BR9908861A - Cyclooctadepsipeptides and their use to combat endoparasites - Google Patents
Cyclooctadepsipeptides and their use to combat endoparasitesInfo
- Publication number
- BR9908861A BR9908861A BR9908861-4A BR9908861A BR9908861A BR 9908861 A BR9908861 A BR 9908861A BR 9908861 A BR9908861 A BR 9908861A BR 9908861 A BR9908861 A BR 9908861A
- Authority
- BR
- Brazil
- Prior art keywords
- cyclooctadepsipeptides
- endoparasites
- preparation
- combat
- combat endoparasites
- Prior art date
Links
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D273/00—Heterocyclic compounds containing rings having nitrogen and oxygen atoms as the only ring hetero atoms, not provided for by groups C07D261/00 - C07D271/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/10—Anthelmintics
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Life Sciences & Earth Sciences (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Pharmacology & Pharmacy (AREA)
- Tropical Medicine & Parasitology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Peptides Or Proteins (AREA)
- Hydrogenated Pyridines (AREA)
Abstract
Patente de Invenção: <B>"CICLOOCTADEPSIPEPTìDEOS E SEU USO PARA O COMBATE DE ENDOPARASITAS"<D>. A invenção refere-se a novos ciclooctadepsipeptídeos da fórmula (I), em que R¹ representa ciano, heterociclila ligada com C-C ou alquenila, alquinila ou arila eventualmente substituídas e R² representa hidrogênio ou representa o mesmo radical que R¹, processo para a sua preparação, produtos intermediários para a sua preparação e seu uso para o combate de endoparasitas e agentes contendo estas substâncias ativas.Invention Patent: <B> "CYCLEOCTADEPSIPEPTIDES AND THEIR USE FOR COMBATING ENDOPARASITES" <D>. The invention relates to new cyclooctadepsipeptides of formula (I), in which R¹ represents cyano, heterocyclyl linked with CC or alkenyl, alkynyl or aryl possibly substituted and R² represents hydrogen or represents the same radical as R¹, process for its preparation, intermediate products for their preparation and their use to fight endoparasites and agents containing these active substances.
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
DE19811559A DE19811559A1 (en) | 1998-03-17 | 1998-03-17 | New substituted derivatives of cyclooctadepsipeptide PF1022, useful as parasiticides, especially anthelmintics |
PCT/EP1999/001407 WO1999047506A1 (en) | 1998-03-17 | 1999-03-04 | Cyclooctadepsipeptides and their use for combating endoparasites |
Publications (1)
Publication Number | Publication Date |
---|---|
BR9908861A true BR9908861A (en) | 2000-11-21 |
Family
ID=7861200
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BR9908861-4A BR9908861A (en) | 1998-03-17 | 1999-03-04 | Cyclooctadepsipeptides and their use to combat endoparasites |
Country Status (10)
Country | Link |
---|---|
EP (1) | EP1064272A1 (en) |
JP (1) | JP2002506857A (en) |
KR (1) | KR20010041450A (en) |
CN (1) | CN1293664A (en) |
AU (1) | AU3143899A (en) |
BR (1) | BR9908861A (en) |
CA (1) | CA2323628A1 (en) |
DE (1) | DE19811559A1 (en) |
PL (1) | PL342948A1 (en) |
WO (1) | WO1999047506A1 (en) |
Families Citing this family (8)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DE102008030764A1 (en) | 2008-06-28 | 2009-12-31 | Bayer Animal Health Gmbh | Combination of amidine derivatives with cyclic depsipeptides |
DE102009012423A1 (en) | 2009-03-10 | 2010-09-16 | Bayer Animal Health Gmbh | Preparation based on oil |
WO2012028556A1 (en) | 2010-08-31 | 2012-03-08 | Bayer Animal Health Gmbh | Macrocyclic lactones and their use and their combinations with other active substances |
DE102010064245A1 (en) | 2010-12-28 | 2012-06-28 | Bayer Animal Health Gmbh | Use of macrocyclic lactones used in controlling endoparasitic filariae and gastrointestinal nematodes, particularly used in controlling heartworm |
SG10202103403SA (en) * | 2015-05-20 | 2021-05-28 | Boehringer Ingelheim Animal Health Usa Inc | Anthelmintic depsipeptide compounds |
SG11201805368YA (en) | 2015-12-28 | 2018-07-30 | Merial Inc | Anthelmintic depsipeptide compounds |
EP3541789A1 (en) | 2016-11-16 | 2019-09-25 | Boehringer Ingelheim Animal Health USA Inc. | Anthelmintic depsipeptide compounds |
NZ769696A (en) * | 2018-05-10 | 2023-12-22 | Zoetis Services Llc | Endoparasitic depsipeptides |
Family Cites Families (5)
Publication number | Priority date | Publication date | Assignee | Title |
---|---|---|---|---|
DK0634408T3 (en) * | 1992-03-17 | 2002-04-22 | Fujisawa Pharmaceutical Co | Depsipeptide derivatives, preparation and use thereof |
WO1994019334A1 (en) * | 1993-02-19 | 1994-09-01 | Meiji Seika Kaisha, Ltd. | Pf1022 derivative, cyclic depsipeptide |
DE4317457A1 (en) * | 1993-05-26 | 1994-12-01 | Bayer Ag | Octacyclodepsipeptides with endoparasiticidal activity |
WO1997011064A1 (en) * | 1995-09-22 | 1997-03-27 | Meiji Seika Kaisha, Ltd. | Novel cyclic depsipeptide pf1022 derivatives |
DE19545639A1 (en) * | 1995-12-07 | 1997-06-12 | Bayer Ag | Process for the preparation of substituted aryl lactic acid-containing cyclodepsipeptides with 24 ring atoms |
-
1998
- 1998-03-17 DE DE19811559A patent/DE19811559A1/en not_active Withdrawn
-
1999
- 1999-03-04 CA CA002323628A patent/CA2323628A1/en not_active Abandoned
- 1999-03-04 CN CN99804115A patent/CN1293664A/en active Pending
- 1999-03-04 AU AU31438/99A patent/AU3143899A/en not_active Abandoned
- 1999-03-04 BR BR9908861-4A patent/BR9908861A/en not_active IP Right Cessation
- 1999-03-04 EP EP99913226A patent/EP1064272A1/en not_active Withdrawn
- 1999-03-04 PL PL99342948A patent/PL342948A1/en unknown
- 1999-03-04 JP JP2000536703A patent/JP2002506857A/en active Pending
- 1999-03-04 WO PCT/EP1999/001407 patent/WO1999047506A1/en not_active Application Discontinuation
- 1999-03-04 KR KR1020007009600A patent/KR20010041450A/en not_active Application Discontinuation
Also Published As
Publication number | Publication date |
---|---|
AU3143899A (en) | 1999-10-11 |
CN1293664A (en) | 2001-05-02 |
DE19811559A1 (en) | 1999-09-23 |
EP1064272A1 (en) | 2001-01-03 |
WO1999047506A1 (en) | 1999-09-23 |
PL342948A1 (en) | 2001-07-16 |
KR20010041450A (en) | 2001-05-25 |
JP2002506857A (en) | 2002-03-05 |
CA2323628A1 (en) | 1999-09-23 |
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Legal Events
Date | Code | Title | Description |
---|---|---|---|
B08F | Application fees: dismissal - article 86 of industrial property law |
Free format text: REFERENTA A 5O, 6O, 7O E 8O ANUIDADES. |
|
B08K | Lapse as no evidence of payment of the annual fee has been furnished to inpi (acc. art. 87) |
Free format text: REFERENTE AO DESPACHO 8.6 PUBLICADO NA RPI 1911 DE 21/08/2007. |