CA1051879A - Synthesis of elymoclavine and derivatives - Google Patents

Synthesis of elymoclavine and derivatives

Info

Publication number
CA1051879A
CA1051879A CA228,474A CA228474A CA1051879A CA 1051879 A CA1051879 A CA 1051879A CA 228474 A CA228474 A CA 228474A CA 1051879 A CA1051879 A CA 1051879A
Authority
CA
Canada
Prior art keywords
methyl
ergolene
methoxy
formula
formyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA228,474A
Other languages
English (en)
French (fr)
Inventor
Edmund C. Kornfeld
Nicholas J. Bach
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Eli Lilly and Co
Original Assignee
Eli Lilly and Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from US494149A external-priority patent/US3923812A/en
Priority claimed from US494147A external-priority patent/US3929796A/en
Application filed by Eli Lilly and Co filed Critical Eli Lilly and Co
Application granted granted Critical
Publication of CA1051879A publication Critical patent/CA1051879A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/04—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached in position 8
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/02—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hydrocarbon or substituted hydrocarbon radicals, attached in position 8
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D457/00—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid
    • C07D457/10—Heterocyclic compounds containing indolo [4, 3-f, g] quinoline ring systems, e.g. derivatives of ergoline, of the formula:, e.g. lysergic acid with hetero atoms directly attached in position 8

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
CA228,474A 1974-08-02 1975-06-04 Synthesis of elymoclavine and derivatives Expired CA1051879A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US494149A US3923812A (en) 1974-08-02 1974-08-02 Synthesis of elymoclavine
US494147A US3929796A (en) 1974-08-02 1974-08-02 Synthesis of penniclavine and elymoclavine

Publications (1)

Publication Number Publication Date
CA1051879A true CA1051879A (en) 1979-04-03

Family

ID=27051314

Family Applications (2)

Application Number Title Priority Date Filing Date
CA228,474A Expired CA1051879A (en) 1974-08-02 1975-06-04 Synthesis of elymoclavine and derivatives
CA228,512A Expired CA1042423A (en) 1974-08-02 1975-06-04 Synthesis of penniclavine and derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
CA228,512A Expired CA1042423A (en) 1974-08-02 1975-06-04 Synthesis of penniclavine and derivatives

Country Status (8)

Country Link
CA (2) CA1051879A ( )
CH (5) CH613967A5 ( )
DE (1) DE2534512A1 ( )
FR (1) FR2284327A1 ( )
GB (2) GB1521311A ( )
IE (1) IE41475B1 ( )
IL (2) IL47485A ( )
NL (2) NL7508939A ( )

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL7102982A ( ) * 1970-03-20 1971-09-22 Farmaceutici Italia

Also Published As

Publication number Publication date
CH614206A5 (en) 1979-11-15
IL47485A0 (en) 1976-03-31
NL7508938A (nl) 1976-02-04
IL53215A0 (en) 1977-12-30
IL47485A (en) 1978-10-31
CH612966A5 (en) 1979-08-31
IE41475L (en) 1976-02-02
CH613704A5 (en) 1979-10-15
FR2284327B1 ( ) 1978-11-10
IE41475B1 (en) 1980-01-16
FR2284327A1 (fr) 1976-04-09
CA1042423A (en) 1978-11-14
DE2534512A1 (de) 1976-02-12
NL7508939A (nl) 1976-02-04
CH613703A5 (en) 1979-10-15
GB1521311A (en) 1978-08-16
CH613967A5 (en) 1979-10-31
GB1521312A (en) 1978-08-16

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