BRPI0607765A2 - pirazolopirimidinas - Google Patents
pirazolopirimidinasInfo
- Publication number
- BRPI0607765A2 BRPI0607765A2 BRPI0607765-0A BRPI0607765A BRPI0607765A2 BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2 BR PI0607765 A BRPI0607765 A BR PI0607765A BR PI0607765 A2 BRPI0607765 A2 BR PI0607765A2
- Authority
- BR
- Brazil
- Prior art keywords
- pyrazolopyrimidines
- pirazolopyrimidines
- formula
- preparation
- description
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- A—HUMAN NECESSITIES
- A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
- A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
- A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
- A01N43/90—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having two or more relevant hetero rings, condensed among themselves or with a common carbocyclic ring system
Landscapes
- Life Sciences & Earth Sciences (AREA)
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Plant Pathology (AREA)
- Engineering & Computer Science (AREA)
- Dentistry (AREA)
- General Health & Medical Sciences (AREA)
- Wood Science & Technology (AREA)
- Zoology (AREA)
- Environmental Sciences (AREA)
- Pest Control & Pesticides (AREA)
- Agronomy & Crop Science (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
Abstract
PIRAZOLOPIRIMIDINAS. A presente invenção refere-se a pirazolopirimidinas da fórmula (I) na qual R^ 1^, R^ 2^, R^ 3^, R^ 4^, R^ 5^ e X têm os significados indicados na descrição, processo para sua preparação e seu emprego para o controle de microor- ganismos indesejados.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE102005007534A DE102005007534A1 (de) | 2005-02-17 | 2005-02-17 | Pyrazolopyrimidine |
PCT/EP2006/001064 WO2006087120A2 (de) | 2005-02-17 | 2006-02-07 | Pyrazolopyrimidine |
Publications (1)
Publication Number | Publication Date |
---|---|
BRPI0607765A2 true BRPI0607765A2 (pt) | 2009-10-06 |
Family
ID=36793966
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI0607765-0A BRPI0607765A2 (pt) | 2005-02-17 | 2006-02-07 | pirazolopirimidinas |
Country Status (16)
Country | Link |
---|---|
US (1) | US7781439B2 (pt) |
EP (1) | EP1853607A2 (pt) |
JP (1) | JP2008530155A (pt) |
KR (1) | KR20070103473A (pt) |
CN (1) | CN101120000B (pt) |
AR (1) | AR052913A1 (pt) |
AU (1) | AU2006215858A1 (pt) |
BR (1) | BRPI0607765A2 (pt) |
CA (1) | CA2597833A1 (pt) |
DE (1) | DE102005007534A1 (pt) |
EA (1) | EA200701707A1 (pt) |
IL (1) | IL185092A0 (pt) |
MX (1) | MX2007010045A (pt) |
TW (1) | TW200640926A (pt) |
WO (1) | WO2006087120A2 (pt) |
ZA (1) | ZA200706734B (pt) |
Families Citing this family (23)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102006039255A1 (de) * | 2006-08-17 | 2008-02-21 | Bayer Cropscience Ag | Insektizide heterocyclische Carbonsäurederivate |
EP2014661A1 (de) * | 2007-06-13 | 2009-01-14 | Bayer CropScience AG | Heterocyclisch substituierte Heterocyclyl-carbonsäurederivate |
GB0712653D0 (en) | 2007-06-28 | 2007-08-08 | Syngenta Ltd | Novel herbicides |
GB0717082D0 (en) | 2007-09-03 | 2007-10-10 | Syngenta Ltd | Novel herbicides |
WO2010045615A2 (en) | 2008-10-16 | 2010-04-22 | Cenomed Biosciences, Llc | Treatment of organophosphate exposure with ocinaplon |
ES2681218T3 (es) | 2010-12-08 | 2018-09-12 | The U.S.A. As Represented By The Secretary, Department Of Health And Human Services | Pirazolopirimidinas sustituidas como activadoras de la glucocerebrosidasa |
EP2723746A1 (en) | 2011-06-22 | 2014-04-30 | Vertex Pharmaceuticals Inc. | Compounds useful as inhibitors of atr kinase |
ES2946360T3 (es) | 2012-12-07 | 2023-07-17 | Vertex Pharma | Pirazolo[1,5-a]pirimidinas útiles como inhibidores de ATR quinasa para el tratamiento de enfermedades de cáncer |
WO2014143240A1 (en) | 2013-03-15 | 2014-09-18 | Vertex Pharmaceuticals Incorporated | Fused pyrazolopyrimidine derivatives useful as inhibitors of atr kinase |
US8969360B2 (en) | 2013-03-15 | 2015-03-03 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of ATR kinase |
WO2014143241A1 (en) | 2013-03-15 | 2014-09-18 | Vertex Pharmaceuticals Incorporated | Compounds useful as inhibitors of atr kinase |
RU2687276C2 (ru) | 2013-12-06 | 2019-05-13 | Вертекс Фармасьютикалз Инкорпорейтед | Соединения, пригодные для использования в качестве ингибиторов atr киназы |
LT3152212T (lt) | 2014-06-05 | 2020-05-11 | Vertex Pharmaceuticals Inc. | Radioaktyviai žymėti 2-amino-6-fluor-n-[5-fluor-piridin-il]- pirazolo[1,5-a]pirimidin-3-karboksamido junginio dariniai, naudingi kaip atr kinazės inhibitoriai, minėto junginio gamybos būdas ir jo skirtingos kietos formos |
SG11201610500WA (en) | 2014-06-17 | 2017-01-27 | Vertex Pharma | Method for treating cancer using a combination of chk1 and atr inhibitors |
EP3215511B1 (en) | 2014-11-06 | 2024-04-17 | Bial-R&D Investments, S.A. | Substituted pyrazolo(1,5-a)pyrimidines and their use in the treatment of medical disorders |
CA3000684A1 (en) | 2015-09-30 | 2017-04-06 | Vertex Pharmaceuticals Incorporated | Method for treating cancer using a combination of dna damaging agents and atr inhibitors |
EP3440080A4 (en) * | 2016-04-06 | 2020-01-22 | Lysosomal Therapeutics Inc. | PYRAZOLO [1,5-A] PYRIMIDINYL CARBOXAMIDE COMPOUNDS AND THEIR USE IN THE TREATMENT OF MEDICAL DISORDERS |
MX2018012208A (es) | 2016-04-06 | 2019-03-28 | Lysosomal Therapeutics Inc | Compuestos a base de imidazo [1,5-a] pirimidinil carboxamida y su uso en el tratamiento de trastornos médicos. |
US11124516B2 (en) | 2016-04-06 | 2021-09-21 | BIAL-BioTech Investments, Inc. | Pyrrolo[1,2-A]pyrimidinyl carboxamide compounds and their use in the treatment of medical disorders |
US11168087B2 (en) | 2016-05-05 | 2021-11-09 | Bial—R&D Investments, S.A. | Substituted imidazo[1,2-b]pyridazines, substituted imidazo[1,5-b]pyridazines, related compounds, and their use in the treatment of medical disorders |
BR112020001714A2 (pt) * | 2017-07-28 | 2020-07-21 | Nimbus Lakshmi, Inc. | inibidores de tyk2 e usos dos mesmos |
CN112996790B (zh) | 2018-10-30 | 2023-11-03 | 克洛诺斯生物公司 | 用于调节cdk9活性的化合物、组合物和方法 |
CN113287620B (zh) * | 2021-06-18 | 2021-11-19 | 浙江大学 | 1H-吡唑并[3,4-d]嘧啶类化合物在制备禾谷镰刀菌杀菌剂中的应用 |
Family Cites Families (21)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
US2444606A (en) * | 1945-12-15 | 1948-07-06 | Gen Aniline & Film Corp | Stabilizers for photographic emulsions |
US3515715A (en) * | 1967-01-23 | 1970-06-02 | Eastman Kodak Co | Quaternized pyrazolylazo dyes |
US3634391A (en) * | 1969-07-25 | 1972-01-11 | Eastman Kodak Co | Pyrazolyl-azo-indole dyestuffs |
US4838925A (en) * | 1986-04-25 | 1989-06-13 | E. I. Du Pont De Nemours And Company | Heterocyclic acyl sulfonamides |
DE3825043A1 (de) | 1988-07-20 | 1990-02-15 | Schering Ag | 3-methylsulfonyl-pyrazolo(1,5-a)pyrimidin-sulfonsaeureamide, verfahren zu ihrer herstellung und ihre verwendung als mittel mit herbizider, pflanzenwuchsregulierender und fungizider wirkung |
US6156925A (en) * | 1998-09-25 | 2000-12-05 | American Cyanamid Company | Process for the preparation of halogenated phenylmaloates |
IL131912A (en) | 1998-09-25 | 2005-12-18 | American Cyanamid Co | Process for preparing halogenated phenylmalonates |
ATE282040T1 (de) | 2000-12-11 | 2004-11-15 | Basf Ag | 6-phenyl-pyrazolpyrimidine |
DE50209786D1 (de) | 2001-07-26 | 2007-05-03 | Basf Ag | 7-aminotriazolopyrimidine zur bekämpfung von schadpilzen |
NZ518658A (en) * | 2002-04-30 | 2004-10-29 | Lionel Evans | Method of water treatment |
DE10223917A1 (de) | 2002-05-29 | 2003-12-11 | Bayer Cropscience Ag | Pyrazolopyrimidine |
FR2841982B1 (fr) | 2002-07-03 | 2005-03-25 | Inst Francais Du Petrole | Capteur de pression a fibre optique compense en temperature |
CA2492379A1 (en) | 2002-07-17 | 2004-01-22 | Warner-Lambert Company Llc | Combination of an allosteric inhibitor of matrix metalloproteinase-13 with celecoxib or valdecoxib |
CA2516824A1 (en) * | 2003-02-28 | 2004-09-10 | Teijin Pharma Limited | Pyrazolo[1,5-a]pyrimidine derivatives |
BRPI0410610A (pt) | 2003-06-03 | 2006-07-04 | Basf Ag | compostos, processos para a produção dos mesmos e para o combate de fungos nocivos fitopatogênicos, produtos intermediários, e, agente adequado para o combate de fungos nocivos |
AU2004251845A1 (en) * | 2003-06-27 | 2005-01-06 | Bayer Cropscience Aktiengesellschaft | Pyrazolopyrimidines |
DE10357565A1 (de) * | 2003-12-10 | 2005-07-07 | Bayer Cropscience Ag | Pyrazolopyrimidine |
DE10357567A1 (de) * | 2003-12-10 | 2005-07-07 | Bayer Cropscience Ag | Pyrazolopyrimidine |
DE10357569A1 (de) * | 2003-12-10 | 2005-07-07 | Bayer Cropscience Ag | Pyrazolopyrimidine |
DE10357568A1 (de) | 2003-12-10 | 2005-07-07 | Bayer Cropscience Ag | Pyrazolopyrimidine |
DE102004008807A1 (de) | 2004-02-20 | 2005-09-08 | Bayer Cropscience Ag | Pyrazolopyrimidine |
-
2005
- 2005-02-17 DE DE102005007534A patent/DE102005007534A1/de not_active Withdrawn
-
2006
- 2006-02-07 EP EP06706711A patent/EP1853607A2/de not_active Ceased
- 2006-02-07 CA CA002597833A patent/CA2597833A1/en not_active Abandoned
- 2006-02-07 BR BRPI0607765-0A patent/BRPI0607765A2/pt not_active IP Right Cessation
- 2006-02-07 JP JP2007555499A patent/JP2008530155A/ja not_active Withdrawn
- 2006-02-07 WO PCT/EP2006/001064 patent/WO2006087120A2/de active Application Filing
- 2006-02-07 KR KR1020077019730A patent/KR20070103473A/ko not_active Application Discontinuation
- 2006-02-07 US US11/816,253 patent/US7781439B2/en not_active Expired - Fee Related
- 2006-02-07 MX MX2007010045A patent/MX2007010045A/es not_active Application Discontinuation
- 2006-02-07 CN CN2006800052137A patent/CN101120000B/zh not_active Expired - Fee Related
- 2006-02-07 EA EA200701707A patent/EA200701707A1/ru unknown
- 2006-02-07 AU AU2006215858A patent/AU2006215858A1/en not_active Abandoned
- 2006-02-16 TW TW095105170A patent/TW200640926A/zh unknown
- 2006-02-17 AR ARP060100581A patent/AR052913A1/es not_active Application Discontinuation
-
2007
- 2007-08-07 IL IL185092A patent/IL185092A0/en unknown
- 2007-08-14 ZA ZA200706734A patent/ZA200706734B/xx unknown
Also Published As
Publication number | Publication date |
---|---|
CA2597833A1 (en) | 2006-08-24 |
AU2006215858A1 (en) | 2006-08-24 |
EA200701707A1 (ru) | 2008-02-28 |
US7781439B2 (en) | 2010-08-24 |
AR052913A1 (es) | 2007-04-11 |
WO2006087120A8 (de) | 2007-08-30 |
MX2007010045A (es) | 2007-10-02 |
US20080287463A1 (en) | 2008-11-20 |
EP1853607A2 (de) | 2007-11-14 |
KR20070103473A (ko) | 2007-10-23 |
CN101120000B (zh) | 2011-05-18 |
ZA200706734B (en) | 2009-01-28 |
DE102005007534A1 (de) | 2006-08-31 |
WO2006087120A2 (de) | 2006-08-24 |
CN101120000A (zh) | 2008-02-06 |
IL185092A0 (en) | 2007-12-03 |
WO2006087120A3 (de) | 2006-12-14 |
TW200640926A (en) | 2006-12-01 |
JP2008530155A (ja) | 2008-08-07 |
Similar Documents
Publication | Publication Date | Title |
---|---|---|
BRPI0607765A2 (pt) | pirazolopirimidinas | |
BRPI0507894A (pt) | pirazolopirimidinas | |
BRPI0510410A (pt) | compostos orgánicos | |
BRPI0514361A (pt) | processo para a produção de dihidropteridinonas | |
BRPI0510412A (pt) | compostos orgánicos | |
BRPI0512335A (pt) | compostos, processo para a sua manufatura, composições farmacêuticas que os compreendem, método para o tratamento e/ou prevenção de enfermidades e sua utilização | |
BRPI0411713B8 (pt) | compostos, processo para a sua manufatura, composições farmacêuticas que compreendem os mesmos, método para tratamento e/ou profilaxia de enfermidades que estão associadas com dpp-iv e sua utilização | |
BRPI0407145A (pt) | Pirazolilcarboxanilidas para combater microorganismos indesejados | |
BRPI0514678A (pt) | bifeniltiazolcarboxamida | |
BRPI0410494A (pt) | iodopirazolilcarboxanilidas | |
BR0312379A (pt) | Produtos de poliadição contendo grupos uretodiona | |
BRPI0514439A (pt) | bifeniltiazolcarboxamidas | |
BRPI0806400A8 (pt) | composto, composição farmacêutica, produtos, usos de pelo menos um composto, método in vitro, kit, ligantes e processo de preparação de um composto | |
BRPI0511500A (pt) | processo para a preparação de um composto de amÈnio quaternário, uso de uma solução de hidróxido de tetrametilamÈnio de alta pureza, e solução aquosa de hidróxido de tetrametilamÈnio de alta pureza | |
BRPI0712889A8 (pt) | composto, processo para a preparação de um composto, composto intermediário, e, composição farmacêutica. | |
BRPI0515813A (pt) | 2 - alquil - cicloalqu( en ) il- carboxamidas | |
BRPI0519578A2 (pt) | pirimidinas substituÍdas | |
BRPI0415203A (pt) | pentanóis reestruturados, um processo para sua produção e seu uso como agentes antiinflamatórios | |
BRPI0512580A (pt) | derivados de n-fenilpirazol como pesticidas | |
BRPI0406596A (pt) | Métodos para tratar a dor articular e melhorar o sono utilizando um agonista/antagonista de estrogênio | |
BR0309568A (pt) | Triazolopirimidinas | |
BRPI0411738A (pt) | compostos orgánicos | |
BRPI0413139A (pt) | processo para a preparação de l-treonina | |
BRPI0415454A (pt) | 1,3-dimetilbutilcarboxanilidas para controle de microorganismos indesejáveis | |
BRPI0416571A (pt) | nicotinoilcarbamatos substituìdos como pesticidas |
Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application dismissed because of non-payment of annual fees [chapter 8.6 patent gazette] |
Free format text: REFERENTE A 6A ANUIDADE. |
|
B08K | Patent lapsed as no evidence of payment of the annual fee has been furnished to inpi [chapter 8.11 patent gazette] |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 2161 DE 05/06/2012. |