BRPI0908953A2 - composto, processo de preparo e composição farmacêutica de derivados cíclicos e lineares de guanidina. - Google Patents
composto, processo de preparo e composição farmacêutica de derivados cíclicos e lineares de guanidina.Info
- Publication number
- BRPI0908953A2 BRPI0908953A2 BRPI0908953A BRPI0908953A BRPI0908953A2 BR PI0908953 A2 BRPI0908953 A2 BR PI0908953A2 BR PI0908953 A BRPI0908953 A BR PI0908953A BR PI0908953 A BRPI0908953 A BR PI0908953A BR PI0908953 A2 BRPI0908953 A2 BR PI0908953A2
- Authority
- BR
- Brazil
- Prior art keywords
- cyclic
- compound
- pharmaceutical composition
- preparation process
- guanidine derivatives
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D255/00—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00
- C07D255/02—Heterocyclic compounds containing rings having three nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D249/00 - C07D253/00 not condensed with other rings
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C279/00—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups
- C07C279/04—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton
- C07C279/12—Derivatives of guanidine, i.e. compounds containing the group, the singly-bound nitrogen atoms not being part of nitro or nitroso groups having nitrogen atoms of guanidine groups bound to acyclic carbon atoms of a carbon skeleton being further substituted by nitrogen atoms not being part of nitro or nitroso groups
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D259/00—Heterocyclic compounds containing rings having more than four nitrogen atoms as the only ring hetero atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C2601/00—Systems containing only non-condensed rings
- C07C2601/02—Systems containing only non-condensed rings with a three-membered ring
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US3616508P | 2008-03-13 | 2008-03-13 | |
| PCT/IB2009/051032 WO2009113033A2 (en) | 2008-03-13 | 2009-03-12 | Linear and cyclic guanidine derivatives, method of preparation and uses thereof |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| BRPI0908953A2 true BRPI0908953A2 (pt) | 2016-06-07 |
Family
ID=40622063
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| BRPI0908953A BRPI0908953A2 (pt) | 2008-03-13 | 2009-03-12 | composto, processo de preparo e composição farmacêutica de derivados cíclicos e lineares de guanidina. |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8685953B2 (pt) |
| EP (1) | EP2274290B1 (pt) |
| JP (1) | JP5733988B2 (pt) |
| CN (1) | CN101977901B (pt) |
| AU (1) | AU2009223204B2 (pt) |
| BR (1) | BRPI0908953A2 (pt) |
| DK (1) | DK2274290T3 (pt) |
| EA (1) | EA018926B1 (pt) |
| ES (1) | ES2396288T3 (pt) |
| MX (1) | MX2010010017A (pt) |
| PL (1) | PL2274290T3 (pt) |
| PT (1) | PT2274290E (pt) |
| WO (1) | WO2009113033A2 (pt) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| CA2915767A1 (en) | 2013-06-18 | 2014-12-24 | Cygnet Biosciences B.V. | New macrocyclic amidinourea derivatives, methods of preparation and uses thereof as chitinase inhibitors |
| JP6378179B2 (ja) | 2013-07-03 | 2018-08-22 | 株式会社新日本科学 | 新規化合物，有機カチオントランスポーター３の検出剤及び活性阻害剤 |
| WO2016055644A1 (en) | 2014-10-10 | 2016-04-14 | Lead Discovery Siena S.R.L. | Linear guanidine derivatives, methods of preparation and uses thereof |
| EP3854789A1 (en) * | 2020-01-22 | 2021-07-28 | Cygnet Biosciences B.V. | Macrocyclic compounds useful as chitinase inhibitors |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB1114155A (en) | 1964-08-24 | 1968-05-15 | Evans Medical Ltd | Guanidino derivatives |
| US3988370A (en) | 1970-10-08 | 1976-10-26 | Sterling Drug Inc. | Amidinoureas |
-
2009
- 2009-03-12 ES ES09719584T patent/ES2396288T3/es active Active
- 2009-03-12 MX MX2010010017A patent/MX2010010017A/es active IP Right Grant
- 2009-03-12 EA EA201071072A patent/EA018926B1/ru not_active IP Right Cessation
- 2009-03-12 PL PL09719584T patent/PL2274290T3/pl unknown
- 2009-03-12 CN CN200980108874.6A patent/CN101977901B/zh not_active Expired - Fee Related
- 2009-03-12 DK DK09719584.6T patent/DK2274290T3/da active
- 2009-03-12 US US12/922,232 patent/US8685953B2/en not_active Expired - Fee Related
- 2009-03-12 JP JP2010550321A patent/JP5733988B2/ja not_active Expired - Fee Related
- 2009-03-12 AU AU2009223204A patent/AU2009223204B2/en not_active Ceased
- 2009-03-12 PT PT97195846T patent/PT2274290E/pt unknown
- 2009-03-12 BR BRPI0908953A patent/BRPI0908953A2/pt not_active IP Right Cessation
- 2009-03-12 WO PCT/IB2009/051032 patent/WO2009113033A2/en active Application Filing
- 2009-03-12 EP EP09719584A patent/EP2274290B1/en not_active Not-in-force
Also Published As
| Publication number | Publication date |
|---|---|
| PT2274290E (pt) | 2013-01-14 |
| US20110039854A1 (en) | 2011-02-17 |
| PL2274290T3 (pl) | 2013-03-29 |
| WO2009113033A2 (en) | 2009-09-17 |
| DK2274290T3 (da) | 2013-01-14 |
| EA201071072A1 (ru) | 2011-04-29 |
| CN101977901A (zh) | 2011-02-16 |
| ES2396288T3 (es) | 2013-02-20 |
| AU2009223204B2 (en) | 2014-07-24 |
| JP5733988B2 (ja) | 2015-06-10 |
| EP2274290B1 (en) | 2012-09-26 |
| WO2009113033A3 (en) | 2009-12-30 |
| CN101977901B (zh) | 2015-04-01 |
| MX2010010017A (es) | 2010-10-07 |
| EP2274290A2 (en) | 2011-01-19 |
| JP2011513477A (ja) | 2011-04-28 |
| US8685953B2 (en) | 2014-04-01 |
| EA018926B1 (ru) | 2013-11-29 |
| AU2009223204A1 (en) | 2009-09-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE AS 6A E 7A ANUIDADES. |
|
| B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2384 DE 13-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |