CA2024071A1 - Pyrido [2, 3-b] [1,5]benzoxazepin (and thiazepin)-5 (6h)-ones and-thiones and their use in prevention or treatment of hiv infection - Google Patents

Pyrido [2, 3-b] [1,5]benzoxazepin (and thiazepin)-5 (6h)-ones and-thiones and their use in prevention or treatment of hiv infection

Info

Publication number
CA2024071A1
CA2024071A1 CA002024071A CA2024071A CA2024071A1 CA 2024071 A1 CA2024071 A1 CA 2024071A1 CA 002024071 A CA002024071 A CA 002024071A CA 2024071 A CA2024071 A CA 2024071A CA 2024071 A1 CA2024071 A1 CA 2024071A1
Authority
CA
Canada
Prior art keywords
thiazepin
benzoxazepin
thiones
pyrido
ones
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
CA002024071A
Other languages
French (fr)
Other versions
CA2024071C (en
Inventor
Karl D. Hargrave
Gunther Schmidt (Deceased)
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Boehringer Ingelheim Pharma GmbH and Co KG
Boehringer Ingelheim Pharmaceuticals Inc
Original Assignee
Individual
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Individual filed Critical Individual
Publication of CA2024071A1 publication Critical patent/CA2024071A1/en
Application granted granted Critical
Publication of CA2024071C publication Critical patent/CA2024071C/en
Anticipated expiration legal-status Critical
Expired - Fee Related legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Disclosed are pyrido[2,3-b][1,5]benzoxazepin (and thiazepin)-5(6H)-ones and -thiones of the formula I. These are useful in the prevention or treatment of AIDS.

(See formula 1)
CA002024071A 1989-08-29 1990-08-27 Pyrido [2, 3-b] [1,5]benzoxazepin (and thiazepin)-5 (6h)-ones and-thiones and their use in prevention or treatment of hiv infection Expired - Fee Related CA2024071C (en)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US40025389A 1989-08-29 1989-08-29
US400,253 1989-08-29
US53929490A 1990-06-15 1990-06-15
US539,294 1990-06-15

Publications (2)

Publication Number Publication Date
CA2024071A1 true CA2024071A1 (en) 1991-03-01
CA2024071C CA2024071C (en) 2002-06-04

Family

ID=27016965

Family Applications (1)

Application Number Title Priority Date Filing Date
CA002024071A Expired - Fee Related CA2024071C (en) 1989-08-29 1990-08-27 Pyrido [2, 3-b] [1,5]benzoxazepin (and thiazepin)-5 (6h)-ones and-thiones and their use in prevention or treatment of hiv infection

Country Status (8)

Country Link
AP (1) AP190A (en)
AU (1) AU624264B2 (en)
CA (1) CA2024071C (en)
FI (1) FI93362C (en)
HU (1) HU206723B (en)
NO (1) NO177786C (en)
OA (1) OA09307A (en)
PT (1) PT95113B (en)

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CA554134A (en) * 1958-03-11 Hoffmann Karl Thia-aza-cycloheptadiene compounds and process for their manufacture
CA799979A (en) * 1968-11-26 Dr. Karl Thomae Gesellschaft Mit Beschrankter Haftung 5,6-dihydro-6-oxo-pyrido(2,3-b) (1,4)-benzoxazepines
CA802216A (en) * 1968-12-24 Hoffmann Charles Heterocyclic compounds
GB1587128A (en) * 1977-04-07 1981-04-01 Hexachimie Benzothiazepine derivatives
US4940704A (en) * 1989-08-16 1990-07-10 Hoechst-Roussel Pharmaceutical Inc. Pyrido[3,4-b][1,4]benzoxazepines

Also Published As

Publication number Publication date
CA2024071C (en) 2002-06-04
NO177786C (en) 1995-11-22
AP190A (en) 1992-05-04
NO903778L (en) 1991-03-01
AP9000203A0 (en) 1990-10-31
AU624264B2 (en) 1992-06-04
FI93362B (en) 1994-12-15
FI93362C (en) 1995-03-27
NO177786B (en) 1995-08-14
PT95113A (en) 1991-05-22
AU6191790A (en) 1991-03-07
HUT57777A (en) 1991-12-30
HU206723B (en) 1992-12-28
HU905510D0 (en) 1991-02-28
OA09307A (en) 1992-09-15
PT95113B (en) 1997-04-30
FI904244A0 (en) 1990-08-28
NO903778D0 (en) 1990-08-28

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Legal Events

Date Code Title Description
EEER Examination request
MKLA Lapsed