BRPI0618452A2 - piridopirazinas e seu uso como moduladores de cinases - Google Patents
piridopirazinas e seu uso como moduladores de cinases Download PDFInfo
- Publication number
- BRPI0618452A2 BRPI0618452A2 BRPI0618452-9A BRPI0618452A BRPI0618452A2 BR PI0618452 A2 BRPI0618452 A2 BR PI0618452A2 BR PI0618452 A BRPI0618452 A BR PI0618452A BR PI0618452 A2 BRPI0618452 A2 BR PI0618452A2
- Authority
- BR
- Brazil
- Prior art keywords
- pyridopyrazines
- kinase modulators
- malignant
- medicament
- modulators
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
- C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
- C07D471/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
Abstract
PIRIDOPIRAZINAS E SEU USO COMO MODULADORES DE CINASES. A presente invenção refere-se a novos derivados de pirido[2,3- b]pirazina da fórmula geral (I), sua produção e uso como medicamento, especialmente para o tratamento de doenças malignas e outras, à base de proliferações de células patológicas.
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US73569805P | 2005-11-11 | 2005-11-11 | |
EP05024693A EP1785423A1 (de) | 2005-11-11 | 2005-11-11 | Neue Pyridopyrazine und deren Verwendung als Modulatoren von Kinasen |
US84976106P | 2006-10-06 | 2006-10-06 | |
PCT/EP2006/068322 WO2007054556A1 (de) | 2005-11-11 | 2006-11-10 | Neue pyridopyrazine und deren verwendung als modulatoren von kinasen |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0618452A2 true BRPI0618452A2 (pt) | 2011-08-30 |
Family
ID=36149056
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0618452-9A BRPI0618452A2 (pt) | 2005-11-11 | 2006-11-10 | piridopirazinas e seu uso como moduladores de cinases |
Country Status (4)
Country | Link |
---|---|
EP (1) | EP1785423A1 (pt) |
BR (1) | BRPI0618452A2 (pt) |
NZ (1) | NZ595658A (pt) |
TW (1) | TWI392675B (pt) |
Families Citing this family (1)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
EP2508184A1 (en) * | 2011-04-06 | 2012-10-10 | Æterna Zentaris GmbH | Pyridopyrazine derivatives and their use |
Family Cites Families (3)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE10323345A1 (de) * | 2003-05-23 | 2004-12-16 | Zentaris Gmbh | Neue Pyridopyrazine und deren Verwendung als Kinase-Inhibitoren |
ATE411992T1 (de) * | 2003-05-23 | 2008-11-15 | Fterna Zentaris Gmbh | Neue pyridopyrazine und deren verwendung als modulatoren von kinasen |
WO2005007099A2 (en) * | 2003-07-10 | 2005-01-27 | Imclone Systems Incorporated | Pkb inhibitors as anti-tumor agents |
-
2005
- 2005-11-11 EP EP05024693A patent/EP1785423A1/de not_active Withdrawn
-
2006
- 2006-11-10 TW TW095141721A patent/TWI392675B/zh not_active IP Right Cessation
- 2006-11-10 NZ NZ595658A patent/NZ595658A/xx unknown
- 2006-11-10 BR BRPI0618452-9A patent/BRPI0618452A2/pt not_active IP Right Cessation
Also Published As
Publication number | Publication date |
---|---|
TWI392675B (zh) | 2013-04-11 |
EP1785423A1 (de) | 2007-05-16 |
TW200736254A (en) | 2007-10-01 |
NZ595658A (en) | 2013-03-28 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTE A 10A ANUIDADE. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2386 DE 27-09-2016 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |