A1 CA 002067540 A CA002067540 A CA 002067540A CA 2067540 A CA2067540 A CA 2067540A CA 2067540 A1 CA2067540 A1 CA 2067540A1
Authority
CA
Canada
Prior art keywords
choh
compound
rapamycin
deoxo
hydroxyrapamycin
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
CA002067540A
Other languages
English (en)
Inventor
Philip F. Hughes
John H. Musser
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Wyeth LLC
Original Assignee
American Home Products Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by American Home Products Corp filed Critical American Home Products Corp
Publication of CA2067540A1 publication Critical patent/CA2067540A1/fr
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains three hetero rings
    • C07D498/18—Bridged systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H19/00—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof
    • C07H19/01—Compounds containing a hetero ring sharing one ring hetero atom with a saccharide radical; Nucleosides; Mononucleotides; Anhydro-derivatives thereof sharing oxygen

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • General Health & Medical Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Molecular Biology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
CA002067540A 1991-08-07 1992-04-29 Analogue de la rapamycine comme immunosuppresseurs et antifongiques Abandoned CA2067540A1 (fr)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US741,714 1991-08-07
US07/741,714 US5138051A (en) 1991-08-07 1991-08-07 Rapamycin analogs as immunosuppressants and antifungals

Publications (1)

Publication Number Publication Date
CA2067540A1 true CA2067540A1 (fr) 1993-02-08

Family

ID=24981857

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002067540A Abandoned CA2067540A1 (fr) 1991-08-07 1992-04-29 Analogue de la rapamycine comme immunosuppresseurs et antifongiques

Country Status (2)

Country Link
US (1) US5138051A (fr)
CA (1) CA2067540A1 (fr)

Families Citing this family (99)

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US9877965B2 (en) 2007-06-25 2018-01-30 Endocyte, Inc. Vitamin receptor drug delivery conjugates for treating inflammation
BRPI0812970A2 (pt) 2007-06-25 2019-09-24 Endocyte Inc conjugados contendo espaçadores hidrofílicos
PT2365802T (pt) 2008-11-11 2017-11-14 Univ Texas Microcápsulas de rapamicina e utilização para o tratamento de cancro
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CA2795544A1 (fr) 2010-04-27 2011-11-03 Roche Glycart Ag Polytherapie d'un anticorps anti-cd20 afucosyle et d'un inhibiteur de mtor
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Also Published As

Publication number Publication date
US5138051A (en) 1992-08-11

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Legal Events

Date Code Title Description
EEER Examination request
FZDE Discontinued